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TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM21190(CHEMBL113142 | 4-(2-{[5-amino-2-(furan-2-yl)-[1,2,...)
Affinity DataKd:  0.330nMAssay Description:The membranes prepared from Flp-In HEK cells transfected with adenosine receptors were used in binding assays. Nonspecific binding was determined in ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50454426(CHEMBL2304158)
Affinity DataEC50:  576nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50454422(CHEMBL2113525)
Affinity DataEC50: >1nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM21220(CHEMBL464859 | N-Ethylcarboxamidoadenosine | Adeno...)
Affinity DataEC50:  394nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50454423(CHEMBL2113528)
Affinity DataEC50:  594nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50454425(CHEMBL2113526)
Affinity DataEC50:  194nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50454421(CHEMBL2113529)
Affinity DataEC50:  1nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50119168((2R,3R,4S,5R)-2-(6-Amino-2-hex-1-ynyl-purin-9-yl)-...)
Affinity DataEC50:  79nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50454091(CHEMBL2113450)
Affinity DataEC50:  497nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50205705((2S,3S,4R)-5-((R)-6-amino-2-phenylethynyl-9H-purin...)
Affinity DataEC50: >1nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453224(CHEMBL410873 | 2-(l-hexyn-l-yl)-adenosine-5'-N-met...)
Affinity DataEC50:  596nMAssay Description:Vasorelaxation as Adenosine A2A receptor activity in rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369101(CHEMBL604647)
Affinity DataEC50:  2.99E+3nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369084(CHEMBL604440)
Affinity DataEC50:  531nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453224(CHEMBL410873 | 2-(l-hexyn-l-yl)-adenosine-5'-N-met...)
Affinity DataEC50:  596nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369098(CHEMBL605055)
Affinity DataEC50:  3.57E+3nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369089(CHEMBL605473)
Affinity DataEC50:  1.30E+3nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369092(CHEMBL604234)
Affinity DataEC50:  1.21E+3nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50454091(CHEMBL2113450)
Affinity DataEC50:  497nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453346(CHEMBL2113449)
Affinity DataEC50:  440nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369108(CHEMBL605691)
Affinity DataEC50: >10nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369099(CHEMBL605690)
Affinity DataEC50:  210nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369102(CHEMBL605265)
Affinity DataEC50:  29nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369090(CHEMBL605478)
Affinity DataEC50:  1.35E+3nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50205705((2S,3S,4R)-5-((R)-6-amino-2-phenylethynyl-9H-purin...)
Affinity DataEC50:  1.50E+3nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369096(CHEMBL605264)
Affinity DataEC50:  6.52E+3nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50085658(2-Cl-CPA | CHEMBL284969 | 2-chloro-N6-cyclopentyla...)
Affinity DataEC50: >10nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369095(CHEMBL605057)
Affinity DataEC50:  468nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369109(CHEMBL605056)
Affinity DataEC50: >10nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369097(CHEMBL604851)
Affinity DataEC50:  406nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369111(CHEMBL604849)
Affinity DataEC50:  3.48E+3nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453792(CHEMBL2113560)
Affinity DataEC50:  677nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453793(CHEMBL2113559)
Affinity DataEC50:  281nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453789(CHEMBL2113564)
Affinity DataEC50:  195nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453790(CHEMBL2113563)
Affinity DataEC50:  269nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM35804(3-(4-{2-[6-Amino-9-((2R,3R,4S,5S)-5-ethylcarbamoyl...)
Affinity DataEC50:  115nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453796(CHEMBL2113552)
Affinity DataEC50:  704nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453795(CHEMBL2113553)
Affinity DataEC50:  728nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453794(CHEMBL2113554)
Affinity DataEC50:  529nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453787(CHEMBL2113556)
Affinity DataEC50:  482nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453791(CHEMBL2113555)
Affinity DataEC50:  800nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50453788(CHEMBL2113558)
Affinity DataEC50:  638nMAssay Description:Functional activity at Adenosine A2A receptor as vasorelaxation of rat aortaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50150766((2R,3R,4S,5R)-2-[6-Amino-2-((S)-1-hydroxymethyl-2-...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at adenosine receptor A2a in isolated rat aorta assessed as efficacyMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50048466(CHEMBL17127 | SCH58261 | 2-(furan-2-yl)-7-phenethy...)
Affinity DataKd:  0.700nMAssay Description:Binding affinity to adenosine receptor A2a in rat striatumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50094037(SCH-442416 | 2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-...)
Affinity DataKd:  0.0480nMAssay Description:Binding affinity to adenosine receptor A2a in rat striatumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50095602(4-[3-(8-Cyclopentyl-2,6-dioxo-1-propyl-1,2,6,7-tet...)
Affinity DataKd:  0.340nMAssay Description:Dissociation constant of [3H]ZM-241385 binding to adenosine A2A receptor(AR)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50039676(4-Fluorosulfonyl-benzoic acid 3-(8-cyclopentyl-2,6...)
Affinity DataKd:  0.230nMAssay Description:Dissociation constant of [3H]ZM-241385 binding to adenosine A2A receptor(AR)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50095604(4-[3-(8-Cyclohexyl-2,6-dioxo-1-propyl-1,2,6,7-tetr...)
Affinity DataKd:  0.270nMAssay Description:Dissociation constant of [3H]ZM-241385 binding to adenosine A2A receptor(AR)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369087(CHEMBL605065)
Affinity DataEC50:  0.00800nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM35804(3-(4-{2-[6-Amino-9-((2R,3R,4S,5S)-5-ethylcarbamoyl...)
Affinity DataEC50:  115nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetAdenosine receptor A2a(Rat)
Neuroscience

LigandPNGBDBM50369091(CHEMBL604019)
Affinity DataEC50:  302nMAssay Description:Functional activity against adenosine A2a receptor from rat aorta.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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