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Report error Found 105 of affinity data for UniProtKB/TrEMBL: P21729
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe-...)
Affinity DataIC50: 0.00100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(cyclopropylbenzene(CO)His-Trp-Ala-Val-DAla-His-DPr...)
Affinity DataIC50: 0.0300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040325(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)DPhe...)
Affinity DataIC50: 0.0380nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040299(cyclopropylbenzene(CO)His-Trp-Ala-Val-DAla-His-DPr...)
Affinity DataIC50: 0.0490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040307(1-naphthyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50: 0.0500nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.0500nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50: 0.0790nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.100nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 0.160nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040315((CH3)2PhC(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe...)
Affinity DataIC50: 0.180nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040317(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Phe-...)
Affinity DataIC50: 0.220nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040301(4-OHPhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 0.230nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040312(2-tetrahydronaphthyl(CO)His-Trp-Ala-Val-DAla-His-D...)
Affinity DataIC50: 0.300nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040320(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Tyr-...)
Affinity DataIC50: 0.330nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407275(CHEMBL2112786)
Affinity DataIC50: 0.490nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040316(3-isoquinolyl(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 0.570nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50: 0.600nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040324(PhCH2CH2(CO)His-(BzthAla)-Ala-Val-DAla-His-Pro(psi...)
Affinity DataIC50: 0.75nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040310(3-CF3PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi...)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407276(CHEMBL2111952)
Affinity DataIC50: 1nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012313(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040314((CH3)2PhCCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 1.20nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407273(CHEMBL2111953)
Affinity DataIC50: 1.30nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012318(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012306(CHEMBL274874 | Ac-His-Trp-Ala-Val-Gly-His-Leu-Met-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012304(2-{2-[2-[2-(2,2-Dimethyl-propionylamino)-3-(3H-imi...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040323(phenothiazoneCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DP...)
Affinity DataIC50: 1.90nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012317(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040308(2-aminoPhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)...)
Affinity DataIC50: 2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040298(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)D2Na...)
Affinity DataIC50: 2nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012311(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012307(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012308(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012318(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 3nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)
Affinity DataIC50: 3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50407277(CHEMBL2112785)
Affinity DataIC50: 3nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012309(CHEMBL263873 | Ac-His-Trp-Ala-Val-D-Ala-His-Leu-Me...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012297(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040319(4-CF3PhCH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)Ph...)
Affinity DataIC50: 3.70nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012300(2-[2-[2-(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-y...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012317(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 4nMAssay Description:Compound was evaluated for mitogenic inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012314(CHEMBL440986 | (CH3)CCO-His-Trp-Ala-Val-Gly-His-Le...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012312(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50012319(2-{2-[2-[2-Acetylamino-3-(3H-imidazol-4-yl)-propio...)
Affinity DataIC50: 5nMAssay Description:Inhibition against Swiss 3T3 murine fibroblast cells.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040298(PhCH2CH2(CO)His-Trp-Ala-Val-DAla-His-DPro(psi)D2Na...)
Affinity DataIC50: 5nMAssay Description:The ability of the peptide to inhibit the binding of 50 pM [125I]gastrin releasing peptide to intact S-3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetGastrin-releasing peptide receptor(Mouse)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50040304(PhCH2CH2(CO)ThiAla-Trp-Ala-Val-DAla-His-DPro(psi)P...)
Affinity DataIC50: 5.60nMAssay Description:Ability of peptide to inhibit binding of 10 pM [125I]gastrin releasing peptide to S-3T3 cell membrane.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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