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Report error Found 9776 for UniProtKB: P03372
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataEC50:  622nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assay was performed by using 96-well microtiterplates containing ER, 17beta-estradiol, and the test compound to be tested and SPA...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19918(5-hydroxy-7-methoxy-3-(4-methoxyphenyl)-3,4-dihydr...)
Affinity DatapH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19919(3-arylquinazolinone, 1aak | 7-hydroxy-3-(4-hydroxy...)
Affinity DatapH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM20607((2-{4-[(1Z)-1,2-diphenylbut-1-en-1-yl]phenoxy}ethy...)
Affinity DataEC50:  622nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assay was performed by using 96-well microtiterplates containing ER, 17beta-estradiol, and the test compound to be tested and SPA...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19922(5,7-dihydroxy-3-(4-hydroxyphenyl)-8-iodo-3,4-dihyd...)
Affinity DataEC50:  8.32E+3nMpH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19923(5,7-dihydroxy-3-(4-hydroxyphenyl)-6,8-diiodo-3,4-d...)
Affinity DatapH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19925(5,7-dihydroxy-3-(4-hydroxyphenyl)-6-iodo-3,4-dihyd...)
Affinity DatapH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19935(5-hydroxy-3-(4-hydroxyphenyl)-7-methoxy-2-sulfanyl...)
Affinity DatapH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19937(2-chloro-5,7-dihydroxy-3-(4-hydroxyphenyl)-3,4-dih...)
Affinity DatapH: 8.0 T: 2°CAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19939(7-hydroxy-3-(4-hydroxyphenyl)-2-methyl-3,4-dihydro...)
Affinity DataAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19941(5-ethoxy-7-hydroxy-3-(4-hydroxyphenyl)-3,4-dihydro...)
Affinity DataAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19919(3-arylquinazolinone, 1aak | 7-hydroxy-3-(4-hydroxy...)
Affinity DataAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19945(7-hydroxy-3-(4-hydroxyphenyl)-4-oxo-3,4-dihydroqui...)
Affinity DataAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19946(7-hydroxy-3-(4-hydroxyphenyl)-4-oxo-3,4-dihydroqui...)
Affinity DataAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19948(5-ethenyl-7-hydroxy-3-(4-hydroxyphenyl)-3,4-dihydr...)
Affinity DataEC50:  4.62E+3nMAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19959(5-(acetyloxy)-3-[4-(acetyloxy)phenyl]-4-sulfanylid...)
Affinity DataAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19960(7-methoxy-3-(4-methoxyphenyl)-4-sulfanylidene-3,4-...)
Affinity DataAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM19961(5-hydroxy-7-methoxy-3-(4-methoxyphenyl)-3,4-dihydr...)
Affinity DataAssay Description:Ligand binding was determined using a scintillation proximity assay with streptavidin-coated SPA beads (Amersham) and biotinylated receptor. Receptor...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM22430((5Z)-6-{4-[2-(dimethylamino)ethoxy]phenyl}-6-(4-hy...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Binding affinity was measured by a scintillation proximity binding assay using [3H]4-OHT (for ERRgamma) or [3H]estradiol (for ERalpha) as radioligand...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM22431(4-[(1Z)-1-{4-[2-(dimethylamino)ethoxy]phenyl}-5-(m...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Binding affinity was measured by a scintillation proximity binding assay using [3H]4-OHT (for ERRgamma) or [3H]estradiol (for ERalpha) as radioligand...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM22432(4-[(1Z)-5-(dimethylamino)-1-{4-[2-(dimethylamino)e...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Binding affinity was measured by a scintillation proximity binding assay using [3H]4-OHT (for ERRgamma) or [3H]estradiol (for ERalpha) as radioligand...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM22433(N-[(4Z)-5-{4-[2-(dimethylamino)ethoxy]phenyl}-5-(4...)
Affinity DatapH: 7.4 T: 2°CAssay Description:Binding affinity was measured by a scintillation proximity binding assay using [3H]4-OHT (for ERRgamma) or [3H]estradiol (for ERalpha) as radioligand...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40483(cid_649431 | 3-[6-(4-chlorophenyl)-2-methoxypyridi...)
Affinity DataEC50:  48.7nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM39937(cid_665299 | 2-[2-(5-bromo-2-furanyl)-3H-benzimida...)
Affinity DataEC50:  1.41nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM39953(4-oxo-4-thiophen-2-ylbutanoic acid [2-(2-furanylme...)
Affinity DataEC50:  4.25nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42022(MLS000053529 | 2-[2-furanyl(oxo)methyl]-N-[2-(4-mo...)
Affinity DataEC50:  367nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40022(SMR000020900 | cid_3239187 | N-[2-[[2-(cyclopropyl...)
Affinity DataEC50:  24.3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42023(2,3-di-2-furyl-6-{[4-(2-methoxyphenyl)piperazin-1-...)
Affinity DataEC50:  15.4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40047(MLS000087249 | SMR000023472 | N-(4-methoxybenzyl)-...)
Affinity DataEC50:  9.68nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42024(N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-...)
Affinity DataEC50:  3.17nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40537(4-[2,5-bis(oxidanylidene)pyrrolidin-1-yl]-N-(3-eth...)
Affinity DataEC50: >1.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40990(SMR000108537 | cid_960705 | 2-(3,5-dimethylphenoxy...)
Affinity DataEC50: >1.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40544(MLS000028696 | 6ALPHA-HYDROXYESTRADIOL | SMR000058...)
Affinity DataEC50:  36.6nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40694(cid_2434862 | [2-[4-(furan-2-ylcarbonyl)piperazin-...)
Affinity DataEC50:  33.9nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40261(SMR000154728 | N-[(2-furanylmethylamino)-oxomethyl...)
Affinity DataEC50:  44.7nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM50303804(cid_3136844 | CHEMBL583543 | (3aS,4R,9bR)-4-(6-bro...)
Affinity DataEC50:  782nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42025(SMR000176871 | cid_6836350 | 4-Methoxy-benzoic aci...)
Affinity DataEC50:  1.43E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42026(SMR000207609 | (3aS,4R,9bR)-6,8-dimethyl-4-[4-(mor...)
Affinity DataEC50:  44.4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42027(cid_3136304 | SMR000230829 | MLS000704836 | 4-{8-[...)
Affinity DataEC50:  3.88E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42028(MLS000705473 | cid_15945793 | SMR000230901 | (3aS,...)
Affinity DataEC50:  1.01E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42029(cid_2868331 | UNM000011059201 | 4-(1-cyclohex-3-en...)
Affinity DataEC50:  4.76nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM50303803(cid_5322399 | cid_3136849 | CHEMBL569766 | 1-((3aS...)
Affinity DataEC50:  48.7nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42030(UNM000011064401 | cid_2865996 | 1-[4-(3-nitropheny...)
Affinity DataEC50: >1.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42031(cid_2854262 | UNM000011065601 | 4-(3-nitrophenyl)-...)
Affinity DataEC50:  276nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42032(UNM000011066901 | cid_2873342 | 4-(4-chlorophenyl)...)
Affinity DataEC50:  1.26E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42033(cid_2900725 | 4-(4-acetyloxyphenyl)-9-nitro-3a,4,5...)
Affinity DataEC50: >1.00E+4nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42034(4-(3-nitro-4-oxidanyl-phenyl)-3a,4,5,9b-tetrahydro...)
Affinity DataEC50:  557nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42035(cid_5322407 | UNM000011068501 | 4-[(3aR,4S,9bS)-8-...)
Affinity DataEC50:  3.60E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM42036(UNM000011068701 | cid_5322461 | (3aS,4R,9bR)-8-bro...)
Affinity DataEC50:  2.49E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1X01 MH077627-01 Assay for Ligands of GPR30 and Classical Estrogen Receptors PI: Eric Prossni...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
TargetEstrogen receptor(Human)
Novartis Pharmaceuticals

LigandPNGBDBM40479(3-(2-phenylimidazol-1-yl)propanoic acid | MLS00007...)
Affinity DataEC50:  1.25E+4nMAssay Description:NIH Molecular Libraries Screening Centers Network [MLSCN] Emory Chemical Biology Discovery Center in MLSCN Assay provider: John A. Katzenellenbogen, ...More data for this Ligand-Target Pair
In DepthDetails
PCBioAssay
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