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Report error Found 168 of affinity data for UniProtKB/TrEMBL: P48546
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275567(CHEMBL4128194)
Affinity DataEC50:  0.189nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275569(CHEMBL4130148)
Affinity DataEC50:  114nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275578(CHEMBL4128112)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275568(CHEMBL4126738)
Affinity DataEC50:  2.03nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275546(CHEMBL4130044)
Affinity DataEC50:  177nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275593(CHEMBL4126812)
Affinity DataEC50:  0.0582nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275594(CHEMBL4130225)
Affinity DataEC50:  0.224nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275545(CHEMBL4126953)
Affinity DataEC50:  2.03nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275598(CHEMBL4126027)
Affinity DataEC50:  1.16nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275596(CHEMBL4129347)
Affinity DataEC50:  0.102nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275595(CHEMBL4127525)
Affinity DataEC50:  0.0397nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275565(CHEMBL4125912)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275566(CHEMBL4128276)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50275564(CHEMBL4128125)
Affinity DataEC50:  1.21nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50241203(exenatide | HGEGTFTSDLSKQMEEEAVRLFIEWLKNGGPSSGSPPP...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as cAMP accumulation after 30 mins by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459980(CHEMBL4227861)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459981(CHEMBL4225594)
Affinity DataEC50:  0.867nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459988(CHEMBL4227045)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459989(CHEMBL4225340)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459984(CHEMBL4225795)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459990(CHEMBL4224968)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459985(CHEMBL4226451)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459986(CHEMBL4226634)
Affinity DataEC50:  0.133nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459982(CHEMBL4226514)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459992(CHEMBL4227180)
Affinity DataEC50:  0.812nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459993(CHEMBL4229251)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459987(CHEMBL4226613)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459983(CHEMBL4224701)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50459991(CHEMBL4226185)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50597204(CHEMBL5196841)
Affinity DataEC50:  12nMAssay Description:Positive allosteric modulator activity at human GIPR expressed in HEK293 cells assessed as potentiation of intracellular cAMP accumulation incubated ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50597205(CHEMBL5184469)
Affinity DataEC50:  38nMAssay Description:Positive allosteric modulator activity at human GIPR expressed in HEK293 cells assessed as potentiation of intracellular cAMP accumulation incubated ...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50245060((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(4-trifluoromet...)
Affinity DataIC50: 12nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50171817(3-(4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluorom...)
Affinity DataIC50: 28nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50202060(3-{4-[1-(4-tert-butylphenyl)-3-(4-trifluoromethoxy...)
Affinity DataIC50: 38nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50334486(trans-4-((1-(4-tert-butylcyclohexyl)-3-(4-(trifluo...)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human GIPR expressed in CHO cells assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50566470(CHEMBL4857523)
Affinity DataIC50: 60nMAssay Description:Antagonist activity at human GIPR expressed in HEK293 cells assessed as inhibition of GIP-induced cAMP productionMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50202031(3-(4-((1-(4-cyclohexenylphenyl)-3-(3,5-dichlorophe...)
Affinity DataIC50: 64nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50245062((R)-3-{4-[3-(3-tert-Butylphenyl)-1-(4-cyclohexylph...)
Affinity DataIC50: 74nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50245099((R)-3-{4-[1-(4-Cyclohex-1-enylphenyl)-3-(2,2,4,4-t...)
Affinity DataIC50: 83nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50244457((R)-trans-3-{4-[3-(3,5-Bis(trifluoromethyl)phenyl)...)
Affinity DataIC50: 87nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50245098((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(3,5-dichloroph...)
Affinity DataIC50: 93nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50202041(trans-3-{4-[3-(3,5-bistrifluoromethylphenyl)-1-(4-...)
Affinity DataIC50: 93nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50245057((R)-trans-3-{4-[1-(4-tert-Butyl-cyclohexyl)-3-(3-m...)
Affinity DataIC50: 98nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50199497(1-(7-((2H-tetrazol-5-yl)carbamoyl)-3,4-dihydro-2H-...)
Affinity DataIC50: 117nMAssay Description:Antagonist activity at human GIP receptor transfected in CHO cells assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50199493(1-(N-((1r,4r)-4-tert-butylcyclohexyl)-2-(4-(triflu...)
Affinity DataIC50: 118nMAssay Description:Antagonist activity at human GIP receptor transfected in CHO cells assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50199498(3-(1-(1-((1r,4r)-4-tert-butylcyclohexyl)-3-(4-(tri...)
Affinity DataIC50: 132nMAssay Description:Antagonist activity at human GIP receptor transfected in CHO cells assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50244509((R)-3-{4-[1-(4-Cyclohexylphenyl)-3-(3-methoxy-5-tr...)
Affinity DataIC50: 145nMAssay Description:Binding affinity to human cloned GIPR expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50199488(3-(1-(1-((1r,4r)-4-tert-butylcyclohexyl)-3-(4-(tri...)
Affinity DataIC50: 171nMAssay Description:Antagonist activity at human GIP receptor transfected in CHO cells assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastric inhibitory polypeptide receptor(Human)
Sanofi-Aventis Deutschland

Curated by ChEMBL
LigandPNGBDBM50199491(1-(6-((2H-tetrazol-5-yl)carbamoyl)-1,2,3,4-tetrahy...)
Affinity DataIC50: 178nMAssay Description:Antagonist activity at human GIP receptor transfected in CHO cells assessed as inhibition of glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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