Compile Data Set for Download or QSAR
Report error Found 214 for UniProtKB: P70605
LigandPNGBDBM92478(CHEMBL1360 | Atracurium besylate)
Affinity DataKd:  6.40E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50366799(TUBOCURARINE | TUBOCURARINE CHLORIDE)
Affinity DataKd:  1.60E+4nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50377979(PENUCURONIUM)
Affinity DataKd:  2.10E+4nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50048403(dequalinium | 1-[10-(4-amino-2-methyl-1-quinoliniu...)
Affinity DataKd:  180nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50061977(CHEMBL117908 | 17,25-diazonia-2,9-diazaheptacyclo[...)
Affinity DataKd:  2.70nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50092131(CHEMBL612120 | UCL-1848 | CHEMBL420873 | 1,7-diazo...)
Affinity DataKd:  0.430nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50199404(1-(3,4-Dimethoxy-benzyl)-6,7-dimethoxy-2,2-dimethy...)
Affinity DataKd:  2.60E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50263331((1H-Benzoimidazol-2-yl)-(R)-1,2,3,4-tetrahydronaph...)
Affinity DataKd:  77nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275156((1H-benzoimidazol-2-yl)benzylamine | CHEMBL456446)
Affinity DataKd:  2.70E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275155((1H-Benzoimidazol-2-yl)-(4-chlorobenzyl)amine | CH...)
Affinity DataKd:  640nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275154((1H-Benzoimidazol-2-yl)-(3,4-dichlorobenzyl)amine ...)
Affinity DataKd:  200nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275153(2-(2-Phenylpyrrolidin-1-yl)-1H-benzoimidazole | CH...)
Affinity DataKd:  1.60E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275152(2-(2-Phenylpiperidin-1-yl)-1H-benzoimidazole | CHE...)
Affinity DataKd:  750nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275131(2-(1H-Benzoimidazol-2-yl)-1,2,3,4-tetrahydroisoqui...)
Affinity DataKd:  1.40E+4nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275130((1H-Benzoimidazol-2-yl)indan-1-ylamine | CHEMBL458...)
Affinity DataKd:  790nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275129((1H-Benzoimidazol-2-yl)-1,2,3,4-tetrahydronaphthal...)
Affinity DataKd:  130nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275128((1H-Benzoimidazol-2-yl)-(6,7,8,9-tetrahydro-5H-ben...)
Affinity DataKd:  590nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275127((1H-Benzoimidazol-2-yl)indan-2-ylamine | CHEMBL453...)
Affinity DataKd:  1.70E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275126((1H-Benzoimidazol-2-yl)-(1,2,3,4-tetrahydronaphtha...)
Affinity DataKd:  2.00E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275125((1H-Benzoimidazol-2-yl)-(2-methyl-1,2,3,4-tetrahyd...)
Affinity DataKd:  170nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275092((1H-Benzoimidazol-2-yl)-(4-methyl-1,2,3,4-tetrahyd...)
Affinity DataKd:  32nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275091((1H-Benzoimidazol-2-yl)-(8-chloro-1,2,3,4-tetrahyd...)
Affinity DataKd:  27nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275053((1H-Benzoimidazol-2-yl)-(7-chloro-1,2,3,4-tetrahyd...)
Affinity DataKd:  17nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275052((1H-Benzoimidazol-2-yl)-(6-chloro-1,2,3,4-tetrahyd...)
Affinity DataKd:  120nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275051((1H-Benzoimidazol-2-yl)-(5-chloro-1,2,3,4-tetrahyd...)
Affinity DataKd:  44nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275050((1H-Benzoimidazol-2-yl)-(7-fluoro-1,2,3,4-tetrahyd...)
Affinity DataKd:  34nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275049((1H-Benzoimidazol-2-yl)-(7-bromo-1,2,3,4-tetrahydr...)
Affinity DataKd:  11nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275090((1H-Benzoimidazol-2-yl)-(6,7-dichloro-1,2,3,4-tetr...)
Affinity DataKd:  9.10nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275089((1H-Benzoimidazol-2-yl)-(7-methyl-1,2,3,4-tetrahyd...)
Affinity DataKd:  20nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275088((1H-Benzoimidazol-2-yl)-(5,7-dimethyl-1,2,3,4-tetr...)
Affinity DataKd:  33nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275087((1H-Benzoimidazol-2-yl)-(7-methoxy-1,2,3,4-tetrahy...)
Affinity DataKd:  61nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275054((1H-Benzoimidazol-2-yl)chroman-4-ylamine | CHEMBL5...)
Affinity DataKd: >1.00E+4nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275207((1H-Benzoimidazol-2-yl)thiochroman-4-yl-amine | CH...)
Affinity DataKd:  130nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275208((1H-Benzoimidazol-2-yl)-(5,6,7,8-tetrahydroisoquin...)
Affinity DataKd:  6.50E+3nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275209((1H-Benzoimidazol-2-yl)-(4,5,6,7-tetrahydrobenzo[b...)
Affinity DataKd:  540nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275232((1H-Benzoimidazol-2-yl)-(1,2,3,4-tetrahydrophenant...)
Affinity DataKd:  31nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275233((1H-Benzoimidazol-2-yl)(7-phenyl-1,2,3,4-tetrahydr...)
Affinity DataKd:  600nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275234((S)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-benzo...)
Affinity DataKd:  450nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50240909(2-phenethyl-1H-benzo[d]imidazole | 2-Phenethyl-1H-...)
Affinity DataKd: >1.00E+4nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50275235(N-(1H-benzo[d]imidazol-2-yl)-4-chlorobenzamide | C...)
Affinity DataKd: >1.00E+4nMAssay Description:Inhibition of Wistar rat recombinant SK3 channel expressed in HEK293 cells by whole cell patch clamp techniqueMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM392076(US10301272, Example 7/9)
Affinity DataIC50: 0.0120nMAssay Description:Displacement of [125I]apamin from rat brain SkCa channel after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50155248(CHEMBL3774478)
Affinity DataIC50: 0.0160nMAssay Description:Displacement of [125I]apamin from rat cerebral cortex small conductance calcium-activated potassium channelMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50092131(CHEMBL612120 | UCL-1848 | CHEMBL420873 | 1,7-diazo...)
Affinity DataIC50: 2nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50061977(CHEMBL117908 | 17,25-diazonia-2,9-diazaheptacyclo[...)
Affinity DataIC50: 3nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50061977(CHEMBL117908 | 17,25-diazonia-2,9-diazaheptacyclo[...)
Affinity DataIC50: 3nMAssay Description:The blocking of apamin-sensitive [Ca2+]-activated K+ (SKCa) channel was assessed by the compounds ability to inhibit the after-hyperpolarization in c...More data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50474856(CHEMBL184300)
Affinity DataIC50: 9nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50474870(CHEMBL185146)
Affinity DataIC50: 10nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50474869(CHEMBL181911)
Affinity DataIC50: 12nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50474865(CHEMBL183644)
Affinity DataIC50: 15nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
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PubMed
LigandPNGBDBM50474867(CHEMBL184858)
Affinity DataIC50: 16nMAssay Description:Inhibition of after hyperpolarization (AHP) of cultured rat sympathetic neurons as SKCa channel blocking activityMore data for this Ligand-Target Pair
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PubMed
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