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Design, synthesis, and evaluation of new endomorphin analogs with enhanced central antinociception after peripheral administration.

Lanzhou University

Synthesis and biological evaluation of 2,4-diaminopyrimidines as selective Aurora A kinase inhibitors.

Lanzhou University

Synthesis of xanthohumol analogues and discovery of potent thioredoxin reductase inhibitor as potential anticancer agent.

Lanzhou University

Ingol-type diterpenes from Euphorbia antiquorum with mouse 11ß-hydroxysteroid dehydrogenase type 1 inhibition activity.

Lanzhou University

Dithiaarsanes induce oxidative stress-mediated apoptosis in HL-60 cells by selectively targeting thioredoxin reductase.

Lanzhou University

Design, synthesis, and pharmacological characterization of novel endomorphin-1 analogues as extremely potentµ-opioid agonists.

Lanzhou University

Molecular modeling studies of vascular endothelial growth factor receptor tyrosine kinase inhibitors using QSAR and docking.

Lanzhou University

A novel quantitative structure-activity relationship method to predict the affinities of MT3 melatonin binding site.

Lanzhou University

A new class of highly potent and selective endomorphin-1 analogues containinga-methylene-ß-aminopropanoic acids (map).

Lanzhou University

Molecular modeling studies to predict the possible binding modes of endomorphin analogs in mu opioid receptor.

Lanzhou University

Structure-activity study of endomorphin-2 analogs with C-terminal modifications by NMR spectroscopy and molecular modeling.

Lanzhou University

Endomorphin-1 analogs with enhanced metabolic stability and systemic analgesic activity: design, synthesis, and pharmacological characterization.

Lanzhou University

Discovery of novel VEGFR-2-PROTAC degraders based on the localization of lysine residues via recruiting VHL for the treatment of gastric cancer.

Lanzhou University

Emerging trends of receptor-mediated tumor targeting peptides: A review with perspective from molecular imaging modalities.

Lanzhou University

Design, synthesis, and biological evaluation of quinoxalinone derivatives as potent BRD4 inhibitors.

Lanzhou University

Recent advance on carbamate-based cholinesterase inhibitors as potential multifunctional agents against Alzheimer's disease.

Lanzhou University

Opioid receptor binding and antinociceptive activity of the analogues of endomorphin-2 and morphiceptin with phenylalanine mimics in the position 3 or 4.

Lanzhou University

-2-(Phenylamino) Benzamide Derivatives as Dual Inhibitors of COX-2 and Topo I Deter Gastrointestinal Cancers via Targeting Inflammation and Tumor Progression.

Lanzhou University

Discovery of dual inhibitors of topoisomerase I and Cyclooxygenase-2 for colon cancer therapy.

Lanzhou University

Structure-activity relationship of the novel bivalent and C-terminal modified analogues of endomorphin-2.

Lanzhou University

Design, synthesis and biological evaluation of novel pyrazinone derivatives as PI3K/HDAC dual inhibitors.

Lanzhou University

Design, synthesis, and biological evaluation of carbamate derivatives of N-salicyloyl tryptamine as multifunctional agents for the treatment of Alzheimer's disease.

Lanzhou University

Development of Multifunctional and Orally Active Cyclic Peptide Agonists of Opioid/Neuropeptide FF Receptors that Produce Potent, Long-Lasting, and Peripherally Restricted Antinociception with Diminished Side Effects.

Lanzhou University

N-2-(phenylamino) benzamide derivatives as novel anti-glioblastoma agents: Synthesis and biological evaluation.

Lanzhou University

Design, synthesis and biological evaluation of N-anthraniloyl tryptamine derivatives as pleiotropic molecules for the therapy of malignant glioma.

Lanzhou University

Design, synthesis and biological evaluation of novel 2-(4-(1H-indazol-6-yl)-1H-pyrazol-1-yl)acetamide derivatives as potent VEGFR-2 inhibitors.

Lanzhou University

Discovery of pyrazole N-aryl sulfonate: A novel and highly potent cyclooxygenase-2 (COX-2) selective inhibitors.

Lanzhou University

Improving NK1R-targeted gene delivery of stearyl-antimicrobial peptide CAMEL by conjugating it with substance P.

Lanzhou University

Design and synthesis of 1,3-benzothiazinone derivatives as potential anti-inflammatory agents.

Lanzhou University

Structure-Based Optimization of Multifunctional Agonists for Opioid and Neuropeptide FF Receptors with Potent Nontolerance Forming Analgesic Activities.

Lanzhou University

Design, synthesis and biological evaluation of indole-2-one derivatives as potent BRD4 inhibitors.

Lanzhou University

Synthesis and Biological Characterization of Cyclic Disulfide-Containing Peptide Analogs of the Multifunctional Opioid/Neuropeptide FF Receptor Agonists That Produce Long-Lasting and Nontolerant Antinociception.

Lanzhou University

Design, synthesis and bioactivity study of N-salicyloyl tryptamine derivatives as multifunctional agents for the treatment of neuroinflammation.

Lanzhou University

The synthesis and anti-tumour properties of novel 4-substituted phthalazinones as Aurora B kinase inhibitors.

Lanzhou University

Design, synthesis, and biological activity of new endomorphin analogs with multi-site modifications.

Lanzhou University

Synthesis, biological evaluation and molecular modeling study of 2-amino-3,5-disubstituted-pyrazines as Aurora kinases inhibitors.

Lanzhou University

Discovery of novel 2,4-disubstituted pyrimidines as Aurora kinase inhibitors.

Lanzhou University

Synthesis and biological evaluation of nitroxide labeled pyrimidines as Aurora kinase inhibitors.

Lanzhou University

Discovery of two novel branched peptidomimetics containing endomorphin-2 and RF9 pharmacophores: Synthesis and neuropharmacological evaluation.

Lanzhou University

Synthesis and identification of 2,4-bisanilinopyrimidines bearing 2,2,6,6-tetramethylpiperidine-N-oxyl as potential Aurora A inhibitors.

Lanzhou University

CoMFA and CoMSIA 3D-QSAR studies on quionolone caroxylic acid derivatives inhibitors of HIV-1 integrase.

Lanzhou University

QSAR models for 2-amino-6-arylsulfonylbenzonitriles and congeners HIV-1 reverse transcriptase inhibitors based on linear and nonlinear regression methods.

Lanzhou University

QSAR study of neuraminidase inhibitors based on heuristic method and radial basis function network.

Lanzhou University

Synthesis and biological evaluation of 2,4-disubstituted phthalazinones as Aurora kinase inhibitors.

Lanzhou University

Bioactive Glycosides from the Twigs of Litsea cubeba.

Lanzhou University

Synthesis of naphthazarin derivatives and identification of novel thioredoxin reductase inhibitor as potential anticancer agent.

Lanzhou University