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14 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
Design and synthesis of selective keto-1,2,4-oxadiazole-based tryptase inhibitors.EBI
Celera Genomics
Keto-1,3,4-oxadiazoles as cathepsin K inhibitors.EBI
Celera Genomics
Development of activity-based probes for trypsin-family serine proteases.EBI
Celera Genomics
Potent 4-amino-5-azaindole factor VIIa inhibitors.EBI
Celera Genomics
Design and synthesis of tetracyclic nonpeptidic biaryl nitrile inhibitors of cathepsin K.EBI
Celera Genomics
Novel, potent, selective, and orally bioavailable human betaII-tryptase inhibitors.EBI
Celera Genomics
Discovery of novel hydroxy pyrazole based factor IXa inhibitor.EBI
Celera Genomics
Factor VIIa inhibitors: a prodrug strategy to improve oral bioavailability.EBI
Celera Genomics
Factor VIIa inhibitors: improved pharmacokinetic parameters.EBI
Celera Genomics
Small molecule inhibitors of plasma kallikrein.EBI
Celera Genomics
Factor VIIa inhibitors: chemical optimization, preclinical pharmacokinetics, pharmacodynamics, and efficacy in an arterial baboon thrombosis model.EBI
Celera Genomics
Design and synthesis of tri-ring P3 benzamide-containing aminonitriles as potent, selective, orally effective inhibitors of cathepsin K.EBI
Celera Genomics
Identification of metabolites of the tryptase inhibitor CRA-9249: observation of a metabolite derived from an unexpected hydroxylation pathway.EBI
Celera Genomics
Aryl, heteroaryl, and heterocycle substituted tetrahydroisoquinolines and use thereofBDB
Albany Molecular Research