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Report error Found 665 of affinity data for UniProtKB/TrEMBL: P05089
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50316603(2-(S)-amino-5-(2-aminoimidazol-1-yl)pentanoic acid...)
Affinity DataKd:  2.00E+3nMAssay Description:Inhibition of human recombinant full length arginase 1 expressed in Escherichia coli BL21(DE3) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350309(CHEMBL1812662)
Affinity DataKd:  880nMAssay Description:Binding affinity to human arginase 1 using L-arginine as substrate by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350310(CHEMBL1812663)
Affinity DataKd:  3.40E+4nMAssay Description:Binding affinity to human arginase 1 using L-arginine as substrate by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  5nMAssay Description:Binding affinity to human arginase 1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  18nMAssay Description:Binding affinity to human arginase 1 using L-arginine as substrate by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50354832(CHEMBL1834160)
Affinity DataKd:  6.00E+4nMAssay Description:Displacement of [14C-guanidino]-L-arginine from human recombinant full length arginase 1 expressed in Escherichia coli BL21(DE3) by fixed point assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  5nMAssay Description:Binding affinity to wild type human Arg I using L-arginine as substrate by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataKd:  47nMAssay Description:Binding affinity to arginase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  5nMAssay Description:Binding affinity to human Arg1 at pH 8.5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561034(CHEMBL4244287)
Affinity DataKd:  270nMAssay Description:Binding affinity to human Arg1 at pH 8.5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50230418(N-OMEGA-HYDROXY-L-ARGININE | Nomega-hydroxy-L-argi...)
Affinity DataKd:  3.60E+3nMAssay Description:Binding affinity to human Arg1 at pH 8.5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataKd:  517nMAssay Description:Binding affinity to human Arg1 at pH 8.5More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577458(CHEMBL4858437)
Affinity DataEC50:  3.40E+3nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577473(CHEMBL4871410)
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577474(CHEMBL4876150)
Affinity DataEC50:  6.30E+3nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577475(CHEMBL4855923)
Affinity DataEC50:  1.10E+4nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577476(CHEMBL4852406)
Affinity DataEC50:  1.40E+4nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577477(CHEMBL4868283)
Affinity DataEC50:  2.80E+3nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577478(CHEMBL4872801)
Affinity DataEC50:  4.20E+3nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577479(CHEMBL4862990)
Affinity DataEC50:  1.60E+4nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561036(CHEMBL4778978)
Affinity DataEC50:  6.90E+3nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577480(CHEMBL4862982)
Affinity DataEC50:  2.80E+4nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561035(CHEMBL4763578)
Affinity DataEC50:  2.00E+4nMAssay Description:Inhibition of human ARG1 in HEK293 cells by cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50608140(CHEMBL1230498)
Affinity DataKd:  6.00E+4nMAssay Description:Binding affinity to human Arg IMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350309(CHEMBL1812662)
Affinity DataKd:  880nMAssay Description:Binding affinity to human Arg I assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350310(CHEMBL1812663)
Affinity DataKd:  3.40E+4nMAssay Description:Binding affinity to human Arg I assessed as inhibition constant by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataKd:  5nMAssay Description:Inhibition of human Arginase I in human myeloid-derived suppressor cells using L-arginine as substrate assessed as L-ornithine product formation by m...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataKd:  50nMAssay Description:Inhibition of human Arginase I assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561047(CHEMBL4764455)
Affinity DataIC50: 0.100nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561040(CHEMBL4754637)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561042(CHEMBL4748950)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561049(CHEMBL4793482)
Affinity DataIC50: 1nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561051(CHEMBL4749434)
Affinity DataIC50: 1nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561052(CHEMBL4755855)
Affinity DataIC50: 1nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561053(CHEMBL4750602)
Affinity DataIC50: 1nMAssay Description:Inhibition of human Arg1More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561042(CHEMBL4748950)
Affinity DataIC50: 1nMAssay Description:Inhibition of human recombinant ARG1 expressed in Escherichia coli using thioarginine as a substrate preincubated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50595723(CHEMBL5193387)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human ARG1 expressed in Escherichia coli using L-arginine hydrochloride as substrate incubated for 1 hr by colorimetric ass...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50595727(CHEMBL5184299)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human ARG1 expressed in Escherichia coli using L-arginine hydrochloride as substrate incubated for 1 hr by colorimetric ass...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50595729(CHEMBL5176739)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human ARG1 expressed in Escherichia coli using L-arginine hydrochloride as substrate incubated for 1 hr by colorimetric ass...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50595730(CHEMBL5171566)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human ARG1 expressed in Escherichia coli using L-arginine hydrochloride as substrate incubated for 1 hr by colorimetric ass...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50595731(CHEMBL5170454)
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant human ARG1 expressed in Escherichia coli using L-arginine hydrochloride as substrate incubated for 1 hr by colorimetric ass...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50509011(CHEMBL4538713)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human recombinant arginase 1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in urea production using L-arginine as subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561041(CHEMBL4791224)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50579614(CHEMBL4871970)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50577469(CHEMBL4850213)
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant ARG1 expressed in Escherichia coli using thioarginine as a substrate preincubated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50579610(CHEMBL4873520)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of ARG1 (unknown origin) assessed as reduction in thio-ornithine production using thioarginine as substrate by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50509016(CHEMBL4450972)
Affinity DataIC50: 2.5nMAssay Description:Inhibition of human recombinant arginase 1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in urea production using L-arginine as subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50509014(CHEMBL4557975)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human recombinant arginase 1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in urea production using L-arginine as subs...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561039(CHEMBL4749355 | US11420984, Example 23)
Affinity DataIC50: 3nMAssay Description:Inhibition of human Arg1 by TOGA assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetArginase-1(Human)
University of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50561035(CHEMBL4763578)
Affinity DataIC50: 3nMAssay Description:Inhibition of human recombinant ARG1 expressed in Escherichia coli using thioarginine as a substrate preincubated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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