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Report error Found 10 of affinity data for UniProtKB/TrEMBL: O55143
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631117(Arm-210 | Rycal dmd | S48168 | ARM210 | S-48168 | ...)
Affinity DataEC50:  3.43E+4nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631111(CHEMBL5437537)
Affinity DataEC50:  2.20E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631112(CHEMBL5398491)
Affinity DataEC50:  8.60E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631113(CHEMBL5413930)
Affinity DataEC50:  7.60E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631118(CHEMBL5409315)
Affinity DataEC50: >1.00E+6nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631114(CHEMBL5435124)
Affinity DataEC50:  9.20E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631115(CHEMBL5426069)
Affinity DataEC50:  1.50E+3nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631116(CHEMBL5409619)
Affinity DataEC50:  1.09E+4nMAssay Description:Activation of SERCA2a in mouse HL-1 cells assessed as increase in caffeine-induced calcium release incubated for 2 hrs by FLIPR Calcium 6 dye based c...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50631114(CHEMBL5435124)
Affinity DataEC50:  383nMAssay Description:Activation of SERCA2a in C57BL/6N mouse sarcoplasmic reticulum assessed as increase in calcium release measured for 10 mins in presence of ATP by NAD...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 2(Mouse)
Max Planck Institute for Multidisciplinary Sciences

Curated by ChEMBL
LigandPNGBDBM50410532(4-NONYLPHENOL)
Affinity DataIC50: 350nMAssay Description:Inhibition of SERCA2b in mouse testicular microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed