Compile Data Set for Download or QSAR
Report error Found 27 for UniProtKB: Q9UBS0
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.726nMAssay Description:Inhibition of human p70S6Kb using KKRNRTLTK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human p70S6Kb using KKRNRTLTK as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168247(2,3-Di-thiophen-2-yl-benzo[g]quinoxaline-7-carboxy...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168248({5-[3-(4-Carboxymethyl-thiophen-2-yl)-benzo[g]quin...)
Affinity DataIC50: 640nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168244(4-(5-{3-[5-(3-Carboxy-propyl)-thiophen-2-yl]-benzo...)
Affinity DataIC50: 820nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168242(3-(5-{3-[5-(2-Carboxy-ethyl)-thiophen-2-yl]-benzo[...)
Affinity DataIC50: 870nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168241(6,7-Di-thiophen-2-yl-2,3-dihydro-1,4-dioxa-5,8-dia...)
Affinity DataIC50: 950nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-1/beta-2(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50126732(2-(2,6-Dichloro-phenylamino)-7-(3-diethylamino-pro...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of Ribosomal protein S6 kinase (P70S6K kinase)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50532181(CHEMBL4474690)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human full-length N-terminal His-tagged p70S6K expressed in baculovirus infected Sf21 insect cells using CKRRRLASLR as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50460772(CHEMBL4225923)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of S6K (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-1/beta-2(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50192071((13R,15S)-13-methyl-16-oxa-8,9,12,22,24-pentaazahe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of p706SKMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-1/beta-2(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196392(3-hydroxy-N-1-hydroxypropan-2-yl)-5-4-phenylamino)...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of p70 S6 kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168239(7,8-Dimethoxy-2,3-di-thiophen-2-yl-pyrazino[2,3-b]...)
Affinity DataIC50: 1.14E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168236({5-[3-(5-Carboxymethyl-thiophen-2-yl)-benzo[g]quin...)
Affinity DataIC50: 1.28E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168235(2,3-Di-thiophen-2-yl-benzo[g]quinoxaline | CHEMBL3...)
Affinity DataIC50: 1.36E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50583520(CHEMBL5094006)
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of human recombinant P70S6Kbeta expressed in Sf9 insect cells using [KKRNRTLTK] as substrate in presence of [33P]-ATP by radiometric hotsp...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-1/beta-2(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50194024(3-hydroxy-N-1-hydroxypropan-2-yl)-5-4-phenoxypheny...)
Affinity DataIC50: 2.62E+3nMAssay Description:Inhibition of p70 S6 kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168243(3-(5-{3-[5-(2-Methoxycarbonyl-ethyl)-thiophen-2-yl...)
Affinity DataIC50: 6.13E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168246(2,3-Di-thiophen-2-yl-quinoxaline-6,7-diol | CHEMBL...)
Affinity DataIC50: 9.61E+3nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168249(5-[3-(5-carboxythien-2-yl)benzo[g]quinoxalin-2-yl]...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50135286(CHEMBL3745885)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human RPS6KB2 using [KKRNRTLTK] as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-1/beta-2(Human)
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50169959([3H-Benzothiazol-(2Z)-ylidene]-[2-(2-pyridin-3-yl-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of p70S6KMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168250({5-[3-(4-Methoxycarbonylmethyl-thiophen-2-yl)-benz...)
Affinity DataIC50: 1.18E+4nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168238(6,7-Dimethoxy-2,3-di-thiophen-2-yl-quinoxaline | C...)
Affinity DataIC50: 1.63E+4nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168237(6,7-Di-thiophen-2-yl-2,3-dihydro-1,4-dioxa-5,8-dia...)
Affinity DataIC50: 2.34E+4nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRibosomal protein S6 kinase beta-2(Human)
Beijing Normal University

Curated by ChEMBL
LigandPNGBDBM50168240(6,7-Di-thiophen-2-yl-[1,3]dioxolo[4,5-g]quinoxalin...)
Affinity DataIC50: 2.85E+4nMAssay Description:In vitro inhibition of SR protein kinase 1 by compound dissolved in 100% DMSO using 5''-[gamma-33P]-triphosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50463479(CHEMBL4249925)
Affinity DataKi:  100nMAssay Description:Inhibition of p70S6K (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed