Compile Data Set for Download or QSAR
Report error Found 91 of affinity data for UniProtKB/TrEMBL: Q63120
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047316(CHEMBL3314525)
Affinity DataEC50:  3.80E+4nMAssay Description:Stimulation of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047200(CHEMBL3314564)
Affinity DataEC50: >2.00E+5nMAssay Description:Stimulation of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047213(CHEMBL3314565)
Affinity DataEC50: >2.00E+5nMAssay Description:Stimulation of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047215(CHEMBL3314567)
Affinity DataEC50: >2.00E+5nMAssay Description:Stimulation of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047309(CHEMBL3314576)
Affinity DataEC50:  1.10E+5nMAssay Description:Stimulation of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50358848(CHEMBL1923433)
Affinity DataEC50:  2.70E+4nMAssay Description:Stimulation of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50420230(CHEMBL2074750)
Affinity DataIC50: 100nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in bile canalicular membranes from Wistar ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50420229(CHEMBL2074720)
Affinity DataIC50: 120nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake (LTC4: 0.05 uM) in bile canalicular membranes from Wistar ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50420221(CHEMBL325447)
Affinity DataIC50: 200nMAssay Description:TP_TRANSPORTER: inhibition of Naf-GlcA uptake (Naf-GlcA: 0.1 uM) in bile canalicular membrane vesicles of Wistar ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485596(Leukotriene C4 | LEUKOTRIEN C4)
Affinity DataIC50: 650nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.055 uM) in membrane vesicles from Mrp2-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50001285(3-(((3-(2-(7-chloroquinoline-2-yl)ethenyl)phenyl)(...)
Affinity DataIC50: 2.62E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.055 uM) in membrane vesicles from Mrp2-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50292408(5S-hydroxy-6R-(S-cysteinylglycinyl)-7E,9E,11E,14Z-...)
Affinity DataIC50: 5.48E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.055 uM) in membrane vesicles from Mrp2-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50297387((5S-(5R*,6S*(S*),7E,9E,11Z,14Z))-6-((2-Amino-2-car...)
Affinity DataIC50: 9.83E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.055 uM) in membrane vesicles from Mrp2-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485605(Leukotriene F4 | LEUKOTRIEN F4)
Affinity DataIC50: 1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.055 uM) in membrane vesicles from Mrp2-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataIC50: 1.20E+4nMAssay Description:TP_TRANSPORTER: inhibition of Naf-GlcA uptake (Naf-GlcA: 0.1 uM) in bile canalicular membrane vesicles of Wistar ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50344959(17beta-Estradiol-17-(beta-D-glucuronide) | estradi...)
Affinity DataIC50: 1.33E+4nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake (DNP-SG: 0.05 uM) in membrane vesicles from Mrp2-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataIC50: 1.93E+4nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake (E217betaG: 0.055 uM) in membrane vesicles from Mrp2-expressing Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50524101(CHEMBL4474619)
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of Sprague-Dawley rat Mrp2 expressed in baculovirus infected Sf21 insect cell vesicles assessed as reduction in CDF uptake by fluorescence...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50524102(CHEMBL4542281)
Affinity DataIC50: 7.40E+4nMAssay Description:Inhibition of Sprague-Dawley rat Mrp2 expressed in baculovirus infected Sf21 insect cell vesicles assessed as reduction in CDF uptake by fluorescence...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047215(CHEMBL3314567)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibition of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047200(CHEMBL3314564)
Affinity DataIC50: 7.80E+4nMAssay Description:Inhibition of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50358848(CHEMBL1923433)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047316(CHEMBL3314525)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047213(CHEMBL3314565)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50047309(CHEMBL3314576)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of ATPase activity of rat Mrp2 assessed as inorganic phosphateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485593(CHEMBL2074809)
Affinity DataKi:  46nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50185127(30-hydroxy-11,30-dioxoolean-12-en-3beta-yl (2-O-be...)
Affinity DataKi:  840nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50420250(INDOCYANINE GREEN)
Affinity DataKi:  1.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50390982(CHEMBL2075008)
Affinity DataKi:  1.01E+3nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485567(CHEMBL2075009)
Affinity DataKi:  1.03E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485569(Glucuronidated Sn-38 | CHEMBL1743143)
Affinity DataKi:  1.62E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50185127(30-hydroxy-11,30-dioxoolean-12-en-3beta-yl (2-O-be...)
Affinity DataKi:  1.91E+3nMAssay Description:TP_TRANSPORTER: inhibition of SN-38 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKi:  1.96E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50390979(BROMOSULFOPHTHALEIN)
Affinity DataKi:  2.18E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50390979(BROMOSULFOPHTHALEIN)
Affinity DataKi:  2.87E+3nMAssay Description:TP_TRANSPORTER: inhibition of SN-38 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391002(CHEMBL2074599)
Affinity DataKi:  3.84E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM58924((2Z)-2-[(3R,4S,5S,8S,9S,10S,11R,13R,14S,16S)-16-ac...)
Affinity DataKi:  5.50E+3nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in canalicular membrane vesicles of rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM58924((2Z)-2-[(3R,4S,5S,8S,9S,10S,11R,13R,14S,16S)-16-ac...)
Affinity DataKi:  7.60E+3nMAssay Description:TP_TRANSPORTER: inhibition of E217betaG uptake in canalicular membrane vesicles of rat liverMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50242173((2S,3S,4S,5R,6S)-6-(5,6-dihydroxy-4-oxo-2-phenyl-4...)
Affinity DataKi:  7.95E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50390985(CHEMBL2074707)
Affinity DataKi:  8.32E+3nMAssay Description:TP_TRANSPORTER: inhibition of BQ-123 uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391008(CHEMBL2074711)
Affinity DataKi:  9.20E+3nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50422690(Cefodizime Sodium | HR-221 [As Sodium] | S-771221B...)
Affinity DataKi:  1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50022815((3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-ethyl-33...)
Affinity DataKi:  1.00E+4nMAssay Description:TP_TRANSPORTER: inhibition of BMG uptake in membrane vesicles from Mrp2-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485591(CHEMBL2075019)
Affinity DataKi:  1.14E+4nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM58924((2Z)-2-[(3R,4S,5S,8S,9S,10S,11R,13R,14S,16S)-16-ac...)
Affinity DataKi:  1.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of LTC4 uptake in Mrp2-expressing HEK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485588(CHEMBL2075023)
Affinity DataKi:  1.48E+4nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485568(CHEMBL2074578)
Affinity DataKi:  1.83E+4nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataKi:  2.58E+4nMAssay Description:TP_TRANSPORTER: inhibition of Temocaprilat uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50485587(CHEMBL2074653)
Affinity DataKi:  3.25E+4nMAssay Description:TP_TRANSPORTER: inhibition of DNP-SG uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetATP-binding cassette sub-family C member 2(Rat)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50391004(CHEMBL213947)
Affinity DataKi:  3.45E+4nMAssay Description:TP_TRANSPORTER: inhibition of 5-methyltetrahydrofolate uptake in bile canalicular membrane vesicles from SD ratMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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