Compile Data Set for Download or QSAR
Report error Found 1227 for UniProtKB: P30872
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065451(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  3.55E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst1) expressed in hSF6 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065452(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  1.32E+4nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst1) expressed in hSF6 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065450(2-Amino-3-phenyl-N-{4-[(2S,5S,8S,14S,17R)-8,10,14-...)
Affinity DataKd:  7.08E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst1) expressed in hSF6 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKd:  4.57E+3nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst1) expressed in hSF6 cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098602(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098610(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.26E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098612(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  316nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098617(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  611nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098616(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  867nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098604(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  862nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098609(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098618(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098613(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  811nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098607(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  956nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098611(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098619(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  761nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098603(10-(4-Amino-butyl)-19-[(2-amino-3-phenyl-propionyl...)
Affinity DataKd:  378nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098606(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  653nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098615(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098614(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  622nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098605(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098608(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst1)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423297(Obelin | CHEMBL251541)
Affinity DataKd:  10nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  1.20nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423464(CHEMBL252231)
Affinity DataKd:  1.95E+3nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423458(CHEMBL252232)
Affinity DataKd:  501nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423465(ERGOLINE)
Affinity DataKd:  1.70nMAssay Description:Binding affinity to human recombinant sst1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50294254((4R,7S,10S,13R,16S,19R)-19-((R)-2-amino-3-(4-hydro...)
Affinity DataEC50:  0.370nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50294252((4R,7S,10S,13R,16S,19R)-19-amino-N-((2S,3R)-1-amin...)
Affinity DataEC50:  3.90nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50294231((4R,7S,10S,13S,16S,19S,22R,25S,28S,31S,34R)-22-((1...)
Affinity DataEC50:  33nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50294255((4R,7S,10S,13S,16S,19S,22S,25S,28S,31S,34S,37R)-31...)
Affinity DataEC50:  0.930nMAssay Description:Agonist activity at human sst1 receptor expressed in Chinese hamster CCL39 cells by luciferase reporter gene assay relative to somatostatin-14More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50473329(CHEMBL311789)
Affinity DataKd:  1.32E+4nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKd:  0.832nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50473330(CHEMBL309948)
Affinity DataKd: <1.00E+5nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50473331(CHEMBL420948)
Affinity DataKd: <1.00E+5nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50192018(CHEMBL3350037)
Affinity DataKd:  389nMAssay Description:Binding assay at human somatostatin receptor 1 (hsst1) expressed in CCL-39 cells using LTT-CST-14-(Tyr10) as radioligand.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50537061(CHEMBL4527856)
Affinity DataKd:  310nMAssay Description:Displacement of [125I]somatostatin from human SSTR1 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50537072(CHEMBL440072)
Affinity DataKd:  0.290nMAssay Description:Displacement of [125I]somatostatin from human SSTR1 expressed in CHO-K1 cell membranes after 120 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50546560(CHEMBL4778342)
Affinity DataEC50:  316nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50592194(CHEMBL5195355)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50592196(CHEMBL5174433)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50592194(CHEMBL5195355)
Affinity DataEC50: <1.00E+3nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50592196(CHEMBL5174433)
Affinity DataEC50: <1.00E+3nMAssay Description:Agonist activity at human SST1More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50294254((4R,7S,10S,13R,16S,19R)-19-((R)-2-amino-3-(4-hydro...)
Affinity DataIC50: 0.190nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst1 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476134(CHEMBL437296)
Affinity DataIC50: 0.200nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476138(CHEMBL376485)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50212467(Sandostatinm)
Affinity DataIC50: 0.460nMAssay Description:Compound was tested for free energy of binding against somatostatin receptorMore data for this Ligand-Target Pair
In DepthDetails

TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476142(CHEMBL376484)
Affinity DataIC50: 0.5nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1/2/3/4/5(Human)
Diatide Research Laboaratories

Curated by ChEMBL
LigandPNGBDBM50476141(CHEMBL426548)
Affinity DataIC50: 0.640nMAssay Description:Displacement of [125I-Tyr-11]-SRIF from SSTR of human NCI-H69 cell membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSomatostatin receptor type 1(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50294232((4R,7S,10S,13R,16S,19R)-19-((S)-2-amino-3-(4-hydro...)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [125I]LTT-SRIF-28 from human sst1 receptor by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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