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Report error Found 138 of affinity data for UniProtKB/TrEMBL: P00761
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50044092(spumigin E)
Affinity DataIC50: 100nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50286441(Ac-LLR-CHO | Ac-Leu-Leu-Arg-H | (S)-2-((S)-2-Acety...)
Affinity DataIC50: 200nMAssay Description:Inhibition of pig pancreas trypsin type IX-SMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50044094(CHEMBL3325623)
Affinity DataIC50: 350nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50286441(Ac-LLR-CHO | Ac-Leu-Leu-Arg-H | (S)-2-((S)-2-Acety...)
Affinity DataIC50: 500nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50041802(CHEMBL46469 | 1,8-dihydroxyanthrone | 1,8-dihydrox...)
Affinity DataIC50: 1.26E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191635(US9182402, 8)
Affinity DataIC50: 1.71E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191638(US9182402, 11)
Affinity DataIC50: 2.00E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50013876(N-Methyl-D-aspartate | N-Methyl aspartic acid | CH...)
Affinity DataIC50: 2.42E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191639(US9182402, 12)
Affinity DataIC50: 3.50E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM123129(CID236790 | 1-(3-nitro-phenyl)-pyrrole-2,5-dione (...)
Affinity DataIC50: 3.88E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085340(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(4-isopro...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191630(US9182402, 3)
Affinity DataIC50: 7.63E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191637(US9182402, 10)
Affinity DataIC50: 7.72E+3nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191633(US9182402, 6)
Affinity DataIC50: 1.02E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191634(US9182402, 7)
Affinity DataIC50: 1.31E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50069104(CHEMBL1449583 | US9182402, 4)
Affinity DataIC50: 1.96E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191632(US9182402, 2)
Affinity DataIC50: 2.00E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM81467(CHEMBL1085765 | NSC_4034 | CAS_569-65-3 | Meclizin...)
Affinity DataIC50: 2.00E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191636(US9182402, 9)
Affinity DataIC50: 2.09E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085346(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(3,4-dich...)
Affinity DataIC50: 2.80E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085354(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(4-triflu...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM191631(US9182402, 5)
Affinity DataIC50: 3.12E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50007260(2,6-di-tert-butyl-4-(2-(3,5-di-tert-butyl-4-hydrox...)
Affinity DataIC50: 3.35E+4nMAssay Description:To identify novel inhibitors of hepsin, the Chembridge DIVERSet 10,000 compound high-diversity library was screened using an assay based on the cleav...More data for this Ligand-Target Pair
In DepthDetails
US Patent

TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085356(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(2-methox...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085341(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(3-triflu...)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085364(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(3-chloro...)
Affinity DataIC50: 4.40E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50044093(CHEMBL3325624)
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of pig pancreas trypsin type IX-S using Boc-Gln-Ala-Arg-MCA substrate by 7-amino-4-methylcoumarin release based spectrofluorometryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085361(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(3-hydrox...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085343(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(2-chloro...)
Affinity DataIC50: 8.50E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085352(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(2,3-dich...)
Affinity DataIC50: 9.70E+4nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085353(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-(4-ethyl-...)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269534((Z,Z,Z)-8,11,14-Eicosatrienoic acid | Dihomo-gamma...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269540(6-(8'Z,11'Z-heptadecadienyl)-salicylicacid | CHEMB...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50259930(6-[10'(Z)-heptade-cenyljsalicylic acid | 6-(10'Z-h...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50242188(6-{8(Z)-pentadecenyl}salicylic acid | Anacardic ac...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50242349(5,8,11,14,17-EICOSAPENTAENOIC ACID | 5Z,8Z,11Z,14Z...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM22319([1-14C]Arachidonic acid | (5Z,8Z,11Z,14Z)-icosa-5,...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269535(all-cis-icosa-11,14,17-trienoic acid | (11Z,14Z,17...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269533(cis-11,14-eicosadienoicacid | CHEMBL464983)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269532((6Z,9Z,12Z)-octadeca-6,9,12-trienoic acid | gamma-...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50240347((Z,Z,Z)-9,12,15-octadecatrienoic acid | cis,cis,ci...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM22231(CHEMBL267476 | (9Z,12Z)-octadeca-9,12-dienoic acid...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50150484(CHEMBL8659 | oleaic acid | Octadec-9-enoic acid | ...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269531((9Z)-hexadec-9-enoic acid | palmitoleic acid | (Z)...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50269530((9Z)-tetradec-9-enoic acid | myristoleic acid | ci...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of pig pancreatic trypsin after 15 minsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085363(N-Tosyl-L-phenylalanine chloromethyl ketone | CHEM...)
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085362(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-phenyl-ac...)
Affinity DataIC50: 2.10E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085339(((S)-1-Benzyl-3-chloro-2-oxo-propyl)-carbamic acid...)
Affinity DataIC50: 2.10E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085360(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-benzamide |...)
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetTrypsin(Pig)
University of Helsinki

Curated by ChEMBL
LigandPNGBDBM50085348(N-((S)-1-Benzyl-3-chloro-2-oxo-propyl)-3-p-tolyl-p...)
Affinity DataIC50: 2.60E+5nMAssay Description:Inhibitory activity against porcine pancreatic trypsin (TRP)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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