Compile Data Set for Download or QSAR
Report error Found 26 of affinity data for UniProtKB/TrEMBL: P03354
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521553(Isopropyl ((((2R,3 S,4R,5R)-5-(4-aminopyrrolo[2,1-...)
Affinity DataEC50:  1.30E+3nMAssay Description:The HeLa-derived cells containing the stable RSV replicon were cultured in DMEM containing 4500 mg/L D-glucose, L-glutamine, and 110 mg/L sodium pyru...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521552(US11149049, No. 10)
Affinity DataEC50:  170nMAssay Description:The HeLa-derived cells containing the stable RSV replicon were cultured in DMEM containing 4500 mg/L D-glucose, L-glutamine, and 110 mg/L sodium pyru...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521551(2-Ethylbutyl ((((2S,3S,4R,5R)-5-(4-aminopyrrolo[2,...)
Affinity DataEC50:  18nMAssay Description:The HeLa-derived cells containing the stable RSV replicon were cultured in DMEM containing 4500 mg/L D-glucose, L-glutamine, and 110 mg/L sodium pyru...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521550(Neopentyl ((((2S,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f...)
Affinity DataEC50:  30nMAssay Description:The HeLa-derived cells containing the stable RSV replicon were cultured in DMEM containing 4500 mg/L D-glucose, L-glutamine, and 110 mg/L sodium pyru...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521549(Diisopentyl ((((2S,3S,4R,5R)-5-(4-aminopyrrolo[2,1...)
Affinity DataEC50:  30nMAssay Description:The HeLa-derived cells containing the stable RSV replicon were cultured in DMEM containing 4500 mg/L D-glucose, L-glutamine, and 110 mg/L sodium pyru...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521548(Isopropyl ((((2S,3 S,4R,5R)-5-(4-aminopyrrolo[2, l...)
Affinity DataEC50:  20nMAssay Description:The HeLa-derived cells containing the stable RSV replicon were cultured in DMEM containing 4500 mg/L D-glucose, L-glutamine, and 110 mg/L sodium pyru...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521547(Isopropyl ((((2S,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f...)
Affinity DataEC50:  2.74E+3nMAssay Description:The HeLa-derived cells containing the stable RSV replicon were cultured in DMEM containing 4500 mg/L D-glucose, L-glutamine, and 110 mg/L sodium pyru...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521546(US11149049, No. C1)
Affinity DataEC50:  20nMAssay Description:The HeLa-derived cells containing the stable RSV replicon were cultured in DMEM containing 4500 mg/L D-glucose, L-glutamine, and 110 mg/L sodium pyru...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521557(((2R,3S,4R,5R)-5-(4-Aminopyrrolo[2,1-f][1,2,4]tria...)
Affinity DataIC50: 30nMAssay Description:Standard RSV polymerase assays were conducted in the presence of 3 μL extract of RSV-infected cells in a reaction buffer containing 50 mM tris-a...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521555(((2S,3S,4R,5R)-5-(4-Aminopyrrolo[2,1-f][1,2,4]tria...)
Affinity DataIC50: 30nMAssay Description:Standard RSV polymerase assays were conducted in the presence of 3 μL extract of RSV-infected cells in a reaction buffer containing 50 mM tris-a...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50236025(CHEMBL2016761 | US11149049, No. C2 | US20240140975...)
Affinity DataIC50: 120nMAssay Description:Standard RSV polymerase assays were conducted in the presence of 3 μL extract of RSV-infected cells in a reaction buffer containing 50 mM tris-a...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065793(8-Hydroxy-2-[(E)-2-(3,4,5-trihydroxy-phenyl)-vinyl...)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065796(2-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065788(2-(3-carboxy-4-hydroxystyryl)-8-hydroxyquinoline-7...)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM521556(((2R,3S,4R,5R)-5-(4-Aminopyrrolo[2,1-f][1,2,4]tria...)
Affinity DataIC50: 1.00E+4nMAssay Description:Standard RSV polymerase assays were conducted in the presence of 3 μL extract of RSV-infected cells in a reaction buffer containing 50 mM tris-a...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50087421(8-hydroxy-2-styrylquinoline-7-carboxylic acid | 8-...)
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50087435(8-hydroxy-2-(4-hydroxystyryl)quinoline-7-carboxyli...)
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065786(2-[2-(3,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065790(2-[2-(2,4-Dihydroxy-phenyl)-vinyl]-8-hydroxy-quino...)
Affinity DataIC50: 3.83E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065787(4-(2-(8-hydroxyquinolin-2-yl)vinyl)benzene-1,2-dio...)
Affinity DataIC50: 6.51E+4nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065789(2-Styryl-quinolin-8-ol | 2-Styrylquinolin-8-ol | 2...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065800((E)-3-(3,4-Dihydroxy-phenyl)-acrylic acid 2-methyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065802(Acetic acid 2-acetoxy-5-[2-(8-acetoxy-quinolin-2-y...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065791(4-[(E)-2-(8-Amino-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065798(Acetic acid 2-((E)-styryl)-quinolin-8-yl ester | A...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetRous sarcoma virus integrase(RSV-Pr-C)
Janssen Biopharma

US Patent
LigandPNGBDBM50065784(4-[(E)-2-(8-Nitro-quinolin-2-yl)-vinyl]-benzene-1,...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of rous sarcoma virus (RSV) Integrase.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed