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TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50353094(CHEMBL1823117)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at rat recombinant TRPA1 receptor expressed in HEK293 cells assessed as stimulation of intracellular calcium level using Fluo4-AM dy...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50362768(CHEMBL1939828)
Affinity DataEC50:  220nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of N-methyl-maleimide-induced current by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50364436(CHEMBL1950597)
Affinity DataEC50:  2.21E+4nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50364435(CHEMBL1950598)
Affinity DataEC50:  2.20E+3nMAssay Description:Agonist activity at rat TRPA1 ion channel expressed in HEK293 cells assessed as calcium influx by fluo-4-Am-based fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037025(CHEBI:5331 | GERANYL ACETATE)
Affinity DataEC50:  2.58E+4nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037026(CHEMBL3355275)
Affinity DataEC50:  330nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037027(CHEMBL3355276)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037028(CHEMBL3355277)
Affinity DataEC50:  480nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037029(CHEMBL3355278)
Affinity DataEC50:  1.19E+4nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037030(CHEMBL3355279)
Affinity DataEC50:  360nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036937(CHEMBL3355280)
Affinity DataEC50:  120nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036938(CHEMBL3355281)
Affinity DataEC50:  510nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036939(CHEMBL3355282)
Affinity DataEC50:  390nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036940(CHEMBL3355283)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036941(CHEMBL3355284)
Affinity DataEC50:  7.50E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036942(CHEMBL3355285)
Affinity DataEC50:  610nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036943(CHEMBL3355286)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036944(CHEMBL3355287)
Affinity DataEC50:  45nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036945(CHEMBL3355288)
Affinity DataEC50:  92nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036946(CHEBI:29452 | Nerol)
Affinity DataEC50:  1.17E+4nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036947(NERYL ACETATE)
Affinity DataEC50:  1.33E+4nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036948(CHEMBL3355289)
Affinity DataEC50:  93nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036949(CHEMBL3355290)
Affinity DataEC50:  140nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036950(CHEMBL3355291)
Affinity DataEC50:  260nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036951(CHEMBL3355292)
Affinity DataEC50:  43nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036952(CHEMBL3355293)
Affinity DataEC50:  16nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036953(CHEMBL3355294)
Affinity DataEC50:  140nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036954(CHEMBL3355295)
Affinity DataEC50:  100nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036955(CHEMBL3355296)
Affinity DataEC50:  81nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036956(CHEMBL3355297)
Affinity DataEC50:  110nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50036957(CHEMBL3355298)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037022(CHEMBL3355299)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037031(CHEMBL3355300)
Affinity DataEC50:  430nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037032(CHEMBL3355301)
Affinity DataEC50:  2.65E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037033(CHEMBL3355302)
Affinity DataEC50:  18nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037034(CHEMBL3355303)
Affinity DataEC50:  41nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037035(CHEBI:50462 | Citronellol | DL-citronellol)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037054(CHEBI:70478 | CITRONELLYL ACETATE)
Affinity DataEC50:  1.22E+4nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037055(CHEMBL3355304)
Affinity DataEC50:  280nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037056(CHEMBL3355305)
Affinity DataEC50:  90nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037057(CHEMBL3355306)
Affinity DataEC50:  53nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50037058(CHEMBL3355307)
Affinity DataEC50:  160nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular Ca2+ concentration by Fluo-4-AM dye based spectrofluori...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50362741(CHEMBL1939826)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50046741(CHEMBL3314490)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50046742(CHEMBL3314489)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50046743(CHEMBL3314488)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50046744(CHEMBL3314487)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50046745(CHEMBL3314486)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50046746(CHEMBL3314485)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
Universita` Del Piemonte Orientale

Curated by ChEMBL
LigandPNGBDBM50046749(CHEMBL3314484)
Affinity DataEC50: >4.00E+4nMAssay Description:Agonist activity at rat TRPA1 by [45Ca2+] fluorimetry assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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