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TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50094702(CHEMBL15844 | indole | Indole, 7 | Indol | 1H-indo...)
Affinity DataKd:  3.00E+6nMAssay Description:Inhibition of human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50078824(2-Phenyl-1H-imidazole | CHEMBL14189 | US9138393, 2...)
Affinity DataKd:  3.00E+6nMAssay Description:Inhibition of human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50094702(CHEMBL15844 | indole | Indole, 7 | Indol | 1H-indo...)
Affinity DataKd:  3.00E+6nMAssay Description:Dissociation constant against adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50533474(CHEMBL4460859)
Affinity DataIC50: 0.0600nMAssay Description:Inhibition of human adenosine kinase assessed as reduction in conversion of adenosine to AMPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090867((2R,3S,4R,5R)-2-(aminomethyl)-5-(4-chloro-5-iodo-7...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090867((2R,3S,4R,5R)-2-(aminomethyl)-5-(4-chloro-5-iodo-7...)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human adenosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090867((2R,3S,4R,5R)-2-(aminomethyl)-5-(4-chloro-5-iodo-7...)
Affinity DataIC50: 0.100nMAssay Description:Concentration required for 50% inhibition of the adenosine kinase (AK) activity.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090843((2R,3R,4S,5R)-2-(4-amino-5-bromo-7H-pyrrolo[2,3-d]...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090843((2R,3R,4S,5R)-2-(4-amino-5-bromo-7H-pyrrolo[2,3-d]...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human adenosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178014(N-(4-chlorophenyl)-2-(5-phenyl-7-(5-deoxy-beta-D-r...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090843((2R,3R,4S,5R)-2-(4-amino-5-bromo-7H-pyrrolo[2,3-d]...)
Affinity DataIC50: 0.200nMAssay Description:Concentration required for 50% inhibition of the adenosine kinase (AK) activity.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50174602((4R,5R,6S)-5-[4-(4-Fluoro-phenylamino)-5-phenyl-py...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50201834(5-benzo[b]thiophen-2-yl-6-(6-morpholin-4-ylpyridin...)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of cytosolic adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50134740((2R,3R,4S,5S)-2-Hydroxymethyl-5-(5-phenyl-4-phenyl...)
Affinity DataIC50: 0.470nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50134740((2R,3R,4S,5S)-2-Hydroxymethyl-5-(5-phenyl-4-phenyl...)
Affinity DataIC50: 0.470nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090887(5-phenyl-4-(phenylamino)-7-(5-deoxy-beta-D-ribofur...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090887(5-phenyl-4-(phenylamino)-7-(5-deoxy-beta-D-ribofur...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against Human Recombinant Adenosine KinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090887(5-phenyl-4-(phenylamino)-7-(5-deoxy-beta-D-ribofur...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178003(N-cyclopropyl-2-(5-phenyl-7-(5-deoxy-beta-D-ribofu...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178015(2-(5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)-pyrro...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090887(5-phenyl-4-(phenylamino)-7-(5-deoxy-beta-D-ribofur...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090887(5-phenyl-4-(phenylamino)-7-(5-deoxy-beta-D-ribofur...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human adenosine kinase assessed as reduction in conversion of adenosine to AMPMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090862((1R,5S)-2-((3R,4aR)-4-Amino-5-iodo-pyrrolo[2,3-d]p...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090862((1R,5S)-2-((3R,4aR)-4-Amino-5-iodo-pyrrolo[2,3-d]p...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of human adenosine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178007(2-(5-phenyl-7-(beta-D-erythrofuranosyl)-pyrrolo[2,...)
Affinity DataIC50: 0.600nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090862((1R,5S)-2-((3R,4aR)-4-Amino-5-iodo-pyrrolo[2,3-d]p...)
Affinity DataIC50: 0.603nMAssay Description:Concentration required for 50% inhibition of the adenosine kinase (AK) activity.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090883((1R,4S,5R)-2-Hydroxymethyl-5-(5-phenyl-4-phenylami...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50134753((2R,3R,4S,5S)-2-Methyl-5-(5-phenyl-4-phenylamino-p...)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory activity against human recombinant adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090883((1R,4S,5R)-2-Hydroxymethyl-5-(5-phenyl-4-phenylami...)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50134753((2R,3R,4S,5S)-2-Methyl-5-(5-phenyl-4-phenylamino-p...)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178023(2-(5-phenyl-7-(5-deoxy-beta-D-ribofuranosyl)-pyrro...)
Affinity DataIC50: 0.800nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178018(2-(3-phenyl-1-(beta-D-ribofuranosyl)-pyrazolo[3,4-...)
Affinity DataIC50: 0.900nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090874(2-[4-(4-Hydroxy-phenylamino)-5-phenyl-pyrrolo[2,3-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090880(4-[7-(3,4-Dihydroxy-5-methyl-tetrahydro-furan-2-yl...)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090881(2-(6-Bromo-5-phenyl-4-phenylamino-pyrrolo[2,3-d]py...)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50143574(7-((4aS,7aS)-6-Benzyl-octahydro-pyrrolo[3,4-b]pyri...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against human adenosine kinase expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50143575(7-(1-Benzyl-hexahydro-pyrrolo[3,4-b]pyrrol-5-yl)-2...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against human adenosine kinase expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50143581(7-[4-(4-Fluoro-benzyl)-[1,4]diazepan-1-yl]-2-pheny...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against human adenosine kinase expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090881(2-(6-Bromo-5-phenyl-4-phenylamino-pyrrolo[2,3-d]py...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against Human Recombinant Adenosine KinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50174603((1R,2R,3R)-2-[4-(2,3-Dihydro-benzo[1,4]dioxin-6-yl...)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against human recombinant adenosine kinase using [14C]AMP as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178027(N-cyclopentyl-2-(5-phenyl-7-(5-deoxy-beta-D-ribofu...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50201814(5-benzofuran-2-yl-6-(6-morpholin-4-ylpyridin-3-yle...)
Affinity DataIC50: 1nMAssay Description:Inhibition of cytosolic adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50201825(5-(4-chlorophenyl)-6-{6-[(2-methoxyethyl)methylami...)
Affinity DataIC50: 1nMAssay Description:Inhibition of cytosolic adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50201865(1-(4-{5-[6-amino-5-(4-chlorophenyl)pyrimidin-4-yle...)
Affinity DataIC50: 1nMAssay Description:Inhibition of cytosolic adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090875(2-[5-(4-Chloro-phenyl)-4-phenylamino-pyrrolo[2,3-d...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178013(N1-cyclopropyl-N2-(5-phenyl-7-(5-deoxy-beta-D-ribo...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50178019(N-cyclobutyl-2-(5-phenyl-7-(5-deoxy-beta-D-ribofur...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50102928(5-(3-Bromo-phenyl)-7-(6-thiomorpholin-4-yl-pyridin...)
Affinity DataIC50: 1.30nMAssay Description:In vitro concentration required for 50% inhibition against Adenosine Kinase (AK) in the presence of enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50102925(5-(3-Bromo-phenyl)-7-[6-(1,4-dioxa-8-aza-spiro[4.5...)
Affinity DataIC50: 1.40nMAssay Description:In vitro concentration required for 50% inhibition against Adenosine Kinase (AK) in the presence of enzymeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine kinase(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50090895(2-[4-(4-Fluoro-phenylamino)-5-phenyl-pyrrolo[2,3-d...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of recombinant human adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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