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Report error Found 188 for UniProtKB: O95263
LigandPNGBDBM50344013(trans-(3R,5S)-N-((6-aminopyridin-2-yl)methyl)-1-((...)
Affinity DataIC50: 0.120nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50594973(CHEMBL5169811)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PDE8B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50594973(CHEMBL5169811)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PDE8B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50594973(CHEMBL5169811)
Affinity DataIC50: 0.300nMAssay Description:Inhibition of PDE8B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails
PubMed
LigandPNGBDBM50344014(trans-(3R,5S)-1-((5-methyl-2-phenyloxazol-4-yl)met...)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390333(CHEMBL2070733)
Affinity DataIC50: 0.900nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344015(trans-(3S,5S)-5-ethyl-1-((5-methyl-2-phenyloxazol-...)
Affinity DataIC50: 0.955nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390334(CHEMBL2070735)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390332(CHEMBL2070732)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344019(trans-(3R,5R)-5-(methoxymethyl)-1-((5-methyl-2-phe...)
Affinity DataIC50: 1.96nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344020(trans-(3R,5R)-5-ethyl-1-((5-methyl-2-phenyloxazol-...)
Affinity DataIC50: 2.91nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344021(trans-(3R,5R)-5-(methoxymethyl)-1-((5-methyl-2-phe...)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390373(CHEMBL2070914)
Affinity DataIC50: 3.63nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344022(trans-(3S,5S)-5-(3-methyl-1,2,4-oxadiazol-5-yl)-1-...)
Affinity DataIC50: 3.86nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344023(trans-(3R,5R)-5-(3-methyl-1,2,4-oxadiazol-5-yl)-1-...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390335(CHEMBL2070736)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344024(trans-(3S,5S)-5-(methoxymethyl)-1-((5-methyl-2-phe...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344025(trans-(3R,5R)-5-(methoxymethyl)-1-((5-methyl-2-phe...)
Affinity DataIC50: 4.36nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344026(trans-(3R,5R)-N-((6-aminopyridin-2-yl)methyl)-5-et...)
Affinity DataIC50: 4.42nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344016(2-((5-methyl-2-phenyloxazol-4-yl)methyl)-N-((6-met...)
Affinity DataIC50: 5nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344018(trans-(3R,5R)-5-ethyl-1-((5-methyl-2-phenyloxazol-...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344027(trans-(3R,5R)-1-((5-methyl-2-phenyloxazol-4-yl)met...)
Affinity DataIC50: 6nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390366(CHEMBL2070935)
Affinity DataIC50: 6.79nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390324(CHEMBL2070604)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344028(trans-(3R,5R)-1-((5-methyl-2-phenyloxazol-4-yl)met...)
Affinity DataIC50: 7nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344029(trans-(3R,5R)-5-ethyl-1-((5-methyl-2-phenyloxazol-...)
Affinity DataIC50: 7.30nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390313(CHEMBL2070595)
Affinity DataIC50: 10nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390352(CHEMBL2070901)
Affinity DataIC50: 12.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344030(trans-(3R,5R)-5-(methoxymethyl)-1-((5-methyl-2-(py...)
Affinity DataIC50: 13nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390367(CHEMBL2070907)
Affinity DataIC50: 13.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390308(CHEMBL2070592)
Affinity DataIC50: 14nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390309(CHEMBL2070591)
Affinity DataIC50: 14nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344031(trans-(3R,5R)-5-butyl-1-((5-methyl-2-phenyloxazol-...)
Affinity DataIC50: 15nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50272569(CHEMBL4128481)
Affinity DataIC50: 16nMAssay Description:Inhibition of full length recombinant human PDE8B using 3',5'-[3H]cAMP as substrate after 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344032(trans-(3R,5R)-N-((6-aminopyridin-2-yl)methyl)-5-et...)
Affinity DataIC50: 16.5nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390339(CHEMBL2070769)
Affinity DataIC50: 17.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390371(CHEMBL2070912)
Affinity DataIC50: 17.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390378(CHEMBL2070919)
Affinity DataIC50: 17.1nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390363(CHEMBL2070932)
Affinity DataIC50: 17.7nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390336(CHEMBL2070737)
Affinity DataIC50: 19nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344033(trans-(3R,5R)-5-ethyl-1-((5-methyl-2-phenyloxazol-...)
Affinity DataIC50: 19.6nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390364(CHEMBL2070933)
Affinity DataIC50: 21.4nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390343(CHEMBL2070773)
Affinity DataIC50: 21.6nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390329(CHEMBL2070729)
Affinity DataIC50: 23nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390338(CHEMBL2070734)
Affinity DataIC50: 23nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390320(CHEMBL2070600)
Affinity DataIC50: 25nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390375(CHEMBL2070916)
Affinity DataIC50: 25.5nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344034(trans-(3R,5R)-5-ethyl-1-((5-methyl-2-(pyrimidin-4-...)
Affinity DataIC50: 26nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50344035(trans-(3R,5R)-5-ethyl-1-((5-methyl-2-(pyrimidin-4-...)
Affinity DataIC50: 26.2nMAssay Description:Inhibition of PDE8BMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50390384(CHEMBL2070925)
Affinity DataIC50: 31.5nMAssay Description:Inhibition of PDE8B expressed in Sf9 insect cellsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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