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TargetNEDD8-activating enzyme E1 catalytic/regulatory subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50285607(MLN-4924 | MLN-4924003 | Pevonedistat)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of NAE-mediated Ubcl2-NEDD8 conjugation in human Caco2 cells after 16 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM67690(SMR000058480 | DHAD | 1,4-bis[2-(2-hydroxyethylami...)
Affinity DataEC50:  1.30E+3nMAssay Description:Inhibition of NAE-mediated Ubcl2-NEDD8 conjugation in human Caco2 cells after 16 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50318907(CHEMBL1014 | TCV-116 | candesartancilexetil | Atac...)
Affinity DataKd:  1.95E+5nMAssay Description:Binding affinity to biotin-labeled GST-tagged NAE (unknown origin) incubated for 1 hr by SPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50285607(MLN-4924 | MLN-4924003 | Pevonedistat)
Affinity DataEC50:  30nMAssay Description:Inhibition of NAE in human HCT-116 cells incubated for 1 hr by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601510(CHEMBL5170838)
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601479(CHEMBL5182746)
Affinity DataIC50: 0.210nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50285607(MLN-4924 | MLN-4924003 | Pevonedistat)
Affinity DataIC50: 0.260nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50594972(CHEMBL5177755)
Affinity DataIC50: 0.550nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601508(CHEMBL5206652)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM320991(4-Amino-7-[(2R,3R,4S,5R)-3,4-dihydroxy-5-[(sulfamo...)
Affinity DataIC50: 0.955nMAssay Description:Inhibition of recombinant human APPBP1/UBA3 expressed in Escherichia coli assessed as Ub/Ubl thioester transferMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601511(CHEMBL5181979)
Affinity DataIC50: 1nMAssay Description:Inhibition of NAE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601501(CHEMBL5173723)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601494(CHEMBL5192493)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601496(CHEMBL5197178)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50285607(MLN-4924 | MLN-4924003 | Pevonedistat)
Affinity DataIC50: 4nMAssay Description:Inhibition of NAE1/UBA3 in human HCT-116 cells assessed as reduction in Ubc12-NEDD8 level incubated for 24 hrs by immunoblot analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50285607(MLN-4924 | MLN-4924003 | Pevonedistat)
Affinity DataIC50: 4nMAssay Description:Inhibition of NAE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601503(CHEMBL5209054)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50285607(MLN-4924 | MLN-4924003 | Pevonedistat)
Affinity DataIC50: 5nMAssay Description:Inhibition of human recombinant His-tagged NAE1 expressed in baculovirus expression system after 90 mins in presence of FLAG-tagged NEDD8 by TR-FRET ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601509(CHEMBL5188530)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601502(CHEMBL5193236)
Affinity DataIC50: 6nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601482(CHEMBL5177700)
Affinity DataIC50: 6.10nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601511(CHEMBL5181979)
Affinity DataIC50: 8nMAssay Description:Inhibition of NAE in human HCT-116 cells incubated for 1 hr by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601505(CHEMBL5178136)
Affinity DataIC50: 9.80nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575579(CHEMBL4847817)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601507(CHEMBL5192527)
Affinity DataIC50: 10nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50427035(CHEMBL2017005)
Affinity DataIC50: 10nMAssay Description:Inhibition of NAE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601484(CHEMBL5169743)
Affinity DataIC50: 16nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601488(CHEMBL5170141)
Affinity DataIC50: 21nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601504(CHEMBL5179467)
Affinity DataIC50: 21nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575577(CHEMBL4860740)
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575555(CHEMBL4878088)
Affinity DataIC50: 29nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575593(CHEMBL4878832)
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601483(CHEMBL5207989)
Affinity DataIC50: 31nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575562(CHEMBL4852015)
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM462715({(1R,2S,4R)-4-[(5-{[4-(3-chlorobenzyl)-5-methyl-2-...)
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM462705(US10780090, Compound I-43 | {(1R,2S,4R)-4-[(5-{[4-...)
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575586(CHEMBL4848442)
Affinity DataIC50: 64nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601499(CHEMBL5201960)
Affinity DataIC50: 67nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601490(CHEMBL5206263)
Affinity DataIC50: 81nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601485(CHEMBL5206633)
Affinity DataIC50: 82nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM462725(US10780090, Compound I-59 | {(1R,2S,4R)-4-[(5-{[4-...)
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575599(CHEMBL4848140)
Affinity DataIC50: 102nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601486(CHEMBL5190183)
Affinity DataIC50: 107nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575581(CHEMBL4860263)
Affinity DataIC50: 114nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575581(CHEMBL4860263)
Affinity DataIC50: 114nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601506(CHEMBL5188300)
Affinity DataIC50: 120nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50575578(CHEMBL4847843)
Affinity DataIC50: 122nMAssay Description:Inhibition of recombinant NAE (unknown origin) in presence of ATP at Km concentration by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601487(CHEMBL5200375)
Affinity DataIC50: 149nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601497(CHEMBL5173277)
Affinity DataIC50: 170nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetNEDD8-activating enzyme E1 catalytic subunit(Human)
University of Macau

Curated by ChEMBL
LigandPNGBDBM50601500(CHEMBL5188093)
Affinity DataIC50: 187nMAssay Description:Inhibition of NAE (unknown origin) mediated neddylation assessed as decrease in NEDD8-Ubcl2 adduct formation incubated for 2 hrs in presence of L-glu...More data for this Ligand-Target Pair
In DepthDetails
PubMed
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