TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 193nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 200nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 219nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 219nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 241nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 246nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 246nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 251nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 300nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 310nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 327nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 333nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 344nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 368nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 420nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 450nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 460nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 700nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 700nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 900nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 900nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 900nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 930nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.29E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 assessed as reduction in NADPH production using 4-NBA and NADP+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of human ALDH3A1 assessed as NADH formation using propionaldehyde as substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMpH: 7.5Assay Description:IC50 values were determined for CB29 and its analogs using propionaldehyde as the substrate for ALDH1A1 and ALDH2 or benzaldehyde as the substrate fo...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human ALDH3A1-mediated benzaldehyde oxidation preincubated for 1 min followed by substrate addition by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.52E+3nMAssay Description:Inhibition of ALDH3A1 (unknown origin) assessed as NADH formation using 4-nitrobenzaldehyde as substrateMore data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of N-terminal-His6 tagged recombinant human ALDH3A1 assessed as reduction in NADPH production using 4-NBA and NADP+ as substrate by fluori...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
TargetAldehyde dehydrogenase, dimeric NADP-preferring(Human)
The Pennsylvania State University College of Medicine
Curated by ChEMBL
The Pennsylvania State University College of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of full length human ALDH3A1 expressed in Escherichia coli BL21 (DE3) using benzaldehyde as substrate preincubated for 2 mins followed by ...More data for this Ligand-Target Pair
