Compile Data Set for Download or QSAR
Report error Found 53 of affinity data for UniProtKB/TrEMBL: P25102
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKd:  1.17E+5nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article

TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM22881(5-(2-aminoethyl)-4-methyl-1,3-thiazol-2-amine | CH...)
Affinity DataKd:  1.15E+4nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PDB3D3D Structure (crystal)
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000964(CHEMBL3228804)
Affinity DataEC50:  1.60E+5nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000963(CHEMBL3228805)
Affinity DataEC50:  9.10E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000962(CHEMBL3228816)
Affinity DataEC50:  7.70E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000961(CHEMBL3228802)
Affinity DataEC50:  5.00E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000960(CHEMBL3228814)
Affinity DataEC50:  3.70E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000959(CHEMBL3228801)
Affinity DataEC50:  3.50E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000958(CHEMBL3228800)
Affinity DataEC50:  2.70E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000957(CHEMBL3228796)
Affinity DataEC50:  1.90E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000956(CHEMBL3228818)
Affinity DataEC50:  1.90E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000955(CHEMBL3228795)
Affinity DataEC50:  1.60E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000954(CHEMBL3228820)
Affinity DataEC50:  1.40E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000952(CHEMBL3228791)
Affinity DataEC50:  9.50E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000444(CHEMBL282206 | CHEMBL3228808)
Affinity DataEC50:  5.50E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000443(CHEMBL280584 | CHEMBL3228799)
Affinity DataEC50:  5.30E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000411(CHEMBL3228809)
Affinity DataEC50:  4.60E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000408(CHEMBL3228806)
Affinity DataEC50:  4.00E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000405(CHEMBL92526 | CHEMBL3228819)
Affinity DataEC50:  4.30E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000391(CHEMBL3228792)
Affinity DataEC50:  3.20E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000385(CHEMBL3228793)
Affinity DataEC50:  2.30E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000382(SK&F-92058 | CHEBI:6896 | METIAMIDE)
Affinity DataEC50:  1.10E+3nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000348(CHEMBL3228794)
Affinity DataEC50:  590nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM22882(5-(2-aminoethyl)-4-methyl-1,3-selenazol-2-amine | ...)
Affinity DataKd:  9.77E+3nMAssay Description:Affinity to the Histamine H2 receptor was determined expressed in CHO cell using [125I]iodoaminopotentidine as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article

TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000953(CHEMBL3228807)
Affinity DataEC50:  1.10E+4nMAssay Description:Antagonist activity at histamine H2 receptor in Charles River rat assessed as inhibition of histamine-mediated electrically stimulated uterine contra...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026279(3-{2-[2-(2-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026297(4-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026288(3-{2-[2-(2-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026298(3-{2-[2-(2-tert-Butoxycarbonylamino-acetylamino)-3...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026282(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026283(1-(2-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026284(2-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026299(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026286(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026291(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026295(3-{2-[2-Benzyloxycarbonylamino-3-(1H-indol-3-yl)-p...)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026296(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50367238(CHEMBL1790763)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026290(3-{2-[2-(2-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026292(2-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026280(2-{2-[2-(2-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataIC50: 7.00E+4nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026281(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026293(3-({1-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026294([1-[1-(1-Carbamoyl-ethylcarbamoyl)-3-methyl-butylc...)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50144035((S)-2-(4-Chloro-benzoylamino)-3-(1H-indol-3-yl)-pr...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026285(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50014888(CHEMBL316561 | 4-Benzoylamino-4-dipropylcarbamoyl-...)
Affinity DataIC50: 2.50E+6nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50026287(3-{2-[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl)...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against binding of [125I](Nle11)-HG-13 to Histamine H2 receptor in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM7966([3H]histamine | 2-(1H-imidazol-4-yl)ethan-1-amine ...)
Affinity DataKi:  17nMMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetHistamine H2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50404029(CHEMBL45728)
Affinity DataKi: >100nMAssay Description:Displacement of [125I]-aminopotentidine from rat H2R expressed in human COS7 cells incubated for 90 mins gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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