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Report error Found 674 of affinity data for UniProtKB/TrEMBL: P15144
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 1nMAssay Description:Inhibition of APN (unknown origin) using Ala-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50570849(CHEMBL4854733)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50570850(CHEMBL4877339)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50076744(CHEMBL3416733)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50570851(CHEMBL4853049)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50457479(CHEMBL1159812)
Affinity DataIC50: 11nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50457468(CHEMBL4216928)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50457471(CHEMBL1159811)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50457478(CHEMBL4208547)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50368599(CHEMBL1159809)
Affinity DataIC50: 20nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50368598(CHEMBL1159810)
Affinity DataIC50: 21nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50457469(CHEMBL4213478)
Affinity DataIC50: 25nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50131276(N-(3-{4-[3-(7-Chloro-quinolin-4-ylamino)-propyl]-p...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against mammalian Aminopeptidase N (APN)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50036828(1-Mercaptomethyl-2-phenyl-ethyl-ammonium | 2-Amino...)
Affinity DataIC50: 30nMAssay Description:Inhibitory potency against aminopeptidase N (APN)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50457470(CHEMBL4204214)
Affinity DataIC50: 40nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50144944(CHEMBL3764919)
Affinity DataIC50: 120nMAssay Description:Inhibition of APN in human ES2 cells preincubated for 5 mins before L-leu-p-nitroanilide substrate addition for 1 hr by photometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50457473(CHEMBL4209822)
Affinity DataIC50: 190nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50457466(CHEMBL4206158)
Affinity DataIC50: 220nMAssay Description:Inhibition of APN (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50570847(CHEMBL4863168)
Affinity DataIC50: 224nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50570847(CHEMBL4863168)
Affinity DataIC50: 230nMAssay Description:Inhibition of APN (unknown origin) using A-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50204146(1-amino-2-phenylethyl(1-hydroxy-3-phenylpropyl)pho...)
Affinity DataIC50: 240nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50277159(CHEMBL4169814)
Affinity DataIC50: 270nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged APN (Lys69 to Lys967 residues) using Ala-AMC as substrate measured for 30 mins by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50144931(CHEMBL3764432)
Affinity DataIC50: 280nMAssay Description:Inhibition of APN in human ES2 cells preincubated for 5 mins before L-leu-p-nitroanilide substrate addition for 1 hr by photometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50277156(CHEMBL4165328)
Affinity DataIC50: 280nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged APN (Lys69 to Lys967 residues) using Ala-AMC as substrate measured for 30 mins by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50517754(CHEMBL4456660)
Affinity DataIC50: 390nMAssay Description:Inhibition of APN on human ES-2 cell surface using L-Leu-p-nitroanilide as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50089194(CHEMBL308333 | N*4*-Hydroxy-N*1*-[1-(2-hydroxymeth...)
Affinity DataIC50: 400nMAssay Description:Competitive inhibition of aminopeptidase-M (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50121710(PIQ-22 | 2-(2,6-Diethyl-phenyl)-4H-isoquinoline-1,...)
Affinity DataIC50: 409nMAssay Description:Inhibitory activity against aminopeptidase N assayed by the L-Ala-MCA method.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50400532(CHEMBL2204959)
Affinity DataIC50: 420nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50277140(CHEMBL3244800)
Affinity DataIC50: 420nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged APN (Lys69 to Lys967 residues) using Ala-AMC as substrate measured for 30 mins by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50400529(CHEMBL2204943)
Affinity DataIC50: 480nMAssay Description:Inhibition of APN in human ES2 cell surface assessed as inhibition of L-Leu-p-nitroanilide substrate hydrolysis incubated for 5 mins before substrate...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50204160(alpha1-(1-amino-2-methylpropane)-alpha2-(1-hydroxy...)
Affinity DataIC50: 500nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50382508(CHEMBL2022234)
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant AP-N ectopeptidase activity using alanine-MCA as substrate preincubated for 10 mins with substrate by fluorimetric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50382512(CHEMBL2022238)
Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant AP-N ectopeptidase activity using alanine-MCA as substrate preincubated for 10 mins with substrate by fluorimetric an...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50204163(alpha1-(1-amino-3-methylbutane)-alpha2-(carbamoylp...)
Affinity DataIC50: 530nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50430635(CHEMBL2332525)
Affinity DataIC50: 530nMAssay Description:Inhibition of aminopeptidase N in human ES2 cells using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50204159(alpha1-(1-amino-1-phenylmethane)-alpha2-(1-hydroxy...)
Affinity DataIC50: 550nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50204161(bis-alpha-(1-amino-1-phenylmethane)phosphinic acid...)
Affinity DataIC50: 600nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50430634(CHEMBL2332526)
Affinity DataIC50: 610nMAssay Description:Inhibition of aminopeptidase N in human ES2 cells using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50517756(CHEMBL4469933)
Affinity DataIC50: 620nMAssay Description:Inhibition of APN on human ES-2 cell surface using L-Leu-p-nitroanilide as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50430632(CHEMBL2332518)
Affinity DataIC50: 650nMAssay Description:Inhibition of aminopeptidase N in human ES2 cells using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50517752(CHEMBL4549692)
Affinity DataIC50: 650nMAssay Description:Inhibition of APN on human ES-2 cell surface using L-Leu-p-nitroanilide as substrate after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50277143(CHR 2797 | CHR-2797 | Tosedostat)
Affinity DataIC50: 680nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged APN (Lys69 to Lys967 residues) using Ala-AMC as substrate measured for 30 mins by fluorescenc...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50430633(CHEMBL2332527)
Affinity DataIC50: 700nMAssay Description:Inhibition of aminopeptidase N in human ES2 cells using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50204157(alpha1-(1-amino-1-phenylmethane)-alpha2-(1-amino-3...)
Affinity DataIC50: 710nMAssay Description:Inhibition of APNMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50430631(CHEMBL2332519)
Affinity DataIC50: 730nMAssay Description:Inhibition of aminopeptidase N in human ES2 cells using L-leu-p-nitroanilide as substrate incubated for 5 mins prior to substrate addition measured a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAminopeptidase N(Human)
Sanofi

Curated by ChEMBL
LigandPNGBDBM50275185(CHEMBL4125687)
Affinity DataIC50: 740nMAssay Description:Inhibition of APN in human ES2 cells using L-Leu-pnitroanilide as substrate pretreated for 5 mins followed by substrate addition measured after 1 hrMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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