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Targets Binding with 22 Compounds
Target Name
Affinity Link(s)
Article(s)
UniProt
Files
1-deoxy-D-xylulose 5-phosphate reductoisomerase, apicoplastic
IC50:
25
2
3
2D
3D
TSV
2-C-methyl-D-erythritol 2,4-cyclodiphosphate synthase
IC50:
5
Kd:
20
Other:
3
5
6
2D
3D
TSV
Acyl-CoA 6-desaturase
IC50:
27
9
12
2D
3D
TSV
Anionic trypsin-2
IC50:
22
1
1
2D
3D
TSV
Basic phospholipase A2 VRV-PL-VIIIa
IC50:
23
2
3
2D
3D
TSV
Bcl-2-like protein 11 [72-87]
IC50:
22
1
20
2D
3D
TSV
Bcl-2-like protein 11 [81-106]
IC50:
22
1
20
2D
3D
TSV
Beta-1,4-galactosyltransferase 1
Ki:
20
IC50:
3
7
13
2D
3D
TSV
Casein kinase I delta/epsilon
IC50:
22
4
5
2D
3D
TSV
Cellular tumor antigen p53 [18-26]/Protein Mdm4 [2-185]
IC50:
22
1
32
2D
3D
TSV
Chymotrypsinogen B2
Ki:
14
IC50:
12
8
3
2D
3D
TSV
Dimer of Gag-Pol polyprotein [514-612]
Ki:
16
IC50:
7
6
2
2D
3D
TSV
Dimer of Receptor-type tyrosine-protein kinase FLT3 [D835V]
Kd:
22
2
6
2D
3D
TSV
Dimer of Receptor-type tyrosine-protein kinase FLT3 [F691L]
Kd:
22
2
6
2D
3D
TSV
DNA repair protein REV1
Ki:
20
IC50:
22
Kd:
22
1
6
2D
3D
TSV
Dopamine receptor D4
Ki:
41
2
2
2D
3D
TSV
Enoyl-[acyl-carrier-protein] reductase [NADH] [T276S]
Ki:
4
IC50:
22
1
1
2D
3D
TSV
Epidermal growth factor receptor [G719C]
IC50:
2
Kd:
21
3
15
2D
3D
TSV
Fatty-acid amide hydrolase 1 [33-574]
IC50:
22
1
3
2D
3D
TSV
Fructose-bisphosphate aldolase class 2
Ki:
38
2
5
2D
3D
TSV
General amino acid permease AGP1
EC50:
23
2
3
2D
3D
TSV
Grp78
IC50:
11
Kd:
14
Koff:
14
ITC:
6
3
6
2D
3D
TSV
Heat sensitive channel TRPV3
IC50:
21
EC50:
17
4
1
2D
3D
TSV
Histone acetyltransferase p300/Myocyte-specific enhancer factor 2D
IC50:
22
1
7
2D
3D
TSV
Histone deacetylase 4 [648-1032]
IC50:
24
1
6
2D
3D
TSV
Holo-[acyl-carrier-protein] synthase
IC50:
22
2
1
2D
3D
TSV
IAG-nucleoside hydrolase
Ki:
23
2
1
2D
3D
TSV
Lysosomal alpha-mannosidase
Ki:
6
IC50:
36
4
7
2D
3D
TSV
Matrix protein 2 [1-96]
IC50:
29
4
5
2D
3D
TSV
Met repressor
Kd:
1
EC50:
22
1
4
2D
3D
TSV
Metallo-beta-lactamase IMP-1
IC50:
22
1
1
2D
3D
TSV
Methionine synthase
IC50:
25
2
8
2D
3D
TSV
Mycothiol S-conjugate amidase
IC50:
32
4
3
2D
3D
TSV
Phospholipase
IC50:
32
1
1
2D
3D
TSV
Phosphopantetheine adenylyltransferase
IC50:
47
2
5
2D
3D
TSV
Probable integral membrane cytochrome D ubiquinol oxidase (Subunit II) CydB (Cytochrome BD-I oxidase subunit II)
IC50:
22
1
5
2D
3D
TSV
Proteasome subunit beta type-6
Ki:
17
IC50:
5
2
5
2D
3D
TSV
Protein Tax-1
IC50:
22
1
1
2D
3D
TSV
Protein tyrosine phosphatase type IVA 1
IC50:
25
6
5
2D
3D
TSV
RAF proto-oncogene serine/threonine-protein kinase [325-648]
IC50:
22
1
6
2D
3D
TSV
Receptor-type tyrosine-protein kinase FLT3 [D835V]
Kd:
22
2
7
2D
3D
TSV
Retinoic acid receptor RXR-alpha [225-462]/Thyroid hormone receptor beta [148-410]
EC50:
22
1
11
2D
3D
TSV
Separin
IC50:
23
1
1
2D
3D
TSV
Shiga toxin subunit A
Ki:
20
IC50:
6
Kd:
1
1
1
2D
3D
TSV
Siderophore-binding protein
Ki:
22
2
1
2D
3D
TSV
Signal transduction protein TRAP
EC50:
44
1
1
2D
3D
TSV
Spindlin-1
IC50:
28
Kd:
19
EC50:
1
2
7
2D
3D
TSV
Transcription factor 4
Ki:
3
IC50:
19
Kd:
2
8
25
2D
3D
TSV
Transcription initiation factor IIA subunit 1
Ki:
24
1
3
2D
3D
TSV
tRNA (cytosine(38)-C(5))-methyltransferase
IC50:
14
Kd:
29
2
8
2D
3D
TSV
Trypsin-3
Ki:
17
IC50:
5
5
12
2D
3D
TSV
TSC22 domain family protein 3
IC50:
22
1
10
2D
3D
TSV
Tyrosine-protein phosphatase non-receptor type 6 [205-595]
IC50:
22
1
6
2D
3D
TSV
Virulence factor transcriptional regulator MvfR
IC50:
5
Kd:
18
EC50:
8
2
3
2D
3D
TSV
Zn finger protein
Ki:
22
1
1
2D
3D
TSV