Compile Data Set for Download or QSAR
Report error Found 501 of affinity data for UniProtKB/TrEMBL: P46059
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50044849(CHEMBL3311308)
Affinity DataEC50: <5.01E+4nMAssay Description:Agonist activity at human PePT1 receptor expressed in HEK cells by FLIPR membrane potential/summary (Abse5) assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50088510(CHEMBL3526259)
Affinity DataKd:  2.20nMAssay Description:Activity at human recombinant PEPT1 expressed in Pichia pastoris GS115 assessed as non-saturable rate constant after 30s by dual-channel liquid scint...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169173((S)-6-Amino-2-((S)-2-amino-4-carboxy-butyrylamino)...)
Affinity DataEC50:  3.10E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169222(glycylglycine | 2-(aminoacetamido)acetic acid | Gl...)
Affinity DataEC50:  4.80E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188481(Phe-Tyr | CHEMBL378907)
Affinity DataEC50:  3.00E+4nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188483(Lys-Gly | ((S)-2,6-Diamino-hexanoylamino)-acetic a...)
Affinity DataEC50:  3.20E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188484(Gly-Gly-Gly | [2-(2-Amino-acetylamino)-acetylamino...)
Affinity DataEC50:  5.80E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50016695((2S)-2-{[(2S)-2-aminopropanoyl]amino}propanoic aci...)
Affinity DataEC50:  8.00E+4nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169199(Gly-His | 2-(2-Amino-acetylamino)-3-(3H-imidazol-4...)
Affinity DataEC50:  4.00E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188489((S)-2-Amino-N-((S)-1-carbamoyl-2-phenyl-ethyl)-3-p...)
Affinity DataEC50:  3.00E+4nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188491((glycyldehydrophenylalanine)2-(2-Amino-acetylamino...)
Affinity DataEC50:  1.30E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188492((S)-2-(2-Amino-acetylamino)-4-methyl-pentanoic aci...)
Affinity DataEC50:  1.70E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188493((S)-2-(2-Amino-acetylamino)-succinic acid | Gly-As...)
Affinity DataEC50:  5.50E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188495(Phe-Ala-NH2 | CHEMBL210616)
Affinity DataEC50:  8.50E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188485((S)-2-((S)-2-Amino-propionylamino)-3-(1H-indol-3-y...)
Affinity DataEC50:  8.00E+4nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188499(2-((S)-2-Amino-acetylamino)-3-(1H-indol-3-yl)-prop...)
Affinity DataEC50:  3.30E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188500(His-His | CHEMBL377872)
Affinity DataEC50:  3.70E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188501(Pro-Leu | 4-Methyl-2-[(pyrrolidine-2-carbonyl)-ami...)
Affinity DataEC50:  2.50E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50081840((S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyla...)
Affinity DataEC50:  6.00E+4nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50139892((S)-2-((S)-2-Amino-3-phenyl-propionylamino)-propio...)
Affinity DataEC50:  1.10E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188482(Gly-Leu-Gly | CHEMBL209341)
Affinity DataEC50:  2.10E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169127((S)-2-((S)-2-Amino-3-carboxy-propionylamino)-succi...)
Affinity DataEC50:  9.90E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188502(Asp-Gly | (S)-3-Amino-N-carboxymethyl-succinamic a...)
Affinity DataEC50:  4.40E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188507(4-Amino-4-(carboxymethyl-carbamoyl)-butyric acid |...)
Affinity DataEC50:  5.10E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188506(Val-Val-Val | CHEMBL380174)
Affinity DataEC50:  2.10E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188510(Pro-Ser | CHEMBL209083)
Affinity DataEC50:  1.60E+6nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188508(2-(2-Amino-acetylamino)-3-(4-hydroxy-phenyl)-propi...)
Affinity DataEC50:  1.40E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188511(Asp-Val | CHEMBL441685)
Affinity DataEC50:  6.90E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169129(Tyr-Ala | (S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataEC50:  1.00E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188496((S)-2-((S)-2-Amino-4-methyl-pentanoylamino)-4-meth...)
Affinity DataEC50:  8.00E+4nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188516(Gly-Sar | 2-(2-amino-N-methylacetamido)acetic acid...)
Affinity DataEC50:  5.40E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188504(Ala-Asp | CHEMBL380047)
Affinity DataEC50:  2.30E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188517(Lys-Pro | CHEMBL209032)
Affinity DataEC50:  1.90E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188486([(S)-2-Amino-3-(3H-imidazol-4-yl)-propionylamino]-...)
Affinity DataEC50:  2.80E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169141(Pro-Pro | i(S)-1-((S)-Pyrrolidine-2-carbonyl)-pyrr...)
Affinity DataEC50:  7.00E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188521((S)-2-((S)-2-Amino-3-methyl-butyrylamino)-3-methyl...)
Affinity DataEC50:  7.00E+4nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188522(Arg-Gly | CHEMBL382777)
Affinity DataEC50:  2.70E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188519([(S)-2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-...)
Affinity DataEC50:  2.40E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169160((S)-2-((S)-2-amino-3-(1H-indol-3-yl)propanamido)pr...)
Affinity DataEC50:  1.00E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169195(Pro-Asp | (S)-2-[((S)-Pyrrolidine-2-carbonyl)-amin...)
Affinity DataEC50: >5.00E+6nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188526((S)-2-[(S)-2-Amino-3-(1H-indol-3-yl)-propionylamin...)
Affinity DataEC50:  5.00E+4nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188498(Trp-Gly | [(S)-2-Amino-3-(1H-indol-3-yl)-propionyl...)
Affinity DataEC50:  2.60E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169189(Gly-Pro | 1-(2-Amino-acetyl)-pyrrolidine-2-carboxy...)
Affinity DataEC50:  1.30E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188529(Gly-Glu | 2-(2-Amino-acetylamino)-pentanedioic aci...)
Affinity DataEC50:  1.10E+6nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188531(Lys-Val | CHEMBL208094)
Affinity DataEC50:  1.40E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188514(Gln-Glu | CHEMBL210850)
Affinity DataEC50:  4.20E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188513((S)-6-Amino-2-(2-amino-acetylamino)-hexanoic acid ...)
Affinity DataEC50:  7.50E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188525(Gly-Leu-Phe | CHEMBL209670)
Affinity DataEC50:  2.80E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50188528(Gln-Gln | CHEMBL438960)
Affinity DataEC50:  1.00E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50169125(Ala-Lys | (S)-6-Amino-2-((S)-2-amino-propionylamin...)
Affinity DataEC50:  2.20E+5nMAssay Description:Activation of human PEPT1 expressed in MDCK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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