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Report error Found 4 of affinity data for UniProtKB/TrEMBL: P20291
TargetArachidonate 5-lipoxygenase-activating protein(Rat)
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052018(MK-591 | Sodium; 3-[3-tert-butylsulfanyl-1-(4-chlo...)
Affinity DataIC50: 10nMAssay Description:Inhibition of FLAP in rat whole blood assessed as inhibition of calcium ionophore A23187-induced LTB4 production preincubated for 4 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Rat)
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50359080(CHEMBL1922660)
Affinity DataIC50: 16nMAssay Description:Inhibition of FLAP in rat whole blood assessed as inhibition of calcium ionophore A23187-induced LTB4 production preincubated for 4 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Rat)
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50052018(MK-591 | Sodium; 3-[3-tert-butylsulfanyl-1-(4-chlo...)
Affinity DataIC50: 117nMAssay Description:Inhibition of FLAP in rat whole blood assessed as inhibition of calcium ionophore A23187-induced LTB4 production preincubated for 15 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArachidonate 5-lipoxygenase-activating protein(Rat)
Amira Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50359080(CHEMBL1922660)
Affinity DataIC50: 239nMAssay Description:Inhibition of FLAP in rat whole blood assessed as inhibition of calcium ionophore A23187-induced LTB4 production preincubated for 15 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed