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TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  5.70nMAssay Description:Binding affinity to human KPNA2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataKd:  72nMAssay Description:Binding affinity against KPNA2 (unknown origin) assessed as apparent dissociation constant incubated for 1 hr by colloidal coomassie staining based L...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM50365463(CHEMBL1232461)
Affinity DataIC50: 140nMAssay Description:Inhibition of KPNA2 (unknown origin) incubated for 1 hr by colloidal coomassie staining based LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75103(MLS001044525 | cid_6184270 | 3-(1,3-benzothiazol-2...)
Affinity DataEC50: <380nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM30856(SMR000029847 | MLS000094257 | 1-(4-methylphenyl)-2...)
Affinity DataEC50:  720nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75285(3-[2-(2-methoxyphenyl)ethynyl]-10-methylacridin-9-...)
Affinity DataEC50:  721nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM55566(2-Cyano-N-[2-(1H-indol-3-yl)-ethyl]-3-(5-piperidin...)
Affinity DataEC50:  753nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74600(SMR000046228 | N-(1-ethyl-8-methyl-pyrazolo[3,4-b]...)
Affinity DataEC50:  862nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM60177(SMR000313017 | MLS000682934 | 4-[5-[(Z)-[1-[(2-chl...)
Affinity DataEC50:  908nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75083(cid_1932059 | 7-Benzyl-3-cyclohexyl-2-hydrazino-5,...)
Affinity DataEC50:  918nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM56912(SMR000040521 | MLS000037714 | 1-benzyl-2-(furan-2-...)
Affinity DataEC50:  932nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74553(5,8-dimethyl-2-pyrrolidin-1-ylquinoline-3-carbonit...)
Affinity DataEC50:  1.21E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM58584(MLS001250005 | ethyl 2-fluoranyl-4-(10-methyl-9-ox...)
Affinity DataEC50:  1.29E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75040(SMR000314559 | N'-[(E)-[5-(hydroxymethyl)-2-methyl...)
Affinity DataEC50:  1.52E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75085((E)-2-Cyano-3-(9-methyl-4-oxo-2-phenoxy-4H-pyrido[...)
Affinity DataEC50:  1.58E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM52272(1-(3,4-dimethylphenyl)-2,5-bis(oxidanylidene)dipyr...)
Affinity DataEC50:  1.78E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74787(N-[2-(2-Amino-3-cyano-pyrrolo[2,3-b]quinoxalin-1-y...)
Affinity DataEC50:  2.04E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74980(3-[(E)-2-(4-chlorophenyl)ethenyl]imidazo[1,5-a]pyr...)
Affinity DataEC50:  2.54E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74846((5Z)-1-(3-methylphenyl)-5-[(E)-3-phenylazanylprop-...)
Affinity DataEC50:  2.77E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75266(6-chloro-3-[2-[4-[2,3-dihydro-1,4-benzodioxin-3-yl...)
Affinity DataEC50:  2.90E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM70582(2-Amino-1-benzo[1,3]dioxol-5-ylmethyl-1H-pyrrolo[2...)
Affinity DataEC50:  3.12E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM52071(MLS000034945 | SMR000014519 | 6-Amino-8-(4-isoprop...)
Affinity DataEC50:  3.34E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75027(N-(5,6-dihydrobenzo[h]quinazolin-2-yl)-2-propan-2-...)
Affinity DataEC50:  3.48E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74784([4-[2-(3,5-dimethoxyphenyl)-5-methyl-pyrazolo[1,5-...)
Affinity DataEC50:  3.68E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM30737(4-chlorobenzoic acid 2-(2-amino-3-cyano-1-pyrrolo[...)
Affinity DataEC50:  3.73E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75078(10-[3-[bis(3-methylbutyl)amino]-2-hydroxypropyl]ac...)
Affinity DataEC50:  3.74E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75000(N-(2-methoxyethyl)-5-methyl-2-(4-methylphenyl)pyra...)
Affinity DataEC50:  3.77E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75094(MLS000779605 | (E)-2-Cyano-N-cyclohexyl-3-(5-morph...)
Affinity DataEC50:  3.85E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75260(MLS000948043 | SMR000620265 | 2-azanylidene-1-cycl...)
Affinity DataEC50:  3.87E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM59056((3Z)-2-(1,3-dihydrobenzimidazol-2-ylidene)-3-(3-ox...)
Affinity DataEC50:  3.93E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM55814(5-[[5-(2,5-dichlorophenyl)-1H-pyrrol-2-yl]methylid...)
Affinity DataEC50:  4.04E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74898(MLS000704256 | SMR000231279 | cid_6014635 | 4-chlo...)
Affinity DataEC50:  4.05E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM68445(MLS000084336 | SMR000048725 | cid_667374)
Affinity DataEC50:  4.07E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75116(SMR000460976 | methyl 4-cyano-1-oxopyrido[2,1-b][1...)
Affinity DataEC50:  4.11E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75070(ethyl (2E)-5-oxo-1-propyl-2-[(pyridin-3-ylcarbonyl...)
Affinity DataEC50:  4.18E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM68441(MLS000084334 | SMR000048547 | cid_667200)
Affinity DataEC50:  4.30E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM53311(cid_4264319 | 2-azanylidene-N-[2-(4-methoxyphenyl)...)
Affinity DataEC50:  4.45E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM53108(methyl 2-[[6,7-bis(oxidanyl)-2-oxidanylidene-chrom...)
Affinity DataEC50:  4.53E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75160(N-[2-[(3-cyano-6-methyl-2-quinolinyl)amino]ethyl]b...)
Affinity DataEC50:  4.66E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74979(SMR000281941 | cid_145758 | MLS000712174 | 2-(9-ac...)
Affinity DataEC50:  4.89E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM61161(SMR000152022 | MLS000564772 | N-[3-(benzenesulfony...)
Affinity DataEC50:  4.90E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74737(MLS000537373 | SMR000143811 | 5-(4-phenylmethoxyph...)
Affinity DataEC50:  4.98E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74829(cid_839240 | (Z)-2-(morpholine-4-carbonyl)-3-(5-mo...)
Affinity DataEC50:  5.08E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74544(cid_645132 | 7,8-dimethyl-2-pyrrolidin-1-ylquinoli...)
Affinity DataEC50:  5.28E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74710(8-(5-Phenyl-2-p-tolyl-pyrazolo[1,5-a]pyrimidin-7-y...)
Affinity DataEC50:  5.56E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74773(4-amino-5-(5-bromothiophene-2-carbonyl)-2-(prop-2-...)
Affinity DataEC50:  5.57E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM74570((8S,8aR)-6-azanyl-8-(7-methoxy-1,3-benzodioxol-5-y...)
Affinity DataEC50:  5.69E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM59935(SMR000219435 | MLS000589661 | (E)-3-[5-(4-morpholi...)
Affinity DataEC50:  5.73E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75097(cid_2025178 | (E)-2-cyano-3-[2-(4-methoxyphenoxy)-...)
Affinity DataEC50:  6.00E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetImportin subunit alpha-1(Human)
Johann Wolfgang Goethe University

Curated by ChEMBL
LigandPNGBDBM75096((E)-2-cyano-3-[5-(dimethylamino)-2-furanyl]-N-prop...)
Affinity DataEC50:  6.38E+3nMAssay Description:Keywords: Counterscreen, FRET assay, HTS, YIC probe, Dose response, Assay Overview: This is a fluorescence resonance energy transfer (FRET)-based b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
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