Compile Data Set for Download or QSAR
Report error Found 20 of affinity data for UniProtKB/TrEMBL: O89017
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364367(CHEMBL1950283)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364353(CHEMBL1950109)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364366(CHEMBL1950282)
Affinity DataIC50: 8.10nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM228618(BDBM50364365 | US9345789, LI-2)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364368(CHEMBL1950284)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM36332(LI-1 | Legumain Inhibitor -1)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364356(CHEMBL1950112)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM36332(LI-1 | Legumain Inhibitor -1)
Affinity DataIC50: 11.5nMpH: 5.8 T: 2°CAssay Description:IC50 measurements and enzyme kinetics assays were performed on a Spectramax M5 fluorescent plate reader (Molecular Devices).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364358(CHEMBL1950273)
Affinity DataIC50: 17nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364354(CHEMBL1950110)
Affinity DataIC50: 141nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364355(CHEMBL1950111)
Affinity DataIC50: 148nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364360(CHEMBL1950275)
Affinity DataIC50: 167nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364357(CHEMBL1950272)
Affinity DataIC50: 198nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364363(CHEMBL1950278)
Affinity DataIC50: 267nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM70989(4-morpholin-4-yl-2,1,3-benzoxadiazol-7-amine | MLS...)
Affinity DataIC50: 301nMAssay Description:Inhibition of AEP in mouse kidney lysate using Cbz-Ala-Ala-Asn-AMC as substrate incubated for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails
PubMedPDB3D3D Structure (crystal)
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364359(CHEMBL1950274)
Affinity DataIC50: 638nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM36333(LI-0 | Legumain Inhibitor -0)
Affinity DataIC50: 704nMpH: 5.8 T: 2°CAssay Description:IC50 measurements and enzyme kinetics assays were performed on a Spectramax M5 fluorescent plate reader (Molecular Devices).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364364(CHEMBL1950279)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364362(CHEMBL1950277)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetLegumain(Mouse)
Stanford University School of Medicine

Curated by ChEMBL
LigandPNGBDBM50364361(CHEMBL1950276)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mouse recombinant legumain using Cbz-Ala-Ala-Asn-AMC as substrate measured every 30 secs for 2.5 hrs by fluorimetryMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed