Compile Data Set for Download or QSAR
Report error Found 925 of affinity data for UniProtKB/TrEMBL: Q92633
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148349((3-Octadec-9-enoylamino-propionyl)-phosphonothioic...)
Affinity DataEC50:  40nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148350([3-((Z)-Octadec-9-enoylamino)-thiopropionyl]-phosp...)
Affinity DataEC50:  318nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  17nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148352([1-Hydroxy-3-((Z)-octadec-9-enoylamino)-propyl]-ph...)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 receptor using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50074700(Phosphoric acid mono-[2-((Z)-octadec-9-enoylamino)...)
Affinity DataEC50:  197nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148353((1-Hydroxy-3-octadec-9-enoylamino-1-phosphono-prop...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148351([3-((Z)-Octadec-9-enoylamino)-propionyl]-phosphoni...)
Affinity DataEC50:  221nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148354([1-Fluoro-3-((Z)-octadec-9-enoylamino)-propyl]-pho...)
Affinity DataEC50: >5.00E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148355([3-((Z)-Octadec-9-enoylamino)-propyl]-phosphonic a...)
Affinity DataEC50:  1.95E+3nMAssay Description:Agonistic activity against lysophosphatidic acid receptor 1 using [35S]GTP-gamma-S as radioligand tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  350nMAssay Description:Agonist activity at human LPA1 expressed in LPA1xLPA2 double knockout mouse MEF cells up to 10 uM by Fura-2AM dye based Ca2+ mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170844(Thiophosphoric acid (E)-octadec-9-enyl ester | CHE...)
Affinity DataEC50:  193nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50170848(2-Hexadecanoylamino-3-phosphonooxy-propionic acid ...)
Affinity DataEC50:  1.85E+3nMAssay Description:Inhibition of LPA-induced calcium transients in RH7777 rat hepatoma cells expressing LPA1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50176390((R)-O-2,3-bis(octyloxy)propyl O,O-dihydrogen phosp...)
Affinity DataEC50:  695nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50176400((R)-2,3-bis(octyloxy)propyl dihydrogen phosphate |...)
Affinity DataEC50:  3.26E+3nMAssay Description:Activity at LPA1 receptor transfected RH7777 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50193516(1,1-difluoro-3(S)-hydroxyl-4-oleoyloxylbutane 1,3-...)
Affinity DataEC50: >1.94E+3nMAssay Description:Activity at human LPA1 receptor expressed in RH7777 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50271700(4-(4-(ethoxycarbonyl)styryl)benzenesulfonic acid |...)
Affinity DataEC50: >1.23E+4nMAssay Description:Agonist activity at LPA1 receptor expressed in rat RH7777 cells assessed as LPA-induced intracellular calcium responseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  31nMAssay Description:Agonist activity at LPA1 expressed in human chem1 cells assessed as intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430006(CHEMBL2335048)
Affinity DataEC50:  8.40nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50381022(CHEMBL2017139)
Affinity DataEC50:  17nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430007(CHEMBL2335051)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430008(CHEMBL2335050)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430009(CHEMBL2335049)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430010(CHEMBL2335047)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430011(CHEMBL153043)
Affinity DataEC50:  24nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430012(CHEMBL357053)
Affinity DataEC50:  15nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50430013(CHEMBL364797)
Affinity DataEC50:  71nMAssay Description:Agonist activity at human LPA1 receptor transfected in HEK293 cells after 1 hr by TGFalpha shedding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50233165(CHEMBL1222042)
Affinity DataEC50:  80nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) expressed in rat RH7777 cells assessed as increase in intracellular calcium level measured every 3...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  2.30nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 0.5 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50195695(CHEMBL3941037)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  0.740nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  0.740nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at room temperature by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50195695(CHEMBL3941037)
Affinity DataKd:  8.10nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 0.5 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  1.30nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50195695(CHEMBL3941037)
Affinity DataKd:  6nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  0.490nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50195695(CHEMBL3941037)
Affinity DataKd:  10nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 4 hrs by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  0.340nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at 37 degC by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50285779(CHEMBL4165205)
Affinity DataKd:  23nMAssay Description:Binding affinity to recombinant human LPA1 expressed in CHO cell membranes measured after 2 hrs at 4 degC by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148351([3-((Z)-Octadec-9-enoylamino)-propionyl]-phosphoni...)
Affinity DataEC50:  221nMAssay Description:Agonist activity at LPA1R (unknown origin) by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50539029(CHEMBL4646443)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at recombinant human full-length LPA1 receptor expressed in dhfr- deficient CHO cells assessed as increase in intracellular calcium ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50539030(CHEMBL4647245)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50539031(CHEMBL4643262)
Affinity DataEC50:  450nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50539032(CHEMBL4633208)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50539033(CHEMBL4632820)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50148348(lysophosphatidic acid | 1-oleoyl lysophosphatidic ...)
Affinity DataEC50:  830nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50539034(CHEMBL4642952)
Affinity DataEC50:  240nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50539035(CHEMBL4642688)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLysophosphatidic acid receptor 1(Human)
Oxford University

Curated by ChEMBL
LigandPNGBDBM50539036(CHEMBL4636453)
Affinity DataEC50:  500nMAssay Description:Agonist activity at LPA1 receptor (unknown origin) stably expressed in rat RH7777 cells assessed as increase in intracellular calcium level by Fluo-4...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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