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Report error Found 635 for UniProtKB: P30553
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50026690(2-[2-(2-{2-[2-{2-[2-(2-Amino-3-phenyl-propionylami...)
Affinity DataEC50:  1.00E+3nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056453(3-(2-{[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl...)
Affinity DataEC50:  1.5nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataEC50:  1nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50024317(Tetragastrin | CHEMBL120632 | 3-{2-[2-Amino-3-(1H-...)
Affinity DataEC50:  1.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataEC50:  1.5nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataEC50:  0.400nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092401(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[2-(1H-indol-3-y...)
Affinity DataEC50:  7nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092391(3-(2-{[2-(2-Carbamoyl-acetylamino)-3-(1H-indol-3-y...)
Affinity DataEC50:  1.64nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092399(3-(2-{[2-(2-Benzylcarbamoyl-acetylamino)-3-(1H-ind...)
Affinity DataEC50:  3.30nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092389(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataEC50:  2nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092395(3-{2-[2-{[9-tert-Butoxycarbonylamino-3-butyl-2,5,8...)
Affinity DataEC50:  17nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092384(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[2-(3-carboxy...)
Affinity DataEC50:  1.5nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092408(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{[3-(1H-indol-...)
Affinity DataEC50:  0.560nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.630nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50092393(3-(2-{[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-su...)
Affinity DataEC50:  3.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50348752(CHEMBL1807150)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50348756(CHEMBL1806532)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50348753(CHEMBL1806528)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056448(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[(2R,5R)-2-(1H-i...)
Affinity DataEC50:  4nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056449(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[(2R,5R)-2-(1H-i...)
Affinity DataEC50:  7nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.630nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056455(N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[(5R,8R)-8-(1H-i...)
Affinity DataEC50:  7nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50026690(2-[2-(2-{2-[2-{2-[2-(2-Amino-3-phenyl-propionylami...)
Affinity DataKd:  1.40nMAssay Description:Tested in vitro by the gastrin binding assay for the competitive binding with iodinated gastrin for the gastrin receptors in AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50037873(CBS-2 | CHEMBL341130)
Affinity DataEC50:  2.00E+5nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50549228(CHEMBL4758706)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50549227(CHEMBL4759105)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50549226(CHEMBL4795913)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50286892(1-[(R)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.0700nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056102(YF-476 | 1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo...)
Affinity DataIC50: 0.100nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50286884(1-{1-[2-(1-Methyl-cyclopentyl)-2-oxo-ethyl]-2-oxo-...)
Affinity DataIC50: 0.100nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056099(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056093(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056103(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50286903(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-2...)
Affinity DataIC50: 0.120nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50286897(1-[2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-2-yl-...)
Affinity DataIC50: 0.130nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056092(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50: 0.140nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056091(1-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-2,3...)
Affinity DataIC50: 0.160nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056089(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.170nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056095(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50056098(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50: 0.210nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50286882(1-[(S)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.230nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50286882(1-[(S)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.230nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50288462((R)-2-{(2R,5S)-2-[(R)-3-((R)-2-Carboxy-pyrrolidine...)
Affinity DataIC50: 0.25nMAssay Description:Tested for displacement of [125I]-CCK-8 from Gastrin/Cholecystokinin type B receptor in rat brain.More data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50286886(1-[1-(3-Cyclohexyl-2-oxo-propyl)-2-oxo-5-phenyl-2,...)
Affinity DataIC50: 0.280nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

TargetGastrin/cholecystokinin type B receptor(Rat)
National Cancer Institute-Frederick

Curated by ChEMBL
LigandPNGBDBM50286888(1-{1-[2-(1-Methyl-cyclohexyl)-2-oxo-ethyl]-2-oxo-5...)
Affinity DataIC50: 0.380nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In DepthDetails Article

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