Compile Data Set for Download or QSAR
Report error Found 29 of affinity data for UniProtKB/TrEMBL: P59594
TargetSpike glycoprotein [668-1255](SARS-CoV)
University of Bonn

LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataEC50:  1.06E+4nMAssay Description:This is a review article.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567444(CHEMBL4873011)
Affinity DataKd:  940nMAssay Description:Binding affinity to SARS-CoV-2 spike glycoprotein S-trimer measured by Surface plasmon resonanceMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM429291(med.21724, Compound 27)
Affinity DataEC50:  760nMAssay Description:This is a review article.More data for this Ligand-Target Pair
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PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM13530(cid_5291 | STI571 | N-(4-methyl-3-{[4-(pyridin-3-y...)
Affinity DataEC50:  1.00E+4nMAssay Description:This is a review article.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM428938(med.21724, Compound 5)
Affinity DataEC50:  3.89E+3nMAssay Description:This is a review article.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein [668-1255](SARS-CoV)
University of Bonn

LigandPNGBDBM428875(med.21724, Compound 2)
Affinity DataEC50:  4.40E+3nMAssay Description:This is a review article.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataEC50:  8.34E+4nMAssay Description:This is a review article.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50559137(CHEMBL4785828)
Affinity DataIC50: 100nMAssay Description:Inhibition of spike protein in SARS-CoV infected in human HeLa cells haboring wild type ACE2 assessed as reduction in virus infectivity preincubated ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50233805(CHEMBL4077922 | US11021454, Compound Salvianolic a...)
Affinity DataIC50: 3.85E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567444(CHEMBL4873011)
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567440(CHEMBL4847112)
Affinity DataIC50: 5.54E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567449(CHEMBL4874301)
Affinity DataIC50: 5.68E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567447(CHEMBL4852531)
Affinity DataIC50: 5.89E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567443(CHEMBL4852791)
Affinity DataIC50: 6.27E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567450(CHEMBL4859094)
Affinity DataIC50: 6.32E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567453(CHEMBL4865746)
Affinity DataIC50: 7.37E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567448(CHEMBL4875210)
Affinity DataIC50: 7.76E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567441(CHEMBL4855702)
Affinity DataIC50: 8.33E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567451(CHEMBL4868650)
Affinity DataIC50: 9.57E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567442(CHEMBL4865677)
Affinity DataIC50: 9.97E+3nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM78433(2-[4-[3-[2-(trifluoromethyl)phenothiazin-10-yl]pro...)
Affinity DataIC50: 1.18E+4nMAssay Description:This is a review article.More data for this Ligand-Target Pair
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PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50001888([3-(2-Chloro-phenothiazin-10-yl)-propyl]-dimethyl-...)
Affinity DataIC50: 1.30E+4nMAssay Description:This is a review article.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567454(CHEMBL4857727)
Affinity DataIC50: 1.31E+4nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567452(CHEMBL4852883)
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567455(CHEMBL3902325)
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567439(CHEMBL4849021)
Affinity DataIC50: 1.81E+4nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567446(CHEMBL4869223)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50567445(CHEMBL4876819)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of spike glycoprotein S in SARS-CoV-2 pseudovirus infected human 293T/ACE2 cells assessed as inhibition of viral infection measured after ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSpike glycoprotein(SARS-CoV)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50017696(N,N,alpha-trimethyl-10H-phenothiazine-10-ethanamin...)
Affinity DataIC50: 2.14E+4nMAssay Description:This is a review article.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed