Compile Data Set for Download or QSAR
Report error Found 60 of affinity data for UniProtKB/TrEMBL: P11021
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32370(adenosine-derived inhibitor (Grp78), 2 | adenosine...)
Affinity DataKd:  6.80E+3nM Kon: >1M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617289(CHEMBL5431926)
Affinity DataKd:  334nMAssay Description:Binding affinity to HspA5 (unknown origin) assessed as dissociation constant by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32381(adenosine-derived inhibitor (Grp78), 14 | adenosin...)
Affinity DataKd:  60nM Kon:  0.0400M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataKd:  80nM Kon:  0.0900M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32377(adenosine-derived inhibitor (Grp78), 12 | adenosin...)
Affinity DataKd:  770nM Kon:  0.300M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32376(adenosine-derived inhibitor (Grp78), 11 | adenosin...)
Affinity DataKd:  250nM Kon:  0.400M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM82129((2R,3R,4S,5R)-2-{6-Amino-8-[(quinolin-2-ylmethyl)a...)
Affinity DataKd:  2.41E+3nM Kon:  0.400M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32375(adenosine-derived inhibitor (Grp78), 9 | adenosine...)
Affinity DataKd:  230nM Kon:  0.200M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM82128(2-[(2R,3S,4R,5R)-5-(6-Amino-8-methylaminopurin-9-y...)
Affinity DataKd:  1.24E+4nM Kon: >1M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM82124(adenosine-derived inhibitor (Grp78), 1)
Affinity DataKd:  2.17E+3nM Kon:  0.00500M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32371(adenosine-derived inhibitor (Grp78), 3 | adenosine...)
Affinity DataKd:  7.46E+3nM Kon: >1M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM82125((2R,3R,4S,5R)-2-(6-Amino-8-methylaminopurin-9-yl)-...)
Affinity DataKd:  990nM Kon: >1M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM82127((2R,3R,4S,5R)-2-(6-Amino-8-methylaminopurin-9-yl)-...)
Affinity DataKd:  2.71E+3nM Kon: >1M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32373(adenosine-derived inhibitor (Grp78), 8 | adenosine...)
Affinity DataKd:  990nM Kon:  0.5M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM82126((2R,3R,4S,5R)-2-(6-Amino-8-methylaminopurin-9-yl)-...)
Affinity DataKd:  4.36E+3nM Kon: >1M-1s-1pH: 7.4 T: 2°CAssay Description:SPR measurements wereperformed on BIAcore T100 instrument (BIAcore GE Healthcare), at25 C on series S NTA chips (certified) according to provider'...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50088528(CHEMBL3576921)
Affinity DataIC50: 300nMAssay Description:Inhibition of 2-deoxyglucose-induced GRP78 (unknown origin) expression transfected in human HT1080 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617288(CHEMBL5410116)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617268(CHEMBL5415571)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617266(CHEMBL5418499)
Affinity DataIC50: 500nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617261(CHEMBL5414287)
Affinity DataIC50: 590nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617277(CHEMBL5419391)
Affinity DataIC50: 700nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM32378(adenosine-derived inhibitor (Grp78), 13 | adenosin...)
Affinity DataIC50: 800nMAssay Description:Inhibition of GRP78 (26 to 636 residues) (unknown origin) expressed in Escherichia coli BL21 DE3 cells pre-incubated for 10 mins before FITC-NRLLLTG ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617276(CHEMBL5403845)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617282(CHEMBL5425293)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617273(CHEMBL5409255)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617258(CHEMBL5424525)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617267(CHEMBL5410567)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617258(CHEMBL5424525)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of FAM-labeled NRLLLTG binding from HspA5 (unknown origin) in presence of ATP by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617271(CHEMBL5407447)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617260(CHEMBL5433282)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617275(CHEMBL5437667)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617257(CHEMBL5308000)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of FAM-labeled NRLLLTG binding from HspA5 (unknown origin) in presence of ATP by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617274(CHEMBL5422252)
Affinity DataIC50: 7.50E+3nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM31712(SMR000058356 | MLS000028433 | cid_3598 | HEXACHLOR...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of GRP78 (26 to 636 residues) (unknown origin) expressed in Escherichia coli BL21 DE3 cells pre-incubated for 10 mins before FITC-NRLLLTG ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM31712(SMR000058356 | MLS000028433 | cid_3598 | HEXACHLOR...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of GRP78 (26 to 636 residues) (unknown origin) expressed in Escherichia coli BL21 DE3 cells pre-incubated for 10 mins before FITC-NRLLLTG ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM31712(SMR000058356 | MLS000028433 | cid_3598 | HEXACHLOR...)
Affinity DataIC50: 9.10E+3nMAssay Description:Inhibition of GRP78 (26 to 636 residues) (unknown origin) expressed in Escherichia coli BL21 DE3 cells pre-incubated for 10 mins before FITC-NRLLLTG ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617272(CHEMBL5435048)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617259(CHEMBL5422755)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617265(CHEMBL5408152)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617281(CHEMBL5429240)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617280(CHEMBL5397525)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617279(CHEMBL5421614)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617278(CHEMBL5410605)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617284(CHEMBL5434599)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617285(CHEMBL5412223)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617283(CHEMBL5395892)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617286(CHEMBL5435520)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617270(CHEMBL5403880)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617269(CHEMBL5405780)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetEndoplasmic reticulum chaperone BiP(Human)
Vernalis (R&D)

LigandPNGBDBM50617287(CHEMBL5410820)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of HspA5 (unknown origin) by FP assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed
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