20 articles for thisTarget
The following articles (labelled with PubMed ID or TBD) are for your review
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Article Title
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Preparation and Evaluation of Radiolabeled Antibody Recruiting Small Molecules That Target Prostate-Specific Membrane Antigen for Combined Radiotherapy and Immunotherapy.
Mcmaster University
Discovery of a new class of cinnamyl-triazole as potent and selective inhibitors of aromatase (cytochrome P450 19A1).
Mcmaster University
Investigation of aryl halides as ketone bioisosteres: refinement of potent and selective inhibitors of human cytochrome P450 19A1 (aromatase).
Mcmaster University
Structural-functional studies of Burkholderia cenocepacia D-glycero-ß-D-manno-heptose 7-phosphate kinase (HldA) and characterization of inhibitors with antibiotic adjuvant and antivirulence properties.
Mcmaster University
Human cytochrome P450 liability studies of trans-dihydronarciclasine: a readily available, potent, and selective cancer cell growth inhibitor.
Mcmaster University
Inhibitors of bacterial cystathionine beta-lyase: leads for new antimicrobial agents and probes of enzyme structure and function.
Mcmaster University
High throughput screening identifies novel inhibitors of Escherichia coli dihydrofolate reductase that are competitive with dihydrofolate.
Mcmaster University
Discovery of a novel class of aldol-derived 1,2,3-triazoles: potent and selective inhibitors of human cytochrome P450 19A1 (aromatase).
Mcmaster University
Structure-activity studies on acetylcholinesterase inhibition in the lycorine series of Amaryllidaceae alkaloids.
Mcmaster University
Potent and selective inhibition of human cytochrome P450 3A4 by seco-pancratistatin structural analogs.
Mcmaster University
Structure-activity studies on seco-pancratistatin analogs: potent inhibitors of human cytochrome P450 3A4.
Mcmaster University
Selective cytochrome P450 3A4 inhibitory activity of Amaryllidaceae alkaloids.
Mcmaster University
Identification of small molecule chemical inhibitors of the collagen-specific chaperone Hsp47.
Mcmaster University
Synthesis of α-methylstilbenes using an aqueous Wittig methodology and application toward the development of potent human aromatase inhibitors.
Mcmaster University
High-throughput screening identifies novel inhibitors of the acetyltransferase activity of Escherichia coli GlmU.
Mcmaster University
Chemical genomics in Escherichia coli identifies an inhibitor of bacterial lipoprotein targeting.
Mcmaster University
Pyrazolonaphthyridinone derivatives as MetAP2 inhibitors (methionine aminopeptidase type-2)
Sanofi