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Report error Found 109 of affinity data for UniProtKB/TrEMBL: P53341
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM152497((E)-N'-(6-Bromo-2-oxoindolin-3-ylidene)-2-(2,4...)
Affinity DataIC50: 2.20E+3nMAssay Description:10 µL of test samples (5 mg/mL DMSO solution) were reconstituted in 100 µL of 100 mM-phosphate buffer (pH6.8) in 96-well microplate and incubated wit...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM152499((E)-N'-(2-oxoindolin-3-ylidene)dodecanehydrazi...)
Affinity DataIC50: 3.00E+3nMAssay Description:10 µL of test samples (5 mg/mL DMSO solution) were reconstituted in 100 µL of 100 mM-phosphate buffer (pH6.8) in 96-well microplate and incubated wit...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM152496((E)-N'-(6-bromo-2-oxoindolin-3-ylidene)-2-(3,4...)
Affinity DataIC50: 3.30E+3nMAssay Description:10 µL of test samples (5 mg/mL DMSO solution) were reconstituted in 100 µL of 100 mM-phosphate buffer (pH6.8) in 96-well microplate and incubated wit...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50308256(1-O-Methyl-2,3-O-isopropylidene-5-(4-cyclohexene-1...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 assessed as inhibition of p-nitrophenol release by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50308259(1-O-Methyl-2,3-O-isopropylidene-5-[4-(1-hydroxycyc...)
Affinity DataIC50: 5.20E+3nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 assessed as inhibition of p-nitrophenol release by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50308258(1-O-Methyl-2,3-O-isopropylidene-5-(4-phenoxymethyl...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 assessed as inhibition of p-nitrophenol release by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181062((E)-N'-(3,5-Dichloro-2-hydroxybenzylidene)-4-(...)
Affinity DataIC50: 6.24E+3nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181064((E)-N'-(5-Chloro-2-hydroxybenzylidene)-4-(2-ox...)
Affinity DataIC50: 8.23E+3nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM243075(α-Gl inhibitor, C3)
Affinity DataIC50: 9.60E+3nMpH: 7.0Assay Description:In this study, the inhibition assay of yeast enzyme was performed in 100 mM phosphate buffer pH 7.0 at 25°C with minor changes, according to the meth...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181061((E)-N'-(3,5-Di-tert-butyl-2-hydroxybenzylidene...)
Affinity DataIC50: 1.02E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181068((E)-N'-(4-Chlorobenzylidene)-4-(2-oxo-2H-chrom...)
Affinity DataIC50: 1.06E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM152498((E)-N'-(6-bromo-2-oxoindolin-3-ylidene)-2- hyd...)
Affinity DataIC50: 1.18E+4nMAssay Description:10 µL of test samples (5 mg/mL DMSO solution) were reconstituted in 100 µL of 100 mM-phosphate buffer (pH6.8) in 96-well microplate and incubated wit...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181069((E)-N'-(3-Chlorobenzylidene)-4-(2-oxo-2H-chrom...)
Affinity DataIC50: 1.20E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181073((E)-N'-(3-bromobenzylidene)-4-(2-oxo-2H-chrome...)
Affinity DataIC50: 1.40E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50308255(1-O-Methyl-2,3-O-isopropylidene-5-(4-phenyl-1H-1,2...)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 assessed as inhibition of p-nitrophenol release by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50308257(1-O-Methyl-2,3-O-isopropylidene-5-(4-carboxylate e...)
Affinity DataIC50: 1.51E+4nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 assessed as inhibition of p-nitrophenol release by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181070((E)-4-(2-Oxo-2H-chromen-3-yl)-N'-(4-(trifluoro...)
Affinity DataIC50: 1.60E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181063((E)-N'-(3-Fluoro-4-hydroxybenzylidene)-4-(2-ox...)
Affinity DataIC50: 1.66E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181067((E)-N'-(3,4-Dihydroxybenzylidene)-4-(2-oxo-2H-...)
Affinity DataIC50: 1.83E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM152494((E)-2-(2,4-dichlorophenyl)-N'-(2-oxo-1-propyli...)
Affinity DataIC50: 1.83E+4nMAssay Description:10 µL of test samples (5 mg/mL DMSO solution) were reconstituted in 100 µL of 100 mM-phosphate buffer (pH6.8) in 96-well microplate and incubated wit...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM60591((E)-N'-(3-Fluorobenzylidene)-4-(2-oxo-2H-chromen-3...)
Affinity DataIC50: 2.26E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181071((E)-N'-(2-Fluorobenzylidene)-4-(2-oxo-2H-chrom...)
Affinity DataIC50: 2.36E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM243068(11-O-(3',4'-dimethoxybenzoyl)-bergenin (6))
Affinity DataIC50: 2.46E+4nMpH: 7.0 T: 2°CAssay Description:α-glucosidase (25 μL, 0.2 U/mL), 25 μL of various concentrations of samples, and 175 μL of 50 mM sodium phosphate buffer (pH 7.0)...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50308260(1-O-Methyl-2,3-O-isopropylidene-5-[4-(tetrahydro-2...)
Affinity DataIC50: 2.47E+4nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 assessed as inhibition of p-nitrophenol release by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM243074(α-Gl inhibitor, C2)
Affinity DataIC50: 2.51E+4nMpH: 7.0Assay Description:In this study, the inhibition assay of yeast enzyme was performed in 100 mM phosphate buffer pH 7.0 at 25°C with minor changes, according to the meth...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181060((E)-N'-(4-Hydroxybenzylidene)-4-(2-oxo-2H-chro...)
Affinity DataIC50: 2.52E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181065((E)-N'-(2-Hydroxy-4-methoxybenzylidene)-4-(2-o...)
Affinity DataIC50: 2.99E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50180587(CHEMBL3734896)
Affinity DataIC50: 3.39E+4nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 using 4-nitrophenyl-alpha-D-glucopyranoside as substrate preincubated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50207546((-)-epivaliolamine | CHEMBL223096)
Affinity DataIC50: 3.60E+4nMAssay Description:Inhibition of baker's yeast alpha-glucosidaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181059((E)-N'-(2-Hydroxybenzylidene)-4-(2-oxo-2H-chro...)
Affinity DataIC50: 3.72E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50333465((2R,3R,4R,5S,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50: 3.83E+4nMpH: 6.8 T: 2°CAssay Description:Reaction mixture (100 µL) contained 70 µL 50 mM Na2HPO4 buffer, pH 6.8, 10 µL test compound (0.5 mM), followed by the addition of 10 &...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181066((E)-N'-(2,4-Dihydroxybenzylidene)-4-(2-oxo-2H-...)
Affinity DataIC50: 3.86E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM23406((3R,4R,5S,6R)-5-{[(2R,3R,4R,5S,6R)-5-{[(2R,3R,4S,5...)
Affinity DataIC50: 4.33E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50190320(CHEMBL3827545)
Affinity DataIC50: 4.98E+4nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 using 4-nitrophenyl-alpha-D-glucopyranoside as substrate preincubated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM84973(Urea derivative, 17)
Affinity DataIC50: 5.88E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM84971(Urea derivative, 15)
Affinity DataIC50: 6.01E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM84965(Urea derivative, 9)
Affinity DataIC50: 6.36E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181074((E)-N'-(2-Methoxybenzylidene)-4-(2-oxo-2H-chro...)
Affinity DataIC50: 6.43E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM84975(Urea derivative, 19)
Affinity DataIC50: 6.43E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM84964(Urea derivative, 8)
Affinity DataIC50: 6.85E+4nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM243073(α-Gl inhibitor, C1)
Affinity DataIC50: 7.49E+4nMpH: 7.0Assay Description:In this study, the inhibition assay of yeast enzyme was performed in 100 mM phosphate buffer pH 7.0 at 25°C with minor changes, according to the meth...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM181058((E)-N'-(4-Methoxybenzylidene)-4-(2-oxo-2H-chro...)
Affinity DataIC50: 8.17E+4nMpH: 6.8Assay Description:The test compounds were dissolved in DMSO to prepare the required distributing concentration. α-Glucosidase inhibitory activity was assayed by u...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM152495((E)-N'-(5-chloro-2-oxoindolin-3-ylidene)-4- me...)
Affinity DataIC50: 8.35E+4nMAssay Description:10 µL of test samples (5 mg/mL DMSO solution) were reconstituted in 100 µL of 100 mM-phosphate buffer (pH6.8) in 96-well microplate and incubated wit...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50100861(Protocatechuic acid (M1) | Protocatechuic acid | 3...)
Affinity DataIC50: 8.51E+4nMAssay Description:The assay was performed using isolated phenolics from maize, and inhibition was determined according to previously described method.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50190323(CHEMBL3827417)
Affinity DataIC50: 8.57E+4nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 using 4-nitrophenyl-alpha-D-glucopyranoside as substrate preincubated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM4374(p-Coumaric Acid | p-hydroxycinnamic acid (M4) | CH...)
Affinity DataIC50: 9.08E+4nMAssay Description:The assay was performed using isolated phenolics from maize, and inhibition was determined according to previously described method.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM108032(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-3-[(2S,3R,4S...)
Affinity DataIC50: 9.82E+4nMAssay Description:The assay was performed using isolated phenolics from maize, and inhibition was determined according to previously described method.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50322066(CHEMBL1172402 | Stilbene derivative, 3 | 3,5-Dihyd...)
Affinity DataIC50: 1.02E+5nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM84974(Urea derivative, 18)
Affinity DataIC50: 1.05E+5nMAssay Description:All enzymatic activities were determined by using the appropriate substrate (p-nitrophenyl-alpha-D-glucopyranoside, p-nitrophenyl-beta-D-gulcopyranos...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAlpha-glucosidase MAL12(Baker's yeast)
Hazara University

LigandPNGBDBM50333465((2R,3R,4R,5S,6R)-5-((2R,3R,4R,5S,6R)-5-((2R,3R,4S,...)
Affinity DataIC50: 1.09E+5nMAssay Description:Inhibition of yeast alpha-glucosidase MAL12 assessed as inhibition of p-nitrophenol release by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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