Compile Data Set for Download or QSAR
Report error Found 133 of affinity data for UniProtKB/TrEMBL: Q9JHG3
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506018(CHEMBL4435973)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at rat APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HT...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506019(CHEMBL4473347)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at rat APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HT...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  0.0620nMAssay Description:Agonist activity at rat APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HT...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50506018(CHEMBL4435973)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at rat APJ-R expressed in HEK293 cells assessed as inhibition of forskolin- stimulated cAMP accumulation incubated for 30 mins by HT...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50556824(CHEMBL4746142)
Affinity DataEC50:  8.80nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50556825(CHEMBL4787784)
Affinity DataEC50:  8nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50556826(CHEMBL4745863)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50556827(CHEMBL4748838)
Affinity DataEC50:  7.80nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50556828(CHEMBL4798771)
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546706(CHEMBL4797693)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546707(CHEMBL4778333)
Affinity DataEC50:  2nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546708(CHEMBL4791658)
Affinity DataEC50:  0.920nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546709(CHEMBL4753509)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546710(CHEMBL4796794)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546711(CHEMBL4751429)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546712(CHEMBL4748581)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546713(CHEMBL4752419)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546714(CHEMBL4799770)
Affinity DataEC50:  6.20nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546715(CHEMBL4791768)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546716(CHEMBL4742782)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546717(CHEMBL4781615)
Affinity DataEC50:  4nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546718(CHEMBL4743536)
Affinity DataEC50:  7.40nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546719(CHEMBL4746298)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546720(CHEMBL4740291)
Affinity DataEC50:  0.490nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546721(CHEMBL4756792)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546722(CHEMBL4749038)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546723(CHEMBL4785561)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546724(CHEMBL4787872)
Affinity DataEC50:  9.30nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546725(CHEMBL4744747)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546726(CHEMBL4796441)
Affinity DataEC50:  56nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50546727(CHEMBL4743846)
Affinity DataEC50:  117nMAssay Description:Agonist activity at rat APJ receptor stably expressed in CHO cell membranes in presence of [35S]GTPgammaS by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570414(CHEMBL4861181)
Affinity DataEC50:  980nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570415(CHEMBL4873340)
Affinity DataEC50:  430nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570416(CHEMBL4871403)
Affinity DataEC50:  120nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570417(CHEMBL4858384)
Affinity DataEC50:  31nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570418(CHEMBL4857233)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570419(CHEMBL4861906)
Affinity DataEC50:  7.30nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570420(CHEMBL4861053)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570421(CHEMBL4878068)
Affinity DataEC50:  450nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570422(CHEMBL4852391)
Affinity DataEC50:  15nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570423(CHEMBL4846150)
Affinity DataEC50:  0.510nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570424(CHEMBL4860991)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570425(CHEMBL4866313)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50570426(CHEMBL4876050)
Affinity DataEC50:  0.580nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50567169(CHEMBL4873876)
Affinity DataEC50:  0.0240nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50014619(CHEMBL3184840)
Affinity DataEC50:  0.0600nMAssay Description:Agonist activity at rat APJ receptor expressed in human HEK293 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 1 hr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM422160(N-[4-(4-{[2-butyl-1- (2,6-dimethoxyphenyl)- 6-hydr...)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at rat APJ receptor assessed as effect on cAMP accumulation by cAMP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50567159(CHEMBL4874447)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at rat APJ receptor assessed as effect on cAMP accumulation by cAMP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetApelin receptor(Rat)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50567160(CHEMBL4873216)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at rat APJ receptor assessed as effect on cAMP accumulation by cAMP-Glo assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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