Compile Data Set for Download or QSAR
Report error Found 16 of affinity data for UniProtKB/TrEMBL: O88506
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267897(CHEMBL4092297)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267911(CHEMBL4096245)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267896(CHEMBL4064614)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267893(CHEMBL4086083)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267909(CHEMBL4094766)
Affinity DataIC50: 6.90E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267895(CHEMBL4084562)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267916(TCMDC-125004 | CHEMBL531227)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267913(GNF-Pf-3043 | CHEMBL602783)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267901(CHEMBL4087066)
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267917(CHEMBL4080499)
Affinity DataIC50: 2.11E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267915(CHEMBL4088361)
Affinity DataIC50: 2.82E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267921(CHEMBL4095711)
Affinity DataIC50: 3.56E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267910(CHEMBL4074261)
Affinity DataIC50: 3.69E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267914(CHEMBL4067097)
Affinity DataIC50: 4.90E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267912(CHEMBL4069800)
Affinity DataIC50: 5.35E+4nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSTE20/SPS1-related proline-alanine-rich protein kinase(Rat)
Tokyo Medical and Dental University (Tmdu)

Curated by ChEMBL
LigandPNGBDBM50267894(CHEMBL4102505)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of TAMRA-labelled WNK4 binding to recombinant rat C-terminal GST-fused SPAK (452 to 553 residues) expressed in Escherichia coli BL21 measu...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed