Compile Data Set for Download or QSAR
Report error Found 75 of affinity data for UniProtKB/TrEMBL: T1QYY3
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM330048(US9663528, 42 | (2R,5S,13aR)-8-hydroxy-7,9-dioxo-N...)
Affinity DataEC50:  3.10nMAssay Description:Inhibition of HIV-1 integrase G140S/Q148K double mutantMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492067(CHEMBL2396766)
Affinity DataIC50: 430nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492076(CHEMBL2396853)
Affinity DataIC50: 460nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492079(CHEMBL2396852)
Affinity DataIC50: 570nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492072(CHEMBL2396845)
Affinity DataIC50: 680nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492071(CHEMBL2396846)
Affinity DataIC50: 720nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492078(CHEMBL2396847)
Affinity DataIC50: 760nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492080(CHEMBL2396848)
Affinity DataIC50: 850nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492081(CHEMBL2396844)
Affinity DataIC50: 910nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492068(CHEMBL3037906)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492069(CHEMBL2396850)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492070(CHEMBL2396849)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492073(CHEMBL2396843)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492074(CHEMBL2396767)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492077(CHEMBL2396768)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50125577(AGERIVDIIATDIQ-CONH2 | CHEMBL265887)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50492075(CHEMBL2396769)
Affinity DataIC50: 3.75E+3nMAssay Description:Inhibition of HIV1 3'-processing activity of integrase F185K/C280S double mutant expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50495689(CHEMBL3116306)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase E138K mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50495689(CHEMBL3116306)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase G140S mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50495689(CHEMBL3116306)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase N155H mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50495689(CHEMBL3116306)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of HIV-1 integrase E92Q mutant expressed in Escherichia coli using [32P]-labeled U5B/U5A DNA as substrate assessed as inhibition of 3'-pro...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480005(CHEMBL462081)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479999(CHEMBL449723)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480011(CHEMBL458653)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479991(CHEMBL444733)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479991(CHEMBL444733)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480005(CHEMBL462081)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480011(CHEMBL458653)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480011(CHEMBL458653)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480005(CHEMBL462081)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479999(CHEMBL449723)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480009(CHEMBL510036)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480001(CHEMBL457554)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479999(CHEMBL449723)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479991(CHEMBL444733)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480010(CHEMBL457106)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480010(CHEMBL457106)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479998(CHEMBL456024)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480009(CHEMBL510036)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479990(CHEMBL512918)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480003(CHEMBL458652)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480003(CHEMBL458652)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480001(CHEMBL457554)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480001(CHEMBL457554)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479998(CHEMBL456024)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV1 integrase H114A mutant 3'-end processing activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479998(CHEMBL456024)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50479990(CHEMBL512918)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480010(CHEMBL457106)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480003(CHEMBL458652)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
Fudan University

Curated by ChEMBL
LigandPNGBDBM50480009(CHEMBL510036)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of HIV1 integrase Y99S mutant strand transfer activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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