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14 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Discovery of novel 2,5-dioxoimidazolidine-based P2X(7) receptor antagonists as constrained analogues of KN62.EBI
Gwangju Institute of Science and Technology (Gist)
Design and synthesis of potent and selective P2X3 receptor antagonists derived from PPADS as potential pain modulators.EBI
Gwangju Institute of Science and Technology (Gist)
Structure-activity relationships and optimization of 3,5-dichloropyridine derivatives as novel P2X(7) receptor antagonists.EBI
Gwangju Institute of Science and Technology (Gist)
Discovery and Binding Mechanism of Pyrazoloisoquinoline-Based Novel β-Arrestin Inverse Agonists of the Kappa-Opioid Receptor.EBI
Gwangju Institute of Science and Technology (GIST)
Discovery of 3-Phenyl Indazole-Based Novel Chemokine-like Receptor 1 Antagonists for the Treatment of Psoriasis.EBI
Gwangju Institute of Science and Technology (GIST)
Interplay among Conformation, Intramolecular Hydrogen Bonds, and Chameleonicity in the Membrane Permeability and Cyclophilin A Binding of Macrocyclic Peptide Cyclosporin O Derivatives.EBI
Gwangju Institute of Science and Technology (Gist)
Synthesis and structure-activity relationship studies of 1,5-isomers of triazole-pyrrolopyrimidine as selective Janus kinase 1 (JAK1) inhibitors.EBI
Gwangju Institute of Science and Technology (Gist)
Discovery of 5-methyl-1H-benzo[d]imidazole derivatives as novel P2X3 Receptor antagonists.EBI
Gwangju Institute of Science and Technology (Gist)
Discovery of Novel Pyrimidine-Based Capsid Assembly Modulators as Potent Anti-HBV Agents.EBI
Gwangju Institute of Science and Technology (Gist)
Potent Suppressive Effects of 1-Piperidinylimidazole Based Novel P2X7 Receptor Antagonists on Cancer Cell Migration and Invasion.EBI
Gwangju Institute of Science and Technology (Gist)
The discovery of 2,5-isomers of triazole-pyrrolopyrimidine as selective Janus kinase 2 (JAK2) inhibitors versus JAK1 and JAK3.EBI
Gwangju Institute of Science and Technology (Gist)
2,3,4-Trihydroxybenzyl-hydrazide analogues as novel potent coxsackievirus B3 3C protease inhibitors.EBI
Gwangju Institute of Science and Technology (Gist)
Structure-activity relationship studies of pyrimidine-2,4-dione derivatives as potent P2X7 receptor antagonists.EBI
Gwangju Institute of Science and Technology (Gist)
Synthesis and structure-activity relationships of quinolinone and quinoline-based P2X7 receptor antagonists and their anti-sphere formation activities in glioblastoma cells.EBI
Gwangju Institute of Science and Technology (Gist)