Compile Data Set for Download or QSAR
Report error Found 9 of affinity data for UniProtKB/TrEMBL: O14983
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165369(12-(4-Amino-4-carboxy-butyrylamino)-dodecanoic aci...)
Affinity DataIC50: 1.20nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165368(Dodecanedioic acid mono-((2S,3aR,4S,6S,6aR,7S,9bS)...)
Affinity DataIC50: 2.08nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
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PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165366(Pentanedioic acid mono-((2S,3aR,4S,6S,6aR,7S,9bS)-...)
Affinity DataIC50: 19.8nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50165367(Octanoic acid (2S,3aR,4S,6S,6aR,7S,9bS)-6-acetoxy-...)
Affinity DataIC50: 9.04E+3nMAssay Description:Inhibitory activity against sarco- endoplasmic reticulum calcium-ATPaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM25524(CHEMBL13045 | 17,18-dimethoxy-21-methyl-5,7-dioxa-...)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of SERCA1a (unknown origin) incubated for 10 mins by enzyme-coupled methodMore data for this Ligand-Target Pair
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PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50035612(OCTANOIC ACID [3S-[3ALPHA, 3ABETA, 4ALPHA, 6BETA, ...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of SERCA1a (unknown origin) ATPase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50453612(CHEMBL4216774)
Affinity DataKi:  17nMAssay Description:Inhibition of SERCA1a (unknown origin) ATPase activityMore data for this Ligand-Target Pair
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PubMedPDB3D3D Structure (crystal)
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50453611(CHEMBL4207081)
Affinity DataKi:  19nMAssay Description:Inhibition of SERCA1a (unknown origin) ATPase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSarcoplasmic/endoplasmic reticulum calcium ATPase 1(Human)
Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50453613(CHEBI:22450 | Alpha-Cyclopiazonic Acid | Cyclopiaz...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of SERCA1a (unknown origin) ATPase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed