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14 articles for thisTarget


The following articles (labelled with PubMed ID or TBD) are for your review

PMID
Data
Article Title
Organization
4-Acyl Pyrrole Derivatives Yield Novel Vectors for Designing Inhibitors of the Acetyl-Lysine Recognition Site of BRD4(1).EBI
Albert-Ludwigs-University of Freiburg
Aminothiazoles as Potent and Selective Sirt2 Inhibitors: A Structure-Activity Relationship Study.EBI
Albert-Ludwigs-University of Freiburg
Synthesis and Biological Investigation of Oxazole Hydroxamates as Highly Selective Histone Deacetylase 6 (HDAC6) Inhibitors.EBI
Albert-Ludwigs-University of Freiburg
Discovery of Tricyclic Clerodane Diterpenes as Sarco/Endoplasmic Reticulum Ca(2+)-ATPase Inhibitors and Structure-Activity Relationships.EBI
Albert-Ludwigs-University of Freiburg
Bornyl (3,4,5-trihydroxy)-cinnamate--an optimized human neutrophil elastase inhibitor designed by free energy calculations.EBI
Albert-Ludwigs-University of Freiburg
Structure-activity studies on splitomicin derivatives as sirtuin inhibitors and computational prediction of binding mode.EBI
Albert-Ludwigs-University of Freiburg
A novel arginine methyltransferase inhibitor with cellular activity.EBI
Albert-Ludwigs-University of Freiburg
Target-based approach to inhibitors of histone arginine methyltransferases.EBI
Albert-Ludwigs-University of Freiburg
Acyl derivatives of p-aminosulfonamides and dapsone as new inhibitors of the arginine methyltransferase hPRMT1.EBI
Albert-Ludwigs-University of Freiburg
Synthesis and biological testing of novel pyridoisothiazolones as histone acetyltransferase inhibitors.EBI
Albert-Ludwigs-University of Freiburg
Catechin derivatives from Parapiptadenia rigida with in vitro wound-healing properties.EBI
Albert-Ludwigs-University of Freiburg
Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition.EBI
Albert-Ludwigs-University of Freiburg
Binding structures and potencies of oxidosqualene cyclase inhibitors with the homologous squalene-hopene cyclase.EBI
Albert-Ludwigs-University of Freiburg
New peptidic cysteine protease inhibitors derived from the electrophilic alpha-amino acid aziridine-2,3-dicarboxylic acid.EBI
Albert-Ludwigs-University of Freiburg