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Report error Found 353 for UniProtKB: P49288
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472541(CHEMBL273888)
Affinity DataEC50: <0.0100nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472538(CHEMBL12418)
Affinity DataEC50: <0.0100nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472540(CHEMBL12815)
Affinity DataEC50: <0.0100nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472537(CHEMBL12664)
Affinity DataEC50: <0.0100nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470712(CHEMBL417988)
Affinity DataKi:  0.0190nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50230657(CHEMBL290493)
Affinity DataKi:  0.0295nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.0324nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataEC50:  0.0370nMAssay Description:Functional activity against melatonin receptor in lightening Xenopus laevis tadpole skinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470694(CHEMBL14483)
Affinity DataKi:  0.0466nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470184(CHEMBL304203)
Affinity DataKi:  0.0500nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470711(CHEMBL14403)
Affinity DataKi:  0.0558nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50034110(Melatonin,2-Phenyl | CHEMBL15060 | N-[2-(5-Methoxy...)
Affinity DataKi:  0.0596nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50035202(N-[2-(2,7-Dimethoxy-naphthalen-1-yl)-ethyl]-propio...)
Affinity DataKi:  0.0700nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50035202(N-[2-(2,7-Dimethoxy-naphthalen-1-yl)-ethyl]-propio...)
Affinity DataKi:  0.0724nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataKi:  0.100nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataKi:  0.100nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470007(CHEMBL322269)
Affinity DataKi:  0.120nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.130nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470000(CHEMBL111599)
Affinity DataKi:  0.141nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470172(CHEMBL294517)
Affinity DataKi:  0.176nMAssay Description:Effect of compound on Melatonin receptor in chicken brain in the presence of MnCl2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.176nMAssay Description:Effect of compound on Melatonin receptor in chicken brain in the presence of MnCl2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50408556(CHEMBL37771)
Affinity DataKi:  0.182nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50231307(CHEMBL34622)
Affinity DataKi:  0.190nMAssay Description:Binding affinity towards melatonin receptor in chicken brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231291(CHEMBL421013)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470187(CHEMBL428882)
Affinity DataKi:  0.240nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231307(CHEMBL34622)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50469784(CHEMBL14975)
Affinity DataKi:  0.305nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472142(CHEMBL142343)
Affinity DataKi:  0.378nMAssay Description:Binding affinity towards melatonin receptor, determined in chicken brain membranes using [2-125I]melatoninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50472142(CHEMBL142343)
Affinity DataKi:  0.378nMAssay Description:Displacement of 2-[125I]iodomelatonin from chick brain melatonin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50212943(CHEMBL290895)
Affinity DataKi:  0.378nMAssay Description:Binding affinity towards melatonin receptor was determined using 2-[125I]iodomelatonin as radioligand in chick brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470180(CHEMBL61626)
Affinity DataKi:  0.389nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470180(CHEMBL61626)
Affinity DataKi:  0.400nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.460nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.537nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.540nMAssay Description:Inhibition of 2-[125I]- iodomelatonin from chicken brain melatonin receptorsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50035179(S 20098 | N-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-...)
Affinity DataKi:  0.540nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470174(CHEMBL62992)
Affinity DataKi:  0.540nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470174(CHEMBL62992)
Affinity DataKi:  0.550nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity towards melatonin receptor using 2-[125I]iodomelatonin as radioligand in chick brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity towards melatonin receptor, determined in chicken brain membranes using [2-125I]melatoninMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.590nMAssay Description:Displacement of 2-[125I]iodomelatonin from chick brain melatonin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2021
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity in chicken brain membranes by using [2-125I]melatonin in a competition radioligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity towards melatonin receptor in chicken brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.590nMAssay Description:Binding affinity towards melatonin receptor was determined using 2-[125I]iodomelatonin as radioligand in chick brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.670nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470172(CHEMBL294517)
Affinity DataKi:  0.676nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.676nMAssay Description:Binding affinity against chicken brain melatonin receptors using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(Chicken)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50470172(CHEMBL294517)
Affinity DataKi:  0.680nMAssay Description:Competitive binding by the displacement of 2-[125I]- Iodomelatonin binding from melatonin receptors in chicken brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
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