Compile Data Set for Download or QSAR
Report error Found 241 of affinity data for UniProtKB/TrEMBL: P11166
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010259(CHEMBL326463 | Acetic acid 10,10b-dihydroxy-6-{2-[...)
Affinity DataKd:  2.80E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010261(colforsinum | cid_47936 | colforsina | colforsine ...)
Affinity DataKd:  5.00E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010263(CHEMBL107985 | Acetic acid 10,10b-dihydroxy-6-(2-i...)
Affinity DataKd:  300nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010262(CHEMBL326703 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010265(CHEMBL327142 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  1.10E+3nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010266(CHEMBL324659 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  400nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010267([2-(4-Hydroxy-phenyl)-ethyl]-carbamic acid (3R,4aR...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010268(CHEMBL91909 | (2-Amino-ethyl)-carbamic acid (3R,4a...)
Affinity DataKd:  2.80E+4nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010264(CHEMBL110686 | (2-Isothiocyanato-ethyl)-carbamic a...)
Affinity DataKd:  500nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010273(CHEMBL111738 | {7-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  100nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010271(CHEMBL111425 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  800nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010274(CHEMBL328561 | Acetic acid (3R,4aR,5S,6S,6aS,10S,1...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010270(CHEMBL111514 | Acetic acid 6-[2-(2-bromo-acetylami...)
Affinity DataKd:  1.70E+4nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010260(CHEMBL107566 | [2-(2-Bromo-acetylamino)-ethyl]-car...)
Affinity DataKd:  1.30E+3nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010272(CHEMBL322952 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010275(CHEMBL324463 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010269(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Affinity DataKd:  240nMAssay Description:Inhibition of [125I]7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50622895(CHEMBL5396476)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50622896(CHEMBL5415555)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50622897(CHEMBL3895916)
Affinity DataKd:  2.60E+3nMAssay Description:Binding affinity to GLUT1 (unknown origin) assessed as dissociation constant at 800 uM by MST assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155671(CHEMBL3780239)
Affinity DataIC50: 1nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50514308(CHEMBL4448899)
Affinity DataIC50: 2nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as glucose uptake by measuring ATP incubated for 15 mins by CellTiter-Glo Luminescent Cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152749(CHEMBL3781913)
Affinity DataIC50: 4nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155656(CHEMBL3781331)
Affinity DataIC50: 5nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152824(CHEMBL3781548)
Affinity DataIC50: 7nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155715(CHEMBL3781149)
Affinity DataIC50: 7nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155751(CHEMBL3780460)
Affinity DataIC50: 8nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155585(CHEMBL3780372)
Affinity DataIC50: 9nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152826(CHEMBL3781347)
Affinity DataIC50: 10nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155673(CHEMBL3780972)
Affinity DataIC50: 10nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152743(CHEMBL3781308)
Affinity DataIC50: 14nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155746(CHEMBL3781151)
Affinity DataIC50: 17nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155747(CHEMBL3781194)
Affinity DataIC50: 17nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155670(CHEMBL3780144)
Affinity DataIC50: 20nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155714(CHEMBL3781157)
Affinity DataIC50: 25nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152776(CHEMBL3780785)
Affinity DataIC50: 27nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155753(CHEMBL3780470)
Affinity DataIC50: 30nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155677(CHEMBL3780765)
Affinity DataIC50: 33nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152827(CHEMBL3781741)
Affinity DataIC50: 35nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM453265(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-7,8-dih...)
Affinity DataIC50: 36nMAssay Description:Inhibition of GLUT1 in human wild-type DLD1 cells assessed as reduction in ATP level measured after 90 mins by Celltiter-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM453246(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-5,7-dih...)
Affinity DataIC50: 37nMAssay Description:Inhibition of GLUT1 in human wild-type DLD1 cells assessed as reduction in ATP level measured after 90 mins by Celltiter-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155680(CHEMBL3780717)
Affinity DataIC50: 39nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155752(CHEMBL3780527)
Affinity DataIC50: 40nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM453264(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-7,8-dih...)
Affinity DataIC50: 48nMAssay Description:Inhibition of GLUT1 in human wild-type DLD1 cells assessed as reduction in ATP level measured after 90 mins by Celltiter-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152774(CHEMBL3781384)
Affinity DataIC50: 49nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152825(CHEMBL3780235)
Affinity DataIC50: 50nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50155745(CHEMBL3780043)
Affinity DataIC50: 50nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50514308(CHEMBL4448899)
Affinity DataIC50: 50nMAssay Description:Inhibition of GLUT1 in human wild-type DLD1 cells assessed as reduction in ATP level measured after 90 mins by Celltiter-glo luminescent assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/11/2021
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM50152823(CHEMBL3780054)
Affinity DataIC50: 53nMAssay Description:Inhibition of human GLUT1 expressed in DLD1 cells assessed as ATP production co-incubated with 100 mM glucose for 16 hrs by CellTiter-Glo assay in pr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/2/2017
Entry Details Article
PubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Human)
Food and Drug Administration

Curated by ChEMBL
LigandPNGBDBM453216(2-(3-(4-((4-(1H-pyrazol-4-yl)phenyl)amino)-6-isobu...)
Affinity DataIC50: 55nMAssay Description:HT1080 cells (as well as other cell types) were plated to confluency in 96-well plates. Cells were exposed to the combination of 10 μM Oligomyci...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2021
Entry Details
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