TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 2.80E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 5.00E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 300nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 1.10E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 400nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 2.80E+4nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 500nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 100nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 800nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 1.70E+4nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 1.30E+3nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 240nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 2.60E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 2.40E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataKd: 2.60E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as glucose uptake by measuring ATP incubated for 15 mins by CellTiter-Glo Luminescent Cell...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Inhibition of GLUT1 in human wild-type DLD1 cells assessed as reduction in ATP level measured after 90 mins by Celltiter-glo luminescent assayMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 37nMAssay Description:Inhibition of GLUT1 in human wild-type DLD1 cells assessed as reduction in ATP level measured after 90 mins by Celltiter-glo luminescent assayMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inhibition of GLUT1 in human wild-type DLD1 cells assessed as reduction in ATP level measured after 90 mins by Celltiter-glo luminescent assayMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of GLUT1 in human wild-type DLD1 cells assessed as reduction in ATP level measured after 90 mins by Celltiter-glo luminescent assayMore data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration
Curated by ChEMBL
Food and Drug Administration
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:HT1080 cells (as well as other cell types) were plated to confluency in 96-well plates. Cells were exposed to the combination of 10 μM Oligomyci...More data for this Ligand-Target Pair
