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Synthesis and biological evaluation of a water-soluble phosphate prodrug salt and structural analogues of KGP94, a lead inhibitor of cathepsin L.

Baylor University

Design, synthesis, and biological evaluation of water-soluble amino acid prodrug conjugates derived from combretastatin, dihydronaphthalene, and benzosuberene-based parent vascular disrupting agents.

Baylor University

Synthesis and biochemical evaluation of benzoylbenzophenone thiosemicarbazone analogues as potent and selective inhibitors of cathepsin L.

Baylor University

Functionalized benzophenone, thiophene, pyridine, and fluorene thiosemicarbazone derivatives as inhibitors of cathepsin L.

Baylor University

Design, synthesis, and biological evaluation of potent thiosemicarbazone based cathepsin L inhibitors.

Baylor University

Structure Guided Design, Synthesis, and Biological Evaluation of Oxetane-Containing Indole Analogues.

Baylor University

Design, synthesis, and biochemical evaluation of novel cruzain inhibitors with potential application in the treatment of Chagas' disease.

Baylor University

Gemfibrozil derivatives as activators of soluble guanylyl cyclase - A structure-activity study.

Baylor University

Design and Catalyzed Activation of Tak-242 Prodrugs for Localized Inhibition of TLR4-Induced Inflammation.

Baylor University

Structure Guided Design, Synthesis, and Biological Evaluation of Novel Benzosuberene Analogues as Inhibitors of Tubulin Polymerization.

Baylor University

An Amino-Benzosuberene Analogue That Inhibits Tubulin Assembly and Demonstrates Remarkable Cytotoxicity.

Baylor University

Small-molecule inhibitors of cathepsin L incorporating functionalized ring-fused molecular frameworks.

Baylor University

A strategy for dual inhibition of the proteasome and fatty acid synthase with belactosin C-orlistat hybrids.

Baylor University

Substituted pyridinyl-pyrimidines and their use as medicaments

Boehringer Ingelheim International