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TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361248(CHEMBL1934890)
Affinity DataKd:  1.10E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361249(CHEMBL1934891)
Affinity DataKd:  5.20E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361250(CHEMBL1934892)
Affinity DataKd:  1.90E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361251(CHEMBL1934893)
Affinity DataKd:  1.30E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361252(CHEMBL1934894)
Affinity DataKd:  3.20E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361253(CHEMBL1934895)
Affinity DataKd:  4.10E+3nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361254(CHEMBL1934896)
Affinity DataKd:  3.30E+3nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361255(CHEMBL1934897)
Affinity DataKd:  1.40E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361256(CHEMBL1934898)
Affinity DataKd:  3.00E+3nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361257(CHEMBL1934899)
Affinity DataKd:  3.00E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361258(CHEMBL1934900)
Affinity DataKd:  7.50E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361259(CHEMBL1934901)
Affinity DataKd:  1.40E+3nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361260(CHEMBL1934902)
Affinity DataKd:  1.20E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361261(CHEMBL1934903)
Affinity DataKd:  2.00E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361262(CHEMBL1934904)
Affinity DataKd:  1.40E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361263(CHEMBL1934905)
Affinity DataKd:  1.10E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361264(CHEMBL1934906)
Affinity DataKd:  1.40E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361265(CHEMBL1934907)
Affinity DataKd:  3.80E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361266(CHEMBL1934908)
Affinity DataKd:  1.10E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361267(CHEMBL1934909)
Affinity DataKd:  1.30E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM50361268(CHEMBL1934910)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase 7(Human)
University of Applied Sciences

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataKd:  3.60E+4nMAssay Description:Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137826(8-Biphenyl-4-yl-8-oxo-octanoic acid (2-amino-pheny...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137843(8-Biphenyl-3-yl-8-oxo-octanoic acid (2-amino-pheny...)
Affinity DataEC50:  2.50E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137828(6-(5-Hydroxy-6-morpholin-4-ylmethyl-1,3-dioxo-1H,3...)
Affinity DataEC50:  2.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137838(6-(6-Bromo-1,3-dioxo-1H,3H-benzo[de]isoquinolin-2-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137832(8-Naphthalen-2-yl-8-oxo-octanoic acid (2-amino-phe...)
Affinity DataEC50:  2.50E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137835(8-(4-Bromo-phenyl)-8-oxo-octanoic acid (2-amino-ph...)
Affinity DataEC50:  1.50E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137829(6-(5-Hydroxy-1,3-dioxo-1H,3H-benzo[de]isoquinolin-...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137850(6-(5,7-Dioxo-5,7-dihydro-pyrrolo[3,4-b]pyridin-6-y...)
Affinity DataEC50: >2.50E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137827(8-Oxo-8-phenyl-octanoic acid (2-amino-phenyl)-amid...)
Affinity DataEC50:  2.50E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137831(8-Oxo-8-(6-phenyl-pyridin-3-yl)-octanoic acid (2-a...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137839(6-(5-Hydroxy-1,3-dioxo-6-piperidin-1-ylmethyl-1H,3...)
Affinity DataEC50:  1.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137837(8-Oxo-8-(4-pyridin-3-yl-phenyl)-octanoic acid (2-a...)
Affinity DataEC50:  2.00E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137841(6-(4-Oxo-4H-benzo[d][1,2,3]triazin-3-yl)-hexanoic ...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137846(6-(4-Oxo-4H-quinazolin-3-yl)-hexanoic acid (2-amin...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137845(6-(5-Methyl-1,3-dioxo-1,3-dihydro-isoindol-2-yl)-h...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137836(8-(3',4'-Dimethoxy-biphenyl-4-yl)-8-oxo-octanoic a...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137830(6-(5-Hydroxy-1,3-dioxo-1,3-dihydro-isoindol-2-yl)-...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137844(6-(1-Oxo-1,3-dihydro-isoindol-2-yl)-hexanoic acid ...)
Affinity DataEC50:  9.90E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137842(8-(4-Methoxy-phenyl)-8-oxo-octanoic acid (2-amino-...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137848(6-(1,3-Dioxo-1,3-dihydro-isoindol-2-yl)-hexanoic a...)
Affinity DataEC50:  5.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137849(6-(1,3-Dioxo-1H,3H-benzo[de]isoquinolin-2-yl)-hexa...)
Affinity DataEC50:  3.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50137834(6-(2,4-Dioxo-1,4-dihydro-2H-quinazolin-3-yl)-hexan...)
Affinity DataEC50:  1.00E+4nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM19410(benzamide-type inhibitor, 3 | CHEMBL27759 | pyridi...)
Affinity DataEC50:  1.00E+3nMAssay Description:Effect on induced hyperacetylation of histones in whole cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM19149(Zolinza | suberoylanilide hydroxamic acid | CHEMBL...)
Affinity DataEC50:  180nMAssay Description:Inhibition of HDAC in human cell lysates using fluoro-substrate peptide/fluoro-deacetylated peptide as substrate incubated for 20 mins measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM25150(Belinostat | (2E)-N-hydroxy-3-[3-(phenylsulfamoyl)...)
Affinity DataEC50:  30nMAssay Description:Inhibition of HDAC in human cell lysates using fluoro-substrate peptide/fluoro-deacetylated peptide as substrate incubated for 20 mins measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50465051(CHEMBL4285950)
Affinity DataEC50:  350nMAssay Description:Inhibition of HDAC in human cell lysates using fluoro-substrate peptide/fluoro-deacetylated peptide as substrate incubated for 20 mins measured at 1 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50483539(CHEMBL1688184)
Affinity DataEC50:  30nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistone deacetylase(Human)
Methylgene

Curated by ChEMBL
LigandPNGBDBM50483540(CHEMBL1688186)
Affinity DataEC50:  190nMAssay Description:Inhibition of HDAC activity in human NB4 cells assessed as acetylation of histone H3 after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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