Compile Data Set for Download or QSAR
Report error Found 883 of affinity data for UniProtKB/TrEMBL: P28190
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50008405(CHEMBL27041 | 2-(4-(2,6-dioxo-1,3-dipropyl-2,3,6,7...)
Affinity DataKd:  17nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of [125-I]-labeled aminobenzyl adenosine binding to bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023391({4-[1-(4-Amino-3-iodo-benzyl)-2,6-dioxo-3-propyl-2...)
Affinity DataKd:  160nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023392({4-[3-(4-Amino-benzyl)-2,6-dioxo-1-propyl-2,3,6,9-...)
Affinity DataKd:  32nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023396((4-{3-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-1-propy...)
Affinity DataKd:  60nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82558(NSC_163889 | CAS_163889 | CHEMBL355370 | I-ABOPX)
Affinity DataKd:  37nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023400((4-{1,3-Bis-[2-(4-amino-phenyl)-ethyl]-2,6-dioxo-2...)
Affinity DataKd:  3.59E+3nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023401((4-{1-[2-(4-Amino-phenyl)-ethyl]-2,6-dioxo-3-propy...)
Affinity DataKd:  2.30E+3nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023395((4-{3-[2-(4-Azido-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  24nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023394((4-{1-[2-(4-Azido-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  2.86E+3nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of [125-I]-labeled aminobenzyl adenosine binding to bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023398((4-{3-[2-(4-Amino-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  29nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023390({4-[1-(4-Amino-benzyl)-2,6-dioxo-3-propyl-2,3,6,9-...)
Affinity DataKd:  44nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023397({4-[1-(4-Azido-3-iodo-benzyl)-2,6-dioxo-3-propyl-2...)
Affinity DataKd:  960nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of [125-I]-labeled aminobenzyl adenosine binding to bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023402((4-{1-[2-(4-Amino-3-iodo-phenyl)-ethyl]-2,6-dioxo-...)
Affinity DataKd:  3.10E+3nMAssay Description:Displacement of [125-I]-labeled aminobenzyl adenosine binding to adenosine A1 receptor of bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50023399({4-[3-(4-Azido-3-iodo-benzyl)-2,6-dioxo-1-propyl-2...)
Affinity DataKd:  55nMAssay Description:Binding affinity for adenosine A1 receptor as inhibition of [125-I]-labeled aminobenzyl adenosine binding to bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020986(CHEMBL11002 | N-(2-Dimethylamino-ethyl)-4-(2,6-dio...)
Affinity DataIC50: 0.0500nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82013(NSC_92411 | 8-(2-Amino-4-chlorophenyl)-1,3-dipropy...)
Affinity DataIC50: 0.0500nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021010(CHEMBL545362 | N-(4-Dimethylamino-butyl)-4-(2,6-di...)
Affinity DataIC50: 0.0700nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021008(CHEMBL11036 | N-(3-Dimethylamino-propyl)-4-(2,6-di...)
Affinity DataIC50: 0.0800nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021004(CHEMBL415971 | 8-(2,4-Diaminophenyl)-1,3-dipropylx...)
Affinity DataIC50: 0.150nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020979(CHEMBL11173 | 4-[4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7...)
Affinity DataIC50: 0.240nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020974(CHEMBL268964 | 8-(2-Amino-4-chloro-phenyl)-1,3-dim...)
Affinity DataIC50: 0.350nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82025(8-Phenyl-1,3-dipropyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataIC50: 0.700nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020976(CHEMBL11104 | 8-(2-Amino-phenyl)-1,3-dipropyl-3,7-...)
Affinity DataIC50: 0.75nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020981(CHEMBL275263 | 8-(4-Bromo-phenyl)-1,3-dimethyl-3,7...)
Affinity DataIC50: 0.75nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020961(CHEMBL11127 | 8-(4-Ethyl-phenyl)-1,3-dimethyl-3,7-...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020963(CHEMBL11410 | 1,3-Diallyl-8-(2-amino-4-chloro-phen...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020966(CHEMBL10995 | 8-(2-Amino-4-chloro-phenyl)-1,3-diet...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020969(CHEMBL268026 | 1,3-Dimethyl-8-p-tolyl-3,7-dihydro-...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020988(CHEMBL269218 | 8-(4-Chlorophenyl)theophylline | 8-...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021002(CHEMBL11027 | 4-(1,3-Diethyl-2,6-dioxo-2,3,6,7-tet...)
Affinity DataIC50: 0.910nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021016(CHEMBL11342 | 8-(4-Bromo-phenyl)-1,3-diethyl-3,7-d...)
Affinity DataIC50: 1nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020997(CHEMBL11271 | 8-(4-Iodo-phenyl)-1,3-dimethyl-3,7-d...)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020965(8-(4-methoxyphenyl)-1,3-dimethyl-1H-purine-2,6(3H,...)
Affinity DataIC50: 1.5nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020967(CHEMBL10913 | 4-(1,3-Diethyl-2,6-dioxo-2,3,6,7-tet...)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020972(CHEMBL11332 | 8-(4-Dimethylamino-phenyl)-1,3-dimet...)
Affinity DataIC50: 1.80nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020852(CHEMBL276830 | 8-(4-Aminophenyl)theophylline | 8-(...)
Affinity DataIC50: 1.80nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021000(CHEMBL276603 | 1-Allyl-8-(2-amino-4-chloro-phenyl)...)
Affinity DataIC50: 2nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82012(8-(4-Hydroxy-phenyl)-1,3-dimethyl-3,7-dihydro-puri...)
Affinity DataIC50: 2nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021017(CHEMBL268701 | 8-(4-Ethoxy-phenyl)-1,3-dimethyl-3,...)
Affinity DataIC50: 2nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021018(CHEMBL11163 | 1,3-Dimethyl-8-(4-methylsulfanyl-phe...)
Affinity DataIC50: 2nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50018157(CHEMBL9069 | 1-Methyl-8-phenyl-3,7-dihydro-purine-...)
Affinity DataIC50: 2.5nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM38453(1,3-dimethyl-8-(4-propan-2-ylphenyl)-7H-purine-2,6...)
Affinity DataIC50: 2.5nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021015(CHEMBL11037 | 8-(2-Amino-4-nitro-phenyl)-1,3-dimet...)
Affinity DataIC50: 2.5nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM82015(1,3-Dimethyl-8-phenyl-3,9-dihydro-purine-2,6-dione...)
Affinity DataIC50: 3nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM81971(1,3-Diethyl-8-phenyl-3,7-dihydro-purine-2,6-dione ...)
Affinity DataIC50: 3nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020998(CHEMBL273295 | 8-(4-Dimethylamino-phenyl)-1,3-diet...)
Affinity DataIC50: 3.30nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020987(CHEMBL276201 | 4-(1,3-Diethyl-2,6-dioxo-2,3,6,7-te...)
Affinity DataIC50: 3.30nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50018162(CHEMBL418333 | 4-(2,6-Dioxo-1,3-dipropyl-2,3,6,7-t...)
Affinity DataIC50: 3.40nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50020996(CHEMBL276401 | 8-Biphenyl-4-yl-1,3-dimethyl-3,7-di...)
Affinity DataIC50: 3.5nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAdenosine receptor A1(Bovine)
University of Virginia School of Medicine

Curated by ChEMBL
LigandPNGBDBM50021011(CHEMBL273267 | 8-(4-Fluoro-phenyl)-1,3-dimethyl-3,...)
Affinity DataIC50: 3.5nMAssay Description:Binding affinity against bovine brain adenosine A1 receptor by using N6-[3H]- cyclohexyladenosineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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