Compile Data Set for Download or QSAR
Report error Found 11 of affinity data for UniProtKB/TrEMBL: P54493
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50460516(CHEMBL4227539)
Affinity DataIC50: 470nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50460510(CHEMBL4225584)
Affinity DataIC50: 1.60E+3nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50460511(CHEMBL4225103)
Affinity DataIC50: 2.80E+3nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50406296(CHEMBL145012)
Affinity DataIC50: 3.70E+3nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP [F193S,L370F,L379S,R499W](Bacillus subtilis (strain 168))
Technische Universität München

LigandPNGBDBM50199883(cid_1609 | 3,4-dichloro-1H-isochromen-1-one | CHEM...)
Affinity DataIC50: 4.10E+3nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50460512(CHEMBL4225312)
Affinity DataIC50: 4.60E+3nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50460514(CHEMBL4229256)
Affinity DataIC50: 6.20E+3nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50288096(5-Chloro-2-ethoxy-benzo[d][1,3]oxazin-4-one | CHEM...)
Affinity DataIC50: 7.10E+3nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50460513(CHEMBL4228380)
Affinity DataIC50: 7.30E+3nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP(Bacillus subtilis (strain 168))
Ku Leuven

Curated by ChEMBL
LigandPNGBDBM50460515(CHEMBL4229280)
Affinity DataIC50: 1.50E+4nMAssay Description:Competitive inhibition of Bacillus subtilis rhomboid YqgP preincubated for 30 mins followed by FP-Rh addition measured after 1 hr by gel-based ABPP m...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRhomboid protease GluP [F193S,L370F,L379S,R499W](Bacillus subtilis (strain 168))
Technische Universität München

LigandPNGBDBM165194(4‐Chloro‐7‐nitro‐3‐[...)
Affinity DataIC50: 2.50E+4nMpH: 7.4 T: 2°CAssay Description:We selected several inhibitor structures and determined their apparent IC50 by competitive ABPP.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed