Compile Data Set for Download or QSAR
Report error Found 132 of affinity data for UniProtKB/TrEMBL: P54132
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50505091(CHEMBL4075790)
Affinity DataKd:  4.90E+3nMAssay Description:Binding affinity to His-tagged BLM M1111A mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50505091(CHEMBL4075790)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50505091(CHEMBL4075790)
Affinity DataKd:  6.00E+3nMAssay Description:Binding affinity to His-tagged BLM E1143A mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50505091(CHEMBL4075790)
Affinity DataKd:  6.50E+3nMAssay Description:Binding affinity to His-tagged BLM I1168A mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50505091(CHEMBL4075790)
Affinity DataKd:  5.00E+3nMAssay Description:Binding affinity to His-tagged BLM Y995A mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) by ITC assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544291(CHEMBL4633662)
Affinity DataKd:  760nMAssay Description:Binding affinity to wild-type His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isothermal cal...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544291(CHEMBL4633662)
Affinity DataKd:  1.40E+3nMAssay Description:Binding affinity to His-tagged BLM H996A mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isothermal calorimetric titration ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544291(CHEMBL4633662)
Affinity DataKd:  6.54E+3nMAssay Description:Binding affinity to His-tagged BLM I1168A mutant (unknown origin) expressed in Escherichia coli BL21 (DE3) cells by isothermal calorimetric titration...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440514(CHEMBL2426190)
Affinity DataIC50: 100nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440527(CHEMBL2426164)
Affinity DataIC50: 110nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440533(CHEMBL2426169)
Affinity DataIC50: 300nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544291(CHEMBL4633662)
Affinity DataIC50: 800nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619887(CHEMBL5423610)
Affinity DataIC50: 800nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440528(CHEMBL2426165)
Affinity DataIC50: 910nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50505091(CHEMBL4075790)
Affinity DataIC50: 950nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in BLM helicase unwinding activity using...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440538(CHEMBL2426174)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440517(CHEMBL2426193)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544262(CHEMBL4647093)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619881(CHEMBL5440285)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM48721(SMR000178207 | 1-(3,4-Dichloro-phenyl)-3-(5-pyridi...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50505091(CHEMBL4075790)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440519(CHEMBL2426195)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440531(CHEMBL2426168)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440541(CHEMBL2426177)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544277(CHEMBL4646986)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544261(CHEMBL4636576)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440524(CHEMBL2426161)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544269(CHEMBL4642601)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440531(CHEMBL2426168)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as reduction in BLM helicase unwinding activity using...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544287(CHEMBL4648936)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619886(CHEMBL5424781)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619869(CHEMBL5433468)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544264(CHEMBL4649302)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544275(CHEMBL4632583)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544289(CHEMBL4647563)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619885(CHEMBL5437731)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440531(CHEMBL2426168)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of BLM helicase (unknown origin) binding to DNAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544288(CHEMBL4647503)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544266(CHEMBL4649146)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440522(CHEMBL2426159)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544263(CHEMBL4637928)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544265(CHEMBL4634966)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440506(CHEMBL2426200)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544290(CHEMBL4640219)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619876(CHEMBL5433068)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50505091(CHEMBL4075790)
Affinity DataIC50: 3.95E+3nMAssay Description:Inhibition of 5'-biotin labeled duplex forked-DNA binding to BLM (unknown origin) assessed as increase in unbound DNA levels after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440509(CHEMBL2426179)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50440510(CHEMBL2426181)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of BLM (unknown origin) by gel-based DNA unwinding assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50544268(CHEMBL4637736)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of His-tagged BLM (642 to 1296 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells assessed as reduction in DNA unwi...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRecQ-like DNA helicase BLM(Human)
Sun Yat-Sen University

Curated by ChEMBL
LigandPNGBDBM50619873(CHEMBL5425282)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of His-tagged BLM (unknown origin) expressed in Escherichia coli BL21 (DE3) using 5'-biotin-labeled duplex forked-DNA as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails
PubMed
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