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Report error Found 11 of affinity data for UniProtKB/TrEMBL: O08966
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50367247(Quinamm | Quinsan | QUININE | cid_3034034)
Affinity DataIC50: 280nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataIC50: 540nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50403559(Brumetadina | CIMETIDINE)
Affinity DataIC50: 590nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM39344(PROCAINAMIDE | PROCAINAMIDE HYDROCHLORIDE | 4-azan...)
Affinity DataIC50: 3.90E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50026220(2-hydroxy-N,N,N-trimethylethanaminium | CHEMBL920 ...)
Affinity DataIC50: 5.50E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50420177(NICOTINYL METHYLAMIDE)
Affinity DataIC50: 7.34E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake (MPP+: 1 uM) in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM18512(cid_4993 | CHEMBL36 | 5-(4-chlorophenyl)-6-ethylpy...)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of mouse Oct1 transfected in HEK293 cells assessed as uptake of [14C]-TEA preincubated for 15 mins by liquid scintillation counting analys...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50416487(CHEMBL1236196 | TETRABUTYLAMMONIUM)
Affinity DataKi:  7.30E+3nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50420179(CHEMBL2074857)
Affinity DataKi:  1.98E+4nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataKi:  1.28E+5nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSolute carrier family 22 member 1(Mouse)
Kyushu University

Curated by ChEMBL
LigandPNGBDBM50079455(CHEMBL46486 | tetramethylammonium)
Affinity DataKi:  2.04E+6nMAssay Description:TP_TRANSPORTER: inhibition of MPP+ uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
In DepthDetails
PubMed