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Targets Binding with 57 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
3-hydroxyacyl-[acyl-carrier-protein] dehydratase FabZ
IC50:
20
Other:
22
2
2
2D
3D
TSV
Bcl-2-like protein 1/Bcl2-associated agonist of cell death [103-127,M117N]
IC50:
67
1
9
2D
3D
TSV
Beta-secretase 1 [1-453]
IC50:
56
Other:
1
3
11
2D
3D
TSV
Cellular tumor antigen p53 [16-27]/E3 ubiquitin-protein ligase Mdm2 [23-117]
IC50:
67
1
42
2D
3D
TSV
Chitinase B
Ki:
7
IC50:
58
Kd:
2
11
1
2D
3D
TSV
Gag-Pol polyprotein [600-1027,Y787L]/[600-1155,Y787L]
IC50:
56
Other:
3
4
5
2D
3D
TSV
Isoform 7 of cAMP-specific 3',5'-cyclic phosphodiesterase 4A (PDE4A8)
IC50:
58
1
11
2D
3D
TSV
NAD(+) hydrolase SARM1
Ki:
4
IC50:
64
6
5
2D
3D
TSV
NAD(+) hydrolase SARM1 [50-724]
IC50:
59
1
5
2D
3D
TSV
Nuclear receptor ROR-gamma [258-518]
Kd:
98
2
5
2D
3D
TSV
Phospholipid-transporting ATPase ABCA1
EC50:
57
1
3
2D
3D
TSV
Receptor-type tyrosine-protein phosphatase epsilon
Ki:
11
IC50:
50
16
6
2D
3D
TSV
Synaptic vesicle glycoprotein 2A
Ki:
14
IC50:
55
3
13
2D
3D
TSV
Transcription activator BRG1
Ki:
1
IC50:
37
Kd:
38
27
9
2D
3D
TSV
UDP-glucuronosyltransferase 1A1
Ki:
8
IC50:
76
19
6
2D
3D
TSV
Vasoactive intestinal polypeptide receptor 2
Ki:
144
IC50:
13
EC50:
20
7
8
2D
3D
TSV