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19 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Synthesis and alpha 2-adrenoceptor effects of substituted catecholimidazoline and catecholimidazole analogues in human platelets.EBI
Ohio State University
Synthesis and evaluation of trimetoquinol derivatives: novel thromboxane A2/prostaglandin H2 antagonists with diminished beta-adrenergic agonist activity.EBI
Ohio State University
Synthesis of halogenated trimetoquinol derivatives and evaluation of their beta-agonist and thromboxane A2 (TXA2) antagonist activities.EBI
Ohio State University
A structure-activity relationship study of benzylic modifications of 4-[1-(1-naphthyl)ethyl]-1H-imidazoles on alpha 1- and alpha 2-adrenergic receptors.EBI
Ohio State University
DNA polymerase and topoisomerase II inhibitors from Psoralea corylifolia.EBI
Ohio State University
Isotope edited NMR studies of glycosidases: design and synthesis of a novel glycosidase inhibitor.EBI
Ohio State University
H-phosphonate derivatives as novel peptide deformylase inhibitors.EBI
Ohio State University
Binding of fluorescent and spin-labeled C-terminal hirudin analogs to thrombin.EBI
Ohio State University
Synthesis, structure elucidation, and biochemical evaluation of 7 alpha- and 7 beta-arylaliphatic-substituted androst-4-ene-3,17-diones as inhibitors of aromatase.EBI
Ohio State University
Synthesis and biological evaluation of 4-(hydroxyalkyl)estradiols and related compounds.EBI
Ohio State University
2-(Hydroxyalkyl)estradiols: synthesis and biological evaluation.EBI
Ohio State University
Medetomidine analogs as alpha 2-adrenergic ligands. 2. Design, synthesis, and biological activity of conformationally restricted naphthalene derivatives of medetomidine.EBI
Ohio State University
Synthesis and D2 dopaminergic activity of pyrrolidinium, tetrahydrothiophenium, and tetrahydrothiophene analogues of sulpiride.EBI
Ohio State University
Synthesis and biochemical studies of 7-substituted 4,6-androstadiene-3,17-diones as aromatase inhibitors.EBI
Ohio State University
Selective irreversible inhibitors of aldose reductase.EBI
Ohio State University
Benzothiophene derivatives and compositions thereof as selective estrogen receptor degradersBDB
Novartis
Non-peptide macrocyclic histone deacetylase inhibitors.BDB
Georgia Institute of Technology
Inhibitors of protein kinase C. 1. 2,3-Bisarylmaleimides.BDB
Roche Products
2-Sulfonyl-4-chloroanilino moiety: a potent pharmacophore for the anti-human immunodeficiency virus type 1 activity of pyrrolyl aryl sulfones.BDB
Universita Di Roma