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Report error Found 186 of affinity data for UniProtKB/TrEMBL: Q9Y2T5
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022147(CHEMBL3299117)
Affinity DataEC50:  646nMAssay Description:Agonist activity at GPR52 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022151(CHEMBL3299118)
Affinity DataEC50:  347nMAssay Description:Agonist activity at GPR52 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022152(CHEMBL3299018)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022153(CHEMBL3299119)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022156(CHEMBL3299120)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022157(CHEMBL3299121)
Affinity DataEC50:  38nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022158(CHEMBL3299122)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022159(CHEMBL3299123)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022162(CHEMBL3299124)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022164(CHEMBL3299125)
Affinity DataEC50:  646nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022165(CHEMBL3297807)
Affinity DataEC50:  209nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022166(CHEMBL3297808)
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022169(CHEMBL3297809)
Affinity DataEC50:  81nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022170(CHEMBL3297810)
Affinity DataEC50:  55nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022189(CHEMBL3297811)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022190(CHEMBL3298233)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50022254(CHEMBL3298234)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as cAMP production after 30 mins by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252092(CHEMBL4082756)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252099(CHEMBL4087237)
Affinity DataEC50:  23nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252102(CHEMBL4059658)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252136(CHEMBL4064577)
Affinity DataEC50:  210nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252137(CHEMBL4074656)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252138(CHEMBL4095110)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252139(CHEMBL4091718)
Affinity DataEC50:  690nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252140(CHEMBL4081439)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252141(CHEMBL4099457)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252151(CHEMBL4073584)
Affinity DataEC50:  110nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252152(CHEMBL4062229)
Affinity DataEC50:  170nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252186(CHEMBL4072782)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252187(CHEMBL4099668)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252188(CHEMBL4098770)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252189(CHEMBL4091030)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252190(CHEMBL4101517)
Affinity DataEC50:  59nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252191(CHEMBL4075971)
Affinity DataEC50:  25nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252192(CHEMBL4070849)
Affinity DataEC50:  260nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252212(CHEMBL4100408)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252213(CHEMBL4083957)
Affinity DataEC50:  380nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50252214(CHEMBL4080724)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460255(CHEMBL4226295)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460256(CHEMBL4226751)
Affinity DataEC50:  146nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460257(CHEMBL4228912)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460258(CHEMBL4228734)
Affinity DataEC50:  45nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460259(CHEMBL4226750)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460260(CHEMBL4226225)
Affinity DataEC50:  87nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460261(CHEMBL4226253)
Affinity DataEC50:  62nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460262(CHEMBL4229063)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460263(CHEMBL4226695)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50460264(CHEMBL4229128)
Affinity DataEC50:  9.60nMAssay Description:Agonist activity at human GPR52 expressed in CHO cells assessed as increase in cAMP level after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50554904(CHEMBL4761550 | US20240059655, Compound PW0955)
Affinity DataEC50:  673nMAssay Description:Agonist activity at human GPR52 expressed in HEK293 cells assessed as increase in cAMP levels incubated for 15 mins by Glosensor cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetG-protein coupled receptor 52(Human)
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50554905(CHEMBL4741318 | US20240059655, Compound PW0948)
Affinity DataEC50:  431nMAssay Description:Agonist activity at human GPR52 expressed in HEK293 cells assessed as increase in cAMP levels incubated for 15 mins by Glosensor cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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