Compile Data Set for Download or QSAR
Report error Found 128 of affinity data for UniProtKB/TrEMBL: Q92551
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605476(CHEMBL5190343)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inhibition of [3H]-InsP6 phosphorylation m...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605488(CHEMBL5169462)
Affinity DataIC50: 26nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605484(CHEMBL5181623)
Affinity DataIC50: 27nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605510(CHEMBL5203174)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant full length human IP6K1 assessed as inorganic phosphate release measured after 30 mins by ADP-Glo Max assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605476(CHEMBL5190343)
Affinity DataIC50: 57nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605508(CHEMBL5200214)
Affinity DataIC50: 78nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605505(CHEMBL5184940)
Affinity DataIC50: 81nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605509(CHEMBL5204881)
Affinity DataIC50: 84nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605491(CHEMBL5186210)
Affinity DataIC50: 110nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605482(CHEMBL5201056)
Affinity DataIC50: 130nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605483(CHEMBL5184960)
Affinity DataIC50: 130nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605485(CHEMBL5190846)
Affinity DataIC50: 160nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605489(CHEMBL5201078)
Affinity DataIC50: 170nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605506(CHEMBL5196483)
Affinity DataIC50: 170nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605498(CHEMBL5197626)
Affinity DataIC50: 190nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605490(CHEMBL5175579)
Affinity DataIC50: 240nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605502(CHEMBL5186729)
Affinity DataIC50: 280nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605497(CHEMBL5188320)
Affinity DataIC50: 320nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605496(CHEMBL5198845)
Affinity DataIC50: 370nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605494(CHEMBL5192487)
Affinity DataIC50: 430nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605495(CHEMBL5206215)
Affinity DataIC50: 430nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605492(CHEMBL5185725)
Affinity DataIC50: 450nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634436(CHEMBL5431012)
Affinity DataIC50: 510nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634439(CHEMBL5430471)
Affinity DataIC50: 595nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605507(CHEMBL5203362)
Affinity DataIC50: 610nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605504(CHEMBL5189856)
Affinity DataIC50: 700nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605500(CHEMBL5171388)
Affinity DataIC50: 710nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50525744(CHEMBL4555782)
Affinity DataIC50: 741nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 mins using IP6 as substrate in presence of ATP by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50525744(CHEMBL4555782)
Affinity DataIC50: 750nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 mins using IP6 as substrate in presence of ATP by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634465(CHEMBL5425948)
Affinity DataIC50: 757nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605501(CHEMBL5185229)
Affinity DataIC50: 800nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM373532(US9903855, Molecule 1)
Affinity DataIC50: 860nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634444(CHEMBL5437046)
Affinity DataIC50: 896nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605486(CHEMBL1460920)
Affinity DataIC50: 910nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50261491(N2-(3-(trifluoromethyl)benzyl)-N6-(4-nitrobenzyl)-...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634434(CHEMBL5394030)
Affinity DataIC50: 1.07E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM115059(cid_17015159 | MLS001199620 | SMR000560152 | 3-(4-...)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634435(CHEMBL5401207)
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605481(CHEMBL5199101)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605503(CHEMBL5205377)
Affinity DataIC50: 1.56E+3nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50525733(CHEMBL4459958)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 mins using IP6 as substrate in presence of ATP by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50605499(CHEMBL5178548)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of N-terminal 6His-MBP-tagged recombinant human IP6K1 expressed in Escherichia coli assessed as inorganic phosphate release using InsP6 as...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50525759(CHEMBL4465245)
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 mins using IP6 as substrate in presence of ATP by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634445(CHEMBL5398720)
Affinity DataIC50: 2.22E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634468(CHEMBL5428140)
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634474(CHEMBL5403179)
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634464(CHEMBL5406283)
Affinity DataIC50: 2.41E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634443(CHEMBL5397708)
Affinity DataIC50: 2.58E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50525741(CHEMBL4563130)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 mins using IP6 as substrate in presence of ATP by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetInositol hexakisphosphate kinase 1(Human)
University of North Carolina At Chapel Hill

Curated by ChEMBL
LigandPNGBDBM50634437(CHEMBL5428644)
Affinity DataIC50: 2.88E+3nMAssay Description:Inhibition of IP6K1 (unknown origin) incubated for 30 min in presence of ATP by ADPGlo reagent based assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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